메뉴 건너뛰기




Volumn 53, Issue 4, 1997, Pages 531-538

Distinction of CYP1A1 and CYP1A2 activity by selective inhibition using fluvoxamine and isosafrole

Author keywords

CYP1A1; CYP1A2; ethoxyresorufin; fluvoxamine; human; isosafrole; O deethylas e

Indexed keywords

ALPHA NAPHTHOFLAVONE; APIGENIN; CYTOCHROME P450 ISOENZYME; FLUVOXAMINE; ISOSAFROLE;

EID: 0031581817     PISSN: 00062952     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0006-2952(96)00769-1     Document Type: Article
Times cited : (80)

References (23)
  • 1
    • 0026750647 scopus 로고
    • The human hepatic cytochromes P450 involved in drug metabolism
    • 1. Wrighton SA and Stevens JC, The human hepatic cytochromes P450 involved in drug metabolism. Crit Rev Toxicol 22: 1-21, 1992.
    • (1992) Crit Rev Toxicol , vol.22 , pp. 1-21
    • Wrighton, S.A.1    Stevens, J.C.2
  • 2
    • 0027756106 scopus 로고
    • In vitro methods for assessing human hepatic drug metabolism: Their use in drug development
    • 2. Wrighton SA, Wandenbranden M, Stevens JC, Shipley LA and Ring BJ, In vitro methods for assessing human hepatic drug metabolism: Their use in drug development. Drug Metab Rev 25: 453-484, 1993.
    • (1993) Drug Metab Rev , vol.25 , pp. 453-484
    • Wrighton, S.A.1    Wandenbranden, M.2    Stevens, J.C.3    Shipley, L.A.4    Ring, B.J.5
  • 3
    • 0027751340 scopus 로고
    • Induction of cytochrome P450 as an indicator of potential chemical carcinogenesis
    • 3. Ioannides C and Parke DV, Induction of cytochrome P450 as an indicator of potential chemical carcinogenesis. Drug Metab Dispos 25: 488-501, 1993.
    • (1993) Drug Metab Dispos , vol.25 , pp. 488-501
    • Ioannides, C.1    Parke, D.V.2
  • 4
    • 0025364520 scopus 로고
    • Differential expression and regulation of cytochrome P4501A gene subfamily in human tissues
    • 4. Sesardic D, Pelkonen O, Pasasen M and Boobis AR, Differential expression and regulation of cytochrome P4501A gene subfamily in human tissues. Carcinogenesis 11: 1183-1188, 1990.
    • (1990) Carcinogenesis , vol.11 , pp. 1183-1188
    • Sesardic, D.1    Pelkonen, O.2    Pasasen, M.3    Boobis, A.R.4
  • 6
    • 0026633834 scopus 로고
    • Roles of human liver cytochrome P4502C and 3A enzymes in the 3-hydroxylation of benzo(a)pyrene
    • 6. Yun C-H, Shimada T and Guengerich FP, Roles of human liver cytochrome P4502C and 3A enzymes in the 3-hydroxylation of benzo(a)pyrene. Cancer Res 52: 1868-1874, 1992.
    • (1992) Cancer Res , vol.52 , pp. 1868-1874
    • Yun, C.-H.1    Shimada, T.2    Guengerich, F.P.3
  • 7
    • 0017709375 scopus 로고
    • Interindividual and intraindividual variations in aryl hydrocarbon hydroxylase in monocytes form monozygotic and dizygotic twins
    • 7. Ocuda T, Vesell SE, Plotkin E, Tarone R, Bast RC and Gelboin HV, Interindividual and intraindividual variations in aryl hydrocarbon hydroxylase in monocytes form monozygotic and dizygotic twins. Cancer Res 37: 3904-3911, 1977.
    • (1977) Cancer Res , vol.37 , pp. 3904-3911
    • Ocuda, T.1    Vesell, S.E.2    Plotkin, E.3    Tarone, R.4    Bast, R.C.5    Gelboin, H.V.6
  • 9
    • 0026053685 scopus 로고
    • Selective in vitro inhibition of hepatic oxidative metabolism by quinolones: 7-Ethoxyresorufin and caffeine as model substrates
