Synthesis and reactivity of pyrrolo[3,2-e]indole: Removal of a N-BOM group from an unactivated indole

Tetrahedron Letters

Volumn 38, Issue 10, 1997, Pages 1673-1676

  Macor, John E ^a,b   Forman, James T ^a   Post, Ronald J ^a   Ryan, Kevin ^a  

^a PFIZER INC   (United States)

^b Astra Arcus USA   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

HETEROCYCLIC COMPOUND; INDOLE DERIVATIVE; PYRROLO[3,2 E]INDOLE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CYCLIZATION; DRUG SYNTHESIS; HYDROGENATION; REACTION ANALYSIS;

EID: 0031562387     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(97)00198-6     Document Type: Article

References (9)

1. 2) Boger, D. L.; Johnson, D. S. Angew Chem., Int. Ed. Engl. 1996, 35, 1439, and references cited therein.
2. 3) Rawal, V. H.; Jones, R. J.; Cava, M. P. J. Org. Chem.., 1987, 52, 19.
3. 4) Lash, T. D.; Bellettini, J. R.; Voiles, S. J. J. Heterocyclic Chem., 1993, 30, 525.
4. 5) Asselin, A. A.; Humber, L. G.; Voith, K.; Metcalf, G. J. Med. Chem., 1986, 29, 648.
5. 6) Wojciechowski, K.; Makosza, M. Synthesis, 1989, 106.
6. 7) (a) Macor, J. E.; Wehner, J. M. Heterocycles, 1993, 35, 349.
7. (b) Makozsa, M.; Danikiewicz, W.; Wojciechowski, