Quantitative structure-activity studies of octopaminergic agonists and antagonists against nervous system of Locusta migratoria

Bioorganic and Medicinal Chemistry

Volumn 6, Issue 7, 1998, Pages 903-910

  Hirashima, Akinori ^a   Pan, Canping ^b   Shinkai, Kenji ^a   Tomita, Jun ^a   Kuwano, Eiichi ^d   Taniguchi, Eiji ^a   Eto, Morifusa ^c  

^a KYUSHU UNIVERSITY   (Japan)

^b CHINA AGRICULTURAL UNIVERSITY   (China)

^c MIYAKONOJO NATIONAL COLLEGE OF TECHNOLOGY   (Japan)

^d NONE

Author keywords

Locusta migratoria; Molecular shape analysis; Quantitative structure activity relationship (QSAR); Receptor surface model (RSM)

Indexed keywords

AMITRAZ; AMITRIPTYLINE; ANTAZOLINE; CHLORPROMAZINE; CYPROHEPTADINE; DESIPRAMINE; DIHYDROERGOTAMINE; GRAMINE; IMIPRAMINE; ISOPRENALINE; METOCLOPRAMIDE; NORADRENALIN; OCTOPAMINE; OCTOPAMINE RECEPTOR BLOCKING AGENT; OCTOPAMINE RECEPTOR STIMULATING AGENT; RECEPTOR BLOCKING AGENT; TRIPROLIDINE; UNCLASSIFIED DRUG;

AGONIST; ARTICLE; DRUG RECEPTOR BINDING; DRUG STRUCTURE; HYDROPHOBICITY; LOCUST; MOLECULAR MODEL; NERVE CORD; NERVOUS SYSTEM; NONHUMAN; PHYSICAL CHEMISTRY; QUANTITATIVE STRUCTURE ACTIVITY RELATION; REGRESSION ANALYSIS;

ANIMALS; GRASSHOPPERS; LIGANDS; MODELS, MOLECULAR; MOLECULAR CONFORMATION; OCTOPAMINE; RECEPTORS, BIOGENIC AMINE; REGRESSION ANALYSIS; STRUCTURE-ACTIVITY RELATIONSHIP;

LOCUSTA MIGRATORIA;

EID: 0031694296     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0968-0896(98)00024-8     Document Type: Article

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