Effect of gastric pH on the bioavailability of albendazole in rabbits

Pharmacy and Pharmacology Communications

Volumn 4, Issue 5, 1998, Pages 267-270

  Kohri, N ^a   Yamayoshi, Y ^b   Iseki, K ^b   Sato, N ^b   Todo, S ^b   Miyazaki, K ^a,b  

^a HOKKAIDO INSTITUTE OF TECHNOLOGY   (Japan)

^b HOKKAIDO UNIVERSITY HOSPITAL   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

ALBENDAZOLE;

ANIMAL EXPERIMENT; ARTICLE; CONTROLLED STUDY; DRUG ABSORPTION; DRUG BIOAVAILABILITY; DRUG SOLUBILITY; NONHUMAN; ORAL DRUG ADMINISTRATION; RABBIT; STOMACH PH;

EID: 0031745410     PISSN: 14608081     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (20)

1. Aoyagi, N., Ogata, H., Kaniwa, N., Ejima, A. (1985) Bioavailability of indomethacin capsules in humans. (I): Bioavailability and effects of gastric acidity. Int. J. Clin. Pharmacol. 23: 469-474
2. Awadzi, K., Hero, M., Opoku, N. O., Büttner, D. W., Coventry, P. A., Prime, M. A., Orme, M. L'E., Edwards, G. (1994) The chemotherapy of onchocerciasis XVII. A clinical evaluation of albendazole in patients with onchocerciasis; effects of food and pretreatment with ivermectin on drug response and phar-macokinetics. Trop. Med. Parasitol. 45: 203-208
3. Ishizu, H., Uchino, J., Sato, N., Aoki, S., Suzuki, K., Kuribayashi, H. (1997) Effect of albendazole on recurrent and residual alveolar echinococcosis of the liver after surgery. Hepatology 25: 528-531
4. Jung, H., Hurtado, M., Sanchez, M., Medina, M. T., Sotelo, J. (1992) Clinical pharmacokinetics of albendazole in patients with brain cysticercosis. J. Clin. Pharmacol. 32: 28-31
5. Kohri, N., Miyata, N., Takahashi, M., Endo, H., Iseki, K., Miyazaki, K., Takechi, S., Nomura, A. (1992) Evaluation of pH-independent sustained-release granules of dipyridamole by using gastric-acidity-controlled rabbits and human subjects. Int. J. Pharm. 81: 49-58
6. Lange, H., Eggers, R., Bircher, J. (1988) Increased systemic availability of albendazole when taken with a fatty meal. Eur. J. Clin. Pharmacol. 34: 315-317
7. Lewis, J. W., Koss, N., Kerstein, M. D. (1975) A review of echinococcal disease. Ann. Surg. 181: 390-396
8. Malagelada, J. R., Longstreth, G. F., Summerskill, W. H. J., Go, V. L. W. (1976) Measurement of gastric functions during digestion of ordinary solid meals in man. Gastroenterology 70: 203-210
9. Marriner, S. E., Morris, D. L., Dickson, B., Bogan, J. A. (1986) Pharmacokinetics of albendazole in man. Eur. J. Clin. Pharmacol. 30: 705-708
10. Meldrum, S. J., Watson, B. W., Riddle, H. C. (1972) pH profile of gut as measured by radiotelemetry capsule. Br. Med. J. 2: 104-106
11. Ogata, H., Aoyagi, N., Kaniwa, N., Koibuchi, M., Shibazaki, T., Ejima, A., Watanabe, Y., Motohashi, K., Thuji, S., Kawazu, Y. (1980) Relation between drug bioavailability from solid dosage form in human and dissolution rate: acidity of human gastric fluid and drug bioavailability. J. Pharmacobio-Dyn. 3: s-17
12. Ogata, H., Aoyagi, N., Kaniwa, N., Koibuchi, M., Shibazaki, T., Ejima, A. (1982) The bioavailability of diazepam from uncoated tablets in humans. I.: Effect of gastric fluid acidity. Int. J. Clin. Pharmacol. Ther. Toxicol. 20: 166-170
13. Ogata, H., Aoyagi, N., Kaniwa, N., Ejima, A., Suzuki, K., Ishioka, T., Morishita, M., Ohta, K., Takagishi, Y., Doi, Y., Ogura, T. (1984) Development and evaluation of a new peroral test agent GA-Test for assessment of gastric acidity. J. Pharmacobio-Dyn. 7: 656-664
14. Ogata, H., Aoyagi, N., Kaniwa, N., Shibazaki, T., Ejima, A., Takagishi, Y., Ogura, T., Tomita, K., Inoue, S., Zaizen, M. (1985) Bioavailability of metronidazole from sugar-coated tablets in humans. I. Effect of gastric acidity and correlation with in vitro dissolution rate. Int. J. Pharm. 23: 277-288
15. Sato, N., Uchino, J., Aoki, S., Taguchi, K., Nishikawa, M., Baba, E., Nakagawa, T., Hata, T., Shimamura, T., Kamiyama, T., Takahashi, M., Matsushita, M., Nakajima, Y., Une, Y., Kuribayashi, H., Suzuki, K., Kohri, N., Iseki, K., Miyazaki, K. (1994) Efficacy of benzimidazole-type drugs on alveolar echinococcosis (AE). Jpn. J. Gastroentero. 91: 1197-1204
16. Takahashi, T., Shirai, Y., Nakamura, Y., Uezono, Y., Makita, H., Nakanishi, Y., Imasato Y. (1985) Movement of granules and tablets in the gastrointestinal tract of gastric-emptying-controlled rabbits. Chem. Pharm. Bull. 33: 5495-5502
17. Uchino, J., Sato, N., Nakajima, Y., Mathushita, M., Takahashi, M., Une, Y. (1993) Alveolar echinococcosis of the liver. In: Uchino, J., Sato., N. (eds) Hokkaido University Medical Library Series. Vol 30. Kokoku Printing, pp 137-149
18. Wen, H., Zou, P. F., Yang, W. G., Lu, J., Wang, Y. H., Zhang, J. H., New, R. R., Craig, P. S. (1994) Albendazole chemotherapy for human cystic and alveolar echinococcosis in north-western China. Trans. R. Soc. Trop. Med. Hyg. 88: 340-343
19. Wilson, J. F., Rausch, R. L., McMahon, B. J., Schantz, P. M. (1992) Parasitocidal effect of chemotherapy in alveolar hydatid disease: review of experience with mebendazole and albendazole in Alaskan Eskimos. Clin. Infect. Dis. 15: 234-249
20. Yamaoka, K., Tanigawara, Y., Nakagawa, T., Uno, T. (1981) A pharmacokinetic analysis program (MULTI) for micro-computer. J. Pharmacobio-Dyn. 4: 879-885