The total synthesis of the natural product endothelin converting enzyme (ECE) inhibitor, WS75624 B

Tetrahedron Letters

Volumn 38, Issue 8, 1997, Pages 1297-1300

  Patt, William C ^a   Massa, Mark A ^a  

^a PFIZER INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

DIPEPTIDYL CARBOXYPEPTIDASE INHIBITOR; UNCLASSIFIED DRUG; WS 75624B;

ARTICLE; DRUG SYNTHESIS; IN VITRO STUDY; MASS SPECTROMETRY; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; REACTION ANALYSIS;

EID: 0031584908     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(97)00076-2     Document Type: Article

References (12)

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5. 5. Similar chemical strucure recently published: Trecourt, F.; Gervais, B.; Mallet, M.; Queguiner, G. J. Org. Chem. 1996, 61, 1673-1676.
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10. 3CN), ret.time= 2.4 min.
11. 11. Authentic sample was obtained from Fujisawa Pharmaceutical Co.
12. 12. Xu, D.; Emoto, N.; Giaid, A.; Slaughter, C.; Kaw, S.; deWit, D.; Yanagisawa, M. Cell 1994, 78, 473-485.