In vitro glucocorticoid receptor binding and transcriptional activation by topically active glucocorticoids

Arzneimittel-Forschung/Drug Research

Volumn 48, Issue 9, 1998, Pages 956-960

  Smith, Carolyn L ^a   Kreutner, William ^b  

^a BAYLOR COLLEGE OF MEDICINE   (United States)

^b MERCK RESEARCH LABORATORIES   (United States)

Author keywords

Budesonide; CAS 51372 29 3; CAS 76 25 5; CAS 80474 14 2; CAS 83919 237; Fluticasone propionate; Glucocorticoids, receptor binding, transactivation; Mometasone furoate; Sch 32088; Triamcinolone acetonide

Indexed keywords

BUDESONIDE; DEXAMETHASONE; FLUTICASONE PROPIONATE; GLUCOCORTICOID RECEPTOR; MOMETASONE FUROATE; RECOMBINANT PROTEIN; TRIAMCINOLONE ACETONIDE;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; DRUG RECEPTOR BINDING; GENE ACTIVATION; HUMAN; NONHUMAN; TRANSACTIVATION;

ANIMALS; ANTI-ALLERGIC AGENTS; ANTI-ASTHMATIC AGENTS; CELL LINE; GENES, REPORTER; GENETIC VECTORS; GLUCOCORTICOIDS; HUMANS; PLASMIDS; RECEPTORS, GLUCOCORTICOID; RECOMBINANT PROTEINS; RESPONSE ELEMENTS; TRANS-ACTIVATION (GENETICS);

EID: 0031752621     PISSN: 00044172     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (33)

1. Barnes, P. J., Am. J. Respir. Crit. Care Med. 154, s21 (1996)
2. Barnes, P. J., N. Engl. J. Med. 332, 868 (1995)
3. Umland, S. P., Nahrebne, K., Razac, S. et al., J. Allergy Clin. Immunol. 100, 511 (1997)
4. Barnes, P. J., J. Allergy Clin. Immunol. 97, 159 (1996)
5. Tsai, M.-J., O'Malley, B. W., Ann. Rev. Biochem. 63, 451 (1994)
6. McEwan, I. J., Wright, A. P., Gustafsson, J. A., Bioassay 19, 153 (1997)
7. Auphan, N., Didonato, J. A., Rosette, C. et al., Science 270, 286 (1995)
8. Jonat, C., Rahmsdorf, H. J., Park, K. K. et al., Cell 62, 1189 (1990)
9. Schule, R., Rangarajan, P., Kliewer, S. et al., Cell 62, 1217 (1990)
10. Yang-Yen, H. F., Chambard, J. C., Sun, Y. L. et al., Cell 62, 1205 (1990)
11. Ray, A., Prefontaine, K. E., Proc. Natl. Acad. Sci. USA 91, 752 (1994)
12. Mori, A., Kaminuma, O., Suko, M. et al., Blood 89, 2891 (1997)
13. Brattsand, R., Linden, M., Ailment Pharmacol Ther. 10 (Suppl. 2), 81 (1996)
14. NHLBI, Guidelines for the Diagnosis and Management of Asthma, p. 89, NIH Publications, No. 97-4051, Bethesda, MD, USA (1997)
15. Giguere, V., Ong, E. S., Segui, P. et al., Nature 330, 624 (1987)
16. Allgood, V. E., Oakley, R. H., Cidlowski, J. A., J. Biol. Chem. 268, 20870 (1993)
17. Apostolakis, E. M., Garai, J., Fox, C. J. et al., Neuroscience 16, 4823 (1996)
18. Allgood, V. E., Zhang, Y., O'Malley, B. W. et al., Biochemistry 36, 224 (1997)
19. Mak, P., McDonnell, D. P., Weigel, N. L. et al., J. Biol. Chem. 264, 21613 (1989)
20. Seed, B., Sheen, J.-Y., Gene 67, 271 (1988)
21. Smith, C. L., Conneely, O. M., O'Malley, B. W., Proc. Natl. Acad. Sci. USA 90, 6120 (1993)
22. Bradford, M. M., Anal. Biochem. 72, 248 (1976)
23. Crocker, I. C., Newton, S., Townley, R. G., J. Allergy Clin. Immunol. 99, s331 (1997)
24. Hochhaus, G., Mollmann, H., Derendorf, H. et al., J. Clin. Pharmacol. 37, 881 (1997)
25. Johnson, M. J., Allergy Clin. Immunol. 97, 169 (1996)
26. Dahlberg, E., Thalen, A., Brattsand, R. et al., Mol. Pharmacol. 25, 70 (1983)
27. Hochhaus, G., Mollmann, J., Barth, J., Pharm. Res. 13, 1699 (1996)
28. Wuerthwein, G., Rehder, S., Rohdewald, P., Pharm. Ztg. Wiss. 137, 161 (1992)
29. Reed, C. E., Am. Rev. Respir. Dis. 140, s82 (1990)
30. Bickel, C. A., Stellato, C., Schleimer, R. P., J. Allergy Clin. Immunol. 99, s401 (1997)
31. Mandl, M., Nolop, K., Lutsky, B. N., Ann. Allergy Asthma Immunol. 79, 237 (1997)
32. Drouin, M., Yang, W. H., Bertrand, B., Ann. Allergy Asthma Immunol. 77, 153 (1996)
33. Hebert, J. R., Nolop, K., Lutsky, B. N., Allergy 51, 569 (1996)