[3H]MDL 105,519 binds with equal high affinity to both assembled and unassembled NR1 subunits of the NMDA receptor

European Journal of Pharmacology

Volumn 353, Issue 1, 1998, Pages 137-140

  Chazot, Paul L ^a   Reiss, Christian ^a   Chopra, Bela ^a   Stephenson, F Anne ^a  

^a UNIVERSITY OF LONDON   (United Kingdom)

Author keywords

Glutamate receptor; Glycine; NMDA receptor; NR1; Triton X 100

Indexed keywords

3 (2 CARBOXY 2 PHENYLETHENYL) 4,6 DICHLORO 1H INDOLE 2 CARBOXYLIC ACID; 5,7 DICHLOROKYNURENIC ACID; 7 CHLOROKYNURENIC ACID; DIZOCILPINE; N METHYL DEXTRO ASPARTIC ACID RECEPTOR; TRITON X 100; UNCLASSIFIED DRUG; AMINO ACID RECEPTOR BLOCKING AGENT; GLYCINE RECEPTOR; INDOLE DERIVATIVE; LIGAND; OCTOXINOL; RECOMBINANT PROTEIN;

ANIMAL TISSUE; ARTICLE; BINDING SITE; CONTROLLED STUDY; DRUG RECEPTOR BINDING; FOREBRAIN; KIDNEY CELL; NONHUMAN; PRIORITY JOURNAL; PROTEIN EXPRESSION; RAT; RECEPTOR AFFINITY; ANIMAL; BIOSYNTHESIS; CELL LINE; CHEMISTRY; DRUG ANTAGONISM; HUMAN; MEMBRANE; METABOLISM; RADIOASSAY; SOLUBILITY; WISTAR RAT;

ANIMALS; CELL LINE; EXCITATORY AMINO ACID ANTAGONISTS; HUMANS; INDOLES; LIGANDS; MEMBRANES; OCTOXYNOL; PROSENCEPHALON; RADIOLIGAND ASSAY; RATS; RATS, WISTAR; RECEPTORS, GLYCINE; RECEPTORS, N-METHYL-D-ASPARTATE; RECOMBINANT PROTEINS; SOLUBILITY;

EID: 0031595108     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(98)00431-2     Document Type: Article

References (12)

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