    • 9. Valero R, Segura J and Torre R, Selective in vitro inhibition of hepatic oxidative metabolism by quinolones: 7-Ethoxyresorufin and caffeine as model substrates. J Pharm Pharmacol 43: 17-21, 1992.
    • (1992) J Pharm Pharmacol , vol.43 , pp. 17-21
    • Valero, R.1    Segura, J.2    Torre, R.3
  • 10
    • 0028064672 scopus 로고
    • Development of a human lymphoblastoid cell line constitutively expressing human liver CYP1A1 cDNA: Substrate specificity with model substrates and promutagens
    • 10. Penman BW, Liping C, Gelboin HV, Gonzalez FJ and Crespi CL, Development of a human lymphoblastoid cell line constitutively expressing human liver CYP1A1 cDNA: Substrate specificity with model substrates and promutagens. Carcinogenesis 15: 1931-1937, 1994.
    • (1994) Carcinogenesis , vol.15 , pp. 1931-1937
    • Penman, B.W.1    Liping, C.2    Gelboin, H.V.3    Gonzalez, F.J.4    Crespi, C.L.5
  • 12
    • 0028174881 scopus 로고
    • Evaluation of triacetyloleandomycin, α-naphthoflavone and diethyldithiocarbamate as selective chemical probes for inhibition of human cytochromes P450
    • 12. Chang TKH, Gonzalez FJ and Waxman DJ, Evaluation of triacetyloleandomycin, α-naphthoflavone and diethyldithiocarbamate as selective chemical probes for inhibition of human cytochromes P450. Arch Biochem Biophys 311: 437-442, 1994.
    • (1994) Arch Biochem Biophys , vol.311 , pp. 437-442
    • Chang, T.K.H.1    Gonzalez, F.J.2    Waxman, D.J.3
  • 13
    • 0028362263 scopus 로고
    • Characterization of the inhibition of P4501A2 by furafylline
    • 13. Clarke SE, Ayrton AD and Chenery RJ, Characterization of the inhibition of P4501A2 by furafylline. Xenobiotica 6: 517-526, 1994.
    • (1994) Xenobiotica , vol.6 , pp. 517-526
    • Clarke, S.E.1    Ayrton, A.D.2    Chenery, R.J.3
  • 15
    • 0026725007 scopus 로고
    • Interaction between fluvoxamine and imipramine/ desipramine in four patients
    • 15. Spina E, Campo GM, Avenoso A, Pollicino MA and Caputi AP, Interaction between fluvoxamine and imipramine/ desipramine in four patients. Ther Drug Monit 14: 194-196, 1992.
    • (1992) Ther Drug Monit , vol.14 , pp. 194-196
    • Spina, E.1    Campo, G.M.2    Avenoso, A.3    Pollicino, M.A.4    Caputi, A.P.5
  • 16
    • 0028898044 scopus 로고
    • Selective serotonin reuptake inhibitors and theophylline metabolism in human liver microsomes: Potent inhibition by fluvoxamine
    • 16. Rasmussen BB, Maenpaa J, Pelkonen O, Loft S, Poulsen HE, Lykkesfeldt J and Brosen K, Selective serotonin reuptake inhibitors and theophylline metabolism in human liver microsomes: Potent inhibition by fluvoxamine. Br J Clin Pharmacol 39: 151-159, 1995.
    • (1995) Br J Clin Pharmacol , vol.39 , pp. 151-159
    • Rasmussen, B.B.1    Maenpaa, J.2    Pelkonen, O.3    Loft, S.4    Poulsen, H.E.5    Lykkesfeldt, J.6    Brosen, K.7
  • 17
    • 0027481679 scopus 로고
    • Inducibility of enzyme activities associated with the cytochrome P450 1A family, ethoxyresorufin O-deethylase, and methoxyresorufin O-demethylase in human hepatocyte lines derived from normal liver tissue
    • 17. Roberts EA, Xie ZW, Yang S and Lipa J, Inducibility of enzyme activities associated with the cytochrome P450 1A family, ethoxyresorufin O-deethylase, and methoxyresorufin O-demethylase in human hepatocyte lines derived from normal liver tissue. Drug Metab Dispos 21: 56-61, 1993.
    • (1993) Drug Metab Dispos , vol.21 , pp. 56-61
