Structure-based design and synthesis of small molecule protein-tyrosine phosphatase 1B inhibitors

Bioorganic and Medicinal Chemistry

Volumn 6, Issue 10, 1998, Pages 1799-1810

  Yao, Zhu Jun ^a   Ye, Bin ^a   Wu, Xiong Wu ^b   Wang, Shaomeng ^b   Wu, Li ^c   Zhang, Zhong Yin ^c   Burke Jr , Terrence R ^a  

^a NATIONAL CANCER INSTITUTE   (United States)

^b GEORGETOWN UNIVERSITY MEDICAL CENTER   (United States)

^c ALBERT EINSTEIN COLLEGE OF MEDICINE   (United States)

Author keywords

Amino acids and derivatives; Mimetics; Phosphonic acids and derivatives; Phosphorylation

Indexed keywords

ARGININE; PROTEIN TYROSINE PHOSPHATASE INHIBITOR;

ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; DRUG DESIGN; DRUG SYNTHESIS; MOLECULAR DYNAMICS; NONHUMAN;

DRUG DESIGN; ENZYME INHIBITORS; HUMANS; MODELS, MOLECULAR; PROTEIN-TYROSINE-PHOSPHATASE; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0031757577     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0968-0896(98)00140-0     Document Type: Article

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