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Volumn 15, Issue 9, 1998, Pages 1370-1375

Prediction of intestinal drug absorption properties by three- dimensional solubility parameters

Author keywords

Carrier mediated transport; Hansen solubility parameters; Passive diffusion; Regional gastrointestinal uptake; Site specific delivery; Sustained release dosage forms

Indexed keywords

ALLOPURINOL; AMPICILLIN; BETAMETHASONE; CHLORAMPHENICOL; DICOUMAROL; DIGOXIN; DOXYCYCLINE; ERYTHROMYCIN; FUROSEMIDE; GLIBENCLAMIDE; HYDROCHLOROTHIAZIDE; INDOMETACIN; ISOSORBIDE MONONITRATE; METACYCLINE; METHAQUALONE; METOPROLOL; METRONIDAZOLE; NITROFURANTOIN; OXYTETRACYCLINE; PARACETAMOL; PENICILLIN V; PHENYTOIN; PREDNISOLONE; PROPRANOLOL; PYRIDOXAL 5 PHOSPHATE; QUINIDINE; RIBOFLAVIN; SULFINPYRAZONE; TETRACYCLINE; UNINDEXED DRUG;

EID: 0031722109     PISSN: 07248741     EISSN: None     Source Type: Journal    
DOI: 10.1023/A:1011941319327     Document Type: Article
Times cited : (100)

