Activation of various subtypes of G-protein α subunits by partial agonists of the adenosine A1 receptor

Biochemical Pharmacology

Volumn 56, Issue 10, 1998, Pages 1287-1293

  Lorenzen, Anna ^a   Lang, Heidrun ^a   Schwabe, Ulrich ^a  

^a UNIVERSITY OF HEIDELBERG   (Germany)

Author keywords

Adenosine A1 receptor; G(i); G(o); GTP S; Partial agonist; Reconstitution

Indexed keywords

2 ANILINOADENOSINE; 2 CHLORO 6 N CYCLOPENTYLADENOSINE; 2' DEOXY N6 CYCLOPENTYLADENOSINE; 3' DEOXY N6 CYCLOPENTYLADENOSINE; 5' METHYLTHIOADENOSINE; 8 AMINOPROPYL N6 CYCLOPENTYLADENOSINE; ADENOSINE A1 RECEPTOR; ADENOSINE A1 RECEPTOR AGONIST; CLADRIBINE; GUANINE NUCLEOTIDE BINDING PROTEIN; GUANOSINE 5' O (3 THIOTRIPHOSPHATE); N ETHYLMALEIMIDE; PARTIAL AGONIST; PROTEIN SUBUNIT; SULFUR 35; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; BRAIN CORTEX; BRAIN MEMBRANE; CONTROLLED STUDY; DRUG POTENCY; NONHUMAN; PRIORITY JOURNAL; RAT;

ADENOSINE; ANIMALS; GTP-BINDING PROTEINS; GUANOSINE 5'-O-(3-THIOTRIPHOSPHATE); PROSENCEPHALON; PROTEIN BINDING; RATS; RECEPTORS, PURINERGIC P1; RECOMBINANT PROTEINS;

EID: 0031741567     PISSN: 00062952     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0006-2952(98)00207-X     Document Type: Article

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