A systematic synthetic approach to phosphinophenyl-glycine and -alanine. Chiral phosphine ligands with amino acid moieties

Tetrahedron Letters

Volumn 38, Issue 13, 1997, Pages 2257-2258

  Tepper, Michael ^a   Stelzer, Othmar ^a   Häusler, Thomas ^b   Sheldrick, William S ^b  

^a UNIVERSITY OF WUPPERTAL   (Germany)

^b RUHR UNIVERSITY BOCHUM   (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

AMINO ACID DERIVATIVE; PHOSPHINE DERIVATIVE;

ARTICLE; DRUG SYNTHESIS; IN VITRO STUDY; METHODOLOGY; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; REACTION ANALYSIS; STEREOCHEMISTRY; X RAY DIFFRACTION;

EID: 0031592571     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(97)00335-3     Document Type: Article

References (13)

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2. 1. Krause, H. W.; Kreuzfeld, H. J.; Döbler, C. Tetrahedron: Asymmetry 1992, 3, 555-566; Hayashi, Y.; Sekiyama, N.; Nakanishi, S.; Jane, D. E.; Sunter, D. C.; Birse, E. F.; Udvarhelyi, P. M.; Watkins, J. C. Neuroscience, 1994, 14, 3370-3377; Thurieau, C.; Guyard, C.; Simonet, S.; Verbeuren, T. J.; Fauchère, J. L. Helv. Chim. Acta 1994, 77, 679-684.
3. 1. Krause, H. W.; Kreuzfeld, H. J.; Döbler, C. Tetrahedron: Asymmetry 1992, 3, 555-566; Hayashi, Y.; Sekiyama, N.; Nakanishi, S.; Jane, D. E.; Sunter, D. C.; Birse, E. F.; Udvarhelyi, P. M.; Watkins, J. C. Neuroscience, 1994, 14, 3370-3377; Thurieau, C.; Guyard, C.; Simonet, S.; Verbeuren, T. J.; Fauchère, J. L. Helv. Chim. Acta 1994, 77, 679-684.
4. 2. Jane, D. E.; Pittaway, K.; Sunter, D. C.; Thomas, N. K.; Watkins, J. C. Neuropharmacology, 1995, 34, 851-856.
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8. b) Wheatley, D. N.; Henderson, J. Y. Nature, 1974, 247, 281-283.
9. nJ(PC) in Hz in parentheses.
10. nJ(PC) in Hz in parentheses.
11. 2 with SHELXL-93 to R = 0.0446 (for I > 2σ(I) ) and wR2 = 0.126 for all 3463 independent reflections. Further details are available from Fachinformationszentrum Karlsruhe, D-76344 Eggenstein-Leopoldshafen on citing the deposition number CSD 405956.
12. 9. Togni, A.; Venanzi, L. M. Angew. Chem. 1994, 106, 517-547; Angew. Chem. Int. Ed. Engl. 1994, 33, 497-526.
13. 9. Togni, A.; Venanzi, L. M. Angew. Chem. 1994, 106, 517-547; Angew. Chem. Int. Ed. Engl. 1994, 33, 497-526.