    • Roberts, E.A.1    Xie, Z.W.2    Yang, S.3    Lipa, J.4
  • 18
    • 0024324192 scopus 로고
    • Evidence in humans for variant alloenzymes of the nondeficient sparteine/debrisoquine monooxygenase in vitro
    • 18. Tyndale RF, Inaba T and Kalow W, Evidence in humans for variant alloenzymes of the nondeficient sparteine/debrisoquine monooxygenase in vitro. Drug Metab Dispos 17: 334-340, 1989.
    • (1989) Drug Metab Dispos , vol.17 , pp. 334-340
    • Tyndale, R.F.1    Inaba, T.2    Kalow, W.3
  • 19
    • 0011194362 scopus 로고
    • Phenacetin O-deethylase in novel human hepatocyte lines: Evidence for preservation of basal and inducible CYP1A2 in vitro
    • 19. Roberts EA, Kohno Y, Pastrakuljic A, Tang BK and Kalow W, Phenacetin O-deethylase in novel human hepatocyte lines: Evidence for preservation of basal and inducible CYP1A2 in vitro. Hepatobgy 20: 187A, 1994.
    • (1994) Hepatobgy , vol.20 , Issue.187 A
    • Roberts, E.A.1    Kohno, Y.2    Pastrakuljic, A.3    Tang, B.K.4    Kalow, W.5
  • 20
    • 0028237729 scopus 로고
    • Interindividual variation in human liver cytochrome P450 enzymes involved in oxidation of drugs, carcinogens and toxic chemicals: Studies with liver microsomes of 30 Japanese and 30 Caucasians
    • 20. Shimada T, Yamazaki H, Mimura M, Inui Y and Guengerich PF, Interindividual variation in human liver cytochrome P450 enzymes involved in oxidation of drugs, carcinogens and toxic chemicals: Studies with liver microsomes of 30 Japanese and 30 Caucasians. J Pharmacol Exp Ther 270: 414-423, 1994.
    • (1994) J Pharmacol Exp Ther , vol.270 , pp. 414-423
    • Shimada, T.1    Yamazaki, H.2    Mimura, M.3    Inui, Y.4    Guengerich, P.F.5
  • 21
    • 0025992864 scopus 로고
    • Oxidation of toxic and carcinogenic chemicals by human cytochrome P450 enzymes
    • 21. Guengerich FP and Shimada T, Oxidation of toxic and carcinogenic chemicals by human cytochrome P450 enzymes. Chem Res Toxicol 4: 391-407, 1991.
    • (1991) Chem Res Toxicol , vol.4 , pp. 391-407
    • Guengerich, F.P.1    Shimada, T.2
  • 22
    • 0023113788 scopus 로고
    • Biotransformation of caffeine, paraxantine, theophylline and theobromine by polycyclic aromatic hydrocarbon-inducibie cytochrome(s) P450 in human liver microsomes
    • 22. Campbell ME, Grant DM, Tadanobu I and Kalow W, Biotransformation of caffeine, paraxantine, theophylline and theobromine by polycyclic aromatic hydrocarbon-inducibie cytochrome(s) P450 in human liver microsomes. Drug Metab Dispos 2: 237-249, 1987.
    • (1987) Drug Metab Dispos , vol.2 , pp. 237-249
    • Campbell, M.E.1    Grant, D.M.2    Tadanobu, I.3    Kalow, W.4
  • 23
    • 0028276386 scopus 로고
    • Complete cDNA sequence of human dioxin-inducible mRNA identifies a new gene subfamily of cytochrome P450 that maps to chromosome 2
    • 23. Sutter TR, Tang YM, Hayes CL, Wo Y-YP, Jabs EW, Li X, Yin H, Cody CW and Greenless WF, Complete cDNA sequence of human dioxin-inducible mRNA identifies a new gene subfamily of cytochrome P450 that maps to chromosome 2. J Biol Chem 269: 13092-13099, 1994.
    • (1994) J Biol Chem , vol.269 , pp. 13092-13099
    • Sutter, T.R.1    Tang, Y.M.2    Hayes, C.L.3    Wo, Y-Y.P.4    Jabs, E.W.5    Li, X.6    Yin, H.7    Cody, C.W.8    Greenless, W.F.9


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.