Structure-activity studies of analogues of neurokinin A mediating contraction of rat uterus

Neuropeptides

Volumn 32, Issue 5, 1998, Pages 405-410

  Fisher, L ^a   Pennefather, J N ^a  

^a MONASH UNIVERSITY   (Australia)

Author keywords

[No Author keywords available]

Indexed keywords

AMASTATIN; N (1 CARBOXY 3 PHENYLPROPYL)PHENYLALANYLISOSERINE; NEUROKININ A; NEUROKININ A DERIVATIVE; NEUROKININ A [4-10]; NEUROKININ A [4-10][10 NORLEUCINE];

AMINO ACID COMPOSITION; ANIMAL TISSUE; ARTICLE; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG POTENCY; FEMALE; NONHUMAN; PRIORITY JOURNAL; RAT; STRUCTURE ACTIVITY RELATION; UTERUS CONTRACTILITY; UTERUS CONTRACTION;

ANIMALIA; ORYCTOLAGUS CUNICULUS;

EID: 0031737222     PISSN: 01434179     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0143-4179(98)90063-4     Document Type: Article

References (21)

1. 2 receptors. Peptides 1993; 14: 903-906.
2. Fisher L, Pennefather J N, Hall S. Tachykinin receptors in the rat isolated uterus. Regul Pept 1993; 46: 396-398.
3. Fisher L, Pennefather J N. Potencies of agonists acting at tachykinin receptors in the oestrogen-primed rat uterus: effects of peptidase inhibitors. Eur J Pharmacol 1997; 335: 221-226.
4. Regoli D, Drapeau G, Dion S, Couture R. New selective agonists for neurokinin receptors: pharmacological tools for receptor characterisation. Trends Pharmacol Sci 1988; 9: 290-295.
5. Rovero P, Pestellini V, Rhaleb N -E et al. Structure-activity studies of neurokinin A. Neuropeptides 1989: 13: 263-270.
6. Cascieri M A, Huang R -R C, Fong T M et al. Determination of the amino acid residues in substance P conferring selectivity for the rat neurokinin receptors. Mol Pharmacol 1992; 41: 1096-1099.
7. 10]NKA(4-10). Biochem Soc Trans 1993; 22: 5S.
8. Regoli D, Nantel F. Pharmacology of neurokinin receptors. Biopolymers 1991; 31: 777-783.
9. Munekata E, Kubo K, Tanaka H, Osakada F. Structure-activity studies of heptapeptide derivatives related to substance P, neurokinin A, B and other tachykinins on smooth muscles. Peptides 1987; 8: 169-173.
10. Regoli D, Dion S, Rhaleb N -E et al. Selective agonists for receptors of substance P and related neurokinins. Biopolymers 1989; 28: 81-90.
11. Drapeau G, D'Orleans-Juste P, Dion S, Rhaleb N -E, Rouissi N -E, Regoli D. Selective agonists for substance P and neurokinin receptors. Neuropeptides 1987; 10: 43-54.
12. 3 bioassay). Neuropeptides 1991; 19: 91-95.
13. Bray A M, Valerio R M, Dipasquale A J, Greig J, Maeji N J. Multiple synthesis by the multipin method as a methodological tool. J Pept Sci 1995; 1: 80-87
14. Regoli D, Drapeau G, Dion S, D'Orleans-Juste P. Pharmacological receptors for substance P and neurokinins. Life Sci 1987; 40: 109-117.
15. Badgery-Parker T, Lovas S, Conlon J M, Burcher E. Receptor binding profile of neuropeptide γ and its fragments: comparison with the non-mammalian peptides carassin and ranakinin at three mammalian tachykinin receptors. Peptides 1993; 14: 771-775.
16. Erspamer V, Anastasi A. Structure and pharmacological actions of eledoisin, the active endecapeptide of the posterior salivary glands of Eledone. Experientia 1962; 18: 58-59.
17. Anastasi A, Erspamer G F. Occurrence of phyllomedusin, a physalaemin-like decapeptide, in the skin of Phyllomedusa bicolor. Experientia 1970; 26: 866-867.
18. Erspamer V, Anastasi A, Bertaccini G, Cei J M. Structure and pharmacological actions of physalaemin, the main active ingredient of the skin of Physalaemus fuscumaculatus. Experientia 1964; 20: 489-490.
19. Anastasi A, Erspamer V, Endean R. Structure of uperolein, a physalaemin-like endecapeptide occurring in the skin of Uperoleia rugosa and Uperoleia marmorata. Experientia 1975; 31: 394-395.
20. Conlon J M, Deacon C F, O'Toole L, Thim L Scyliorhinin I and II: two novel tachykinins from dog-fish gut. FEES Lett 1986; 200: 111-116.
21. D'Orleans-Juste P, Dion S, Drapeau G, Regoli D. Different receptors are involved in the endothelium-mediated relaxation and the smooth muscle contraction of the rabbit pulmonary artery in response to substance P and related neurokinins. Eur J Pharmacol 1985; 125: 37-44.