The synthesis of N-aryl androsterone pyrazoles as aromatase inhibitors

Bioorganic and Medicinal Chemistry Letters

Volumn 7, Issue 4, 1997, Pages 403-408

  Li, Shengrong ^a   Parish, Edward J ^a   Webb, Thomas ^a   Brodie, Angela M H ^b  

^a AUBURN UNIVERSITY   (United States)

^b UNIVERSITY OF MARYLAND SCHOOL OF MEDICINE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ANDROSTERONE DERIVATIVE; AROMATASE INHIBITOR;

ARTICLE; CONTROLLED STUDY; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME ACTIVE SITE; ENZYME INHIBITION; FEMALE; HUMAN; HUMAN TISSUE; IN VITRO STUDY; MICROSOME; MOLECULAR MODEL; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; X RAY DIFFRACTION;

EID: 0031576810     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(97)00033-4     Document Type: Article

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12. W(F) = 7.13%.
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