References (30)
  • 1
    • 0002019378 scopus 로고
    • Ratelimiting steps and factors in drug absorption
    • L. F. Prescott, W. S. Nimmo, MTP Press Limited, Lancaster UK
    • W. I. Higuchi, N. F. H. Ho, J. Y. Park, and I. Komiya. Ratelimiting steps and factors in drug absorption. In L. F. Prescott, W. S. Nimmo, Drug absorption, MTP Press Limited, Lancaster UK, 1981, pp. 35-60.
    • (1981) Drug Absorption , pp. 35-60
    • Higuchi, W.I.1    Ho, N.F.H.2    Park, J.Y.3    Komiya, I.4
  • 2
    • 0029953050 scopus 로고    scopus 로고
    • Drug absorption sites in the gastrointestinal tract and dosage forms for site-specific delivery
    • N. Rouge, P. Buri, and E. Doelker. Drug absorption sites in the gastrointestinal tract and dosage forms for site-specific delivery. Int. J. Pharm. 136:117-139 (1996).
    • (1996) Int. J. Pharm. , vol.136 , pp. 117-139
    • Rouge, N.1    Buri, P.2    Doelker, E.3
  • 3
    • 0029782485 scopus 로고    scopus 로고
    • Carrier-mediated intestinal transport of drugs
    • A. Tsuji and I. Tamai. Carrier-mediated intestinal transport of drugs. Pharm. Res. 13:963-977 (1996).
    • (1996) Pharm. Res. , vol.13 , pp. 963-977
    • Tsuji, A.1    Tamai, I.2
  • 4
    • 0028948839 scopus 로고
    • A theoretical basis for a biopharmaceutic drug classification: The correlation of in vitro drug product dissolution and in vivo bioavailability
    • G. L. Amidon, H. Lennernäs, V. P. Shah, and J. R. Crison. A theoretical basis for a biopharmaceutic drug classification: The correlation of in vitro drug product dissolution and in vivo bioavailability. Pharm. Res. 12:413-420 (1995).
    • (1995) Pharm. Res. , vol.12 , pp. 413-420
    • Amidon, G.L.1    Lennernäs, H.2    Shah, V.P.3    Crison, J.R.4
  • 5
    • 0030580951 scopus 로고    scopus 로고
    • Transport approaches to the biopharmaceutical design of oral drug delivery systems: Prediction of intestinal absorption
    • L. X. Yu, E. Lipka, J. R. Crison, and G. L. Amidon. Transport approaches to the biopharmaceutical design of oral drug delivery systems: prediction of intestinal absorption. Adv. Drug Deliver. Rev. 19:359-376 (1996).
    • (1996) Adv. Drug Deliver. Rev. , vol.19 , pp. 359-376
    • Yu, L.X.1    Lipka, E.2    Crison, J.R.3    Amidon, G.L.4
  • 6
    • 0031026707 scopus 로고    scopus 로고
    • Simulation models to predict oral drug absorption from in vitro data
    • G. M. Grass. Simulation models to predict oral drug absorption from in vitro data. Adv. Drug Deliver. Rev. 23:199-219 (1997).
    • (1997) Adv. Drug Deliver. Rev. , vol.23 , pp. 199-219
    • Grass, G.M.1
  • 7
    • 0015545469 scopus 로고
    • Lipophilic character and biological activity of drugs II: The parabolic case
    • C. Hansch and J. M. Clayton. Lipophilic character and biological activity of drugs II: The parabolic case. J. Pharm. Sci. 62:1-21 (1973).
    • (1973) J. Pharm. Sci. , vol.62 , pp. 1-21
    • Hansch, C.1    Clayton, J.M.2
  • 8
    • 0025731738 scopus 로고
    • Partitioning of solutes in different solvent systems: The contribution of hydrogen-bonding capacity and polarity
    • N. El-Tayar, R.-S. Tsai, B. Testa, P.-A. Carrupt, and A. Leo. Partitioning of solutes in different solvent systems: The contribution of hydrogen-bonding capacity and polarity. J. Pharm. Sci. 80:590-598 (1991).
    • (1991) J. Pharm. Sci. , vol.80 , pp. 590-598
    • El-Tayar, N.1    Tsai, R.-S.2    Testa, B.3    Carrupt, P.-A.4    Leo, A.5
  • 9
    • 0014479469 scopus 로고
    • The universality of the solubility parameter
    • C. M. Hansen. The universality of the solubility parameter. Ind. Eng. Chem. Res. Devel. 8:2-11 (1969).
    • (1969) Ind. Eng. Chem. Res. Devel. , vol.8 , pp. 2-11
    • Hansen, C.M.1
  • 11
    • 0027078680 scopus 로고
    • A new method for the estimation of the aqueous solubility of organic compounds
    • N. Bodor and M.-J. Huang. A new method for the estimation of the aqueous solubility of organic compounds. J. Pharm. Sci. 81:954-960 (1992).
    • (1992) J. Pharm. Sci. , vol.81 , pp. 954-960
    • Bodor, N.1    Huang, M.-J.2
  • 12
    • 0026640391 scopus 로고
    • Topological inidices in correlation analysis. Part 3: The modelling of hydrophobic properties using molecular connectivity and shape indices
    • J. L. Mokrosz, B. Duszynska, and L. Strekowski. Topological inidices in correlation analysis. Part 3: The modelling of hydrophobic properties using molecular connectivity and shape indices. Pharmazie 47:538-541 (1992).
    • (1992) Pharmazie , vol.47 , pp. 538-541
    • Mokrosz, J.L.1    Duszynska, B.2    Strekowski, L.3
  • 13
    • 0030914681 scopus 로고    scopus 로고
    • Polar molecular surface properties predict the intestinal absorption of drugs in humans
    • K. Palm, P. Stenberg, K. Luthmann, and P. Artursson. Polar molecular surface properties predict the intestinal absorption of drugs in humans. Pharm. Res. 14:568-571 (1997).
    • (1997) Pharm. Res. , vol.14 , pp. 568-571
    • Palm, K.1    Stenberg, P.2    Luthmann, K.3    Artursson, P.4
  • 14
    • 0030004786 scopus 로고    scopus 로고
    • Threedimensional solubility parameters and their use in characterising the permeation of drugs through the skin
    • R. Gröning and F.-J. Braun. Threedimensional solubility parameters and their use in characterising the permeation of drugs through the skin. Pharmazie 51:337-341 (1996).
    • (1996) Pharmazie , vol.51 , pp. 337-341
    • Gröning, R.1    Braun, F.-J.2
  • 15
    • 4243243993 scopus 로고    scopus 로고
    • Rectal absorption of drugs - Indirect characterisation of the rectal membrane using the Bagley diagram and in vivo drug absorption data
