Sulfonylamido derivatives of 2-aminophenoxathiin-10,10-dioxide and related compounds possess antifungal action due to the possible inhibition of lanosterol-14-α-demethylase

Journal of Enzyme Inhibition

Volumn 13, Issue 4, 1998, Pages 291-310

  Supuran, Claudiu T ^a   Scozzafava, Andrea ^a   Briganti, Fabrizio ^a   Loloiu, George ^b   Maior, Ovidiu ^b  

^a UNIVERSITY OF FLORENCE   (Italy)

^b UNIVERSITY OF BUCHAREST   (Romania)

Author keywords

(Thio)ureas; Antifungal compounds; Lanosterol 14 demethylase

Indexed keywords

ANTIFUNGAL AGENT; KETOCONAZOLE; LANOSTEROL DERIVATIVE; SULFANILAMIDE;

ANTIFUNGAL ACTIVITY; ARTICLE; ASPERGILLUS; CANDIDA; CHEMICAL REACTION; CONTROLLED STUDY; DERIVATIZATION; DRUG MECHANISM; DRUG SYNTHESIS; ENZYME INHIBITION; NONHUMAN; PRIORITY JOURNAL;

ASPERGILLUS; CANDIDA;

ANTIFUNGAL AGENTS; ASPERGILLUS; CANDIDA ALBICANS; CYCLIC S-OXIDES; CYTOCHROME P-450 ENZYME SYSTEM; HETEROCYCLIC COMPOUNDS; MAGNETIC RESONANCE SPECTROSCOPY; MICROBIAL SENSITIVITY TESTS; MOLECULAR STRUCTURE; OXIDOREDUCTASES; SPECTROPHOTOMETRY, INFRARED; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0031692059     PISSN: 87555093     EISSN: None     Source Type: Journal    
DOI: 10.3109/14756369809021477     Document Type: Article

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