    • R. Gröning, W. Sakran, F.-J. Braun, M. S. Adel, A: Abd El-Bary, and M. F. El-Miligi. Rectal absorption of drugs - indirect characterisation of the rectal membrane using the Bagley diagram and in vivo drug absorption data. Eur. J. Pharm. Biopharm. 42(Suppl.):55 S (1996).
    • (1996) Eur. J. Pharm. Biopharm. , vol.42 , Issue.SUPPL.
    • Gröning, R.1    Sakran, W.2    Braun, F.-J.3    Adel, M.S.4    Abd El-Bary, A.5    El-Miligi, M.F.6
  • 16
    • 0016025821 scopus 로고
    • A method for estimating both the solubility parameters and molar volumes of liquids
    • R. F. Fedors. A method for estimating both the solubility parameters and molar volumes of liquids. Polymer Engin. Sci. 14:147-154 (1974).
    • (1974) Polymer Engin. Sci. , vol.14 , pp. 147-154
    • Fedors, R.F.1
  • 19
    • 33847802745 scopus 로고
    • Solubility parameters
    • A. F. M. Barton. Solubility parameters. Chem. Rev. 75:731-753 (1975).
    • (1975) Chem. Rev. , vol.75 , pp. 731-753
    • Barton, A.F.M.1
  • 20
    • 0002815444 scopus 로고
    • Three-dimensional solubility parameters and their relationship to internal pressure measurements in polar and hydrogen bonding solvents
    • E. B. Bagley, T. P. Nelson, and J. M. Scigliano. Three-dimensional solubility parameters and their relationship to internal pressure measurements in polar and hydrogen bonding solvents. J. Paint Technol. 43:35-42 (1971).
    • (1971) J. Paint Technol. , vol.43 , pp. 35-42
    • Bagley, E.B.1    Nelson, T.P.2    Scigliano, J.M.3
  • 21
    • 0024591344 scopus 로고
    • Charakterisierung der Arzneistoffabsorption aus dem Gastrointestinaltrakt mit Hilfe der numerischen Dekonvolution
    • R. Gröning and G. Heun. Charakterisierung der Arzneistoffabsorption aus dem Gastrointestinaltrakt mit Hilfe der numerischen Dekonvolution. Pharm. Acta Helv. 64:71-75 (1989).
    • (1989) Pharm. Acta Helv. , vol.64 , pp. 71-75
    • Gröning, R.1    Heun, G.2
  • 22
    • 15444348044 scopus 로고    scopus 로고
    • Methods used to investigate drug absorption in the colon: A review
    • Düsseldorf
    • A. H. Staib. Methods used to investigate drug absorption in the colon: A review. Workshop "Colon-Resorption und Colon-Targeting", Düsseldorf, 1996.
    • (1996) Workshop "Colon-Resorption und Colon-Targeting"
    • Staib, A.H.1
  • 23
    • 0024599205 scopus 로고
    • Acyclovir - An updated review of its antiviral activity, pharmacokinetic properties and therapeutic efficacy
    • J. J. O'Brien and D. M. Campoli-Richards. Acyclovir - an updated review of its antiviral activity, pharmacokinetic properties and therapeutic efficacy. Drugs 37:233-309 (1989).
    • (1989) Drugs , vol.37 , pp. 233-309
    • O'Brien, J.J.1    Campoli-Richards, D.M.2
  • 24
    • 0023404750 scopus 로고
    • Clinical Pharmacokinetics of Anti-Parkinsonian Drugs
    • J. M. Cedarbaum. Clinical Pharmacokinetics of Anti-Parkinsonian Drugs. Clin. Pharmacokin. 13:141-178 (1987).
    • (1987) Clin. Pharmacokin. , vol.13 , pp. 141-178
    • Cedarbaum, J.M.1
  • 26
    • 0026567874 scopus 로고
    • The absorption site of cyclosporin in the human gastrointestinal tract
    • J. Drewe, C. Beglinger, and T. Kissel. The absorption site of cyclosporin in the human gastrointestinal tract. Br. J. Clin. Pharmac. 30:35-39 (1992).
    • (1992) Br. J. Clin. Pharmac. , vol.30 , pp. 35-39
    • Drewe, J.1    Beglinger, C.2    Kissel, T.3
  • 27
    • 0022640190 scopus 로고
    • The absorption of piretanide from the gastro-intestinal tract is site-dependent
    • D. Brockmeier, H. G. Grigleit, H. Leonhardt. The absorption of piretanide from the gastro-intestinal tract is site-dependent. Eur. J. Clin. Pharmacol. 30:79-82 (1986).
    • (1986) Eur. J. Clin. Pharmacol. , vol.30 , pp. 79-82
    • Brockmeier, D.1    Grigleit, H.G.2    Leonhardt, H.3
  • 28
    • 0023732860 scopus 로고
    • Relationship between the rate of appearance of oxprenolol in the systemic circulation and the location of an oxprenolol oros 16/260 drug delivery system within the gastrointestinal tract as determined by scintigraphy
    • S. S. Davis, N. Washington, A. H. Short, V. A. John, P. Lloyd, S. M. Walker. Relationship between the rate of appearance of oxprenolol in the systemic circulation and the location of an oxprenolol oros 16/260 drug delivery system within the gastrointestinal tract as determined by scintigraphy Br. J. Clin. Pharmac. 26:435-443 (1988).
    • (1988) Br. J. Clin. Pharmac. , vol.26 , pp. 435-443
    • Davis, S.S.1    Washington, N.2    Short, A.H.3    John, V.A.4    Lloyd, P.5    Walker, S.M.6
  • 29
    • 0029585123 scopus 로고
    • Atom/fragment contribution method for estimating octanol-water partition coefficients
    • W. M. Meylan and P. H. Howard. Atom/fragment contribution method for estimating octanol-water partition coefficients. J. Pharm. Sci. 84:83-92 (1995).
    • (1995) J. Pharm. Sci. , vol.84 , pp. 83-92
    • Meylan, W.M.1    Howard, P.H.2
  • 30
    • 84958632244 scopus 로고    scopus 로고
    • Physicochemical and biological factors that influence a drug's cellular permeability by passive diffusion
    • V. Pliska, B. Testa, H. van rie Waterbeemd, VCH Verlagsgesellschaft, Weinheim, Germany
    • R. A. Conradi, P. S. Burton, and R. T. Borchardt. Physicochemical and biological factors that influence a drug's cellular permeability by passive diffusion. In V. Pliska, B. Testa, H. van rie Waterbeemd, Lipophilicity in drug action and toxicology, VCH Verlagsgesellschaft, Weinheim, Germany, 1996 pp. 233-252.
    • (1996) Lipophilicity in Drug Action and Toxicology , pp. 233-252
    • Conradi, R.A.1    Burton, P.S.2    Borchardt, R.T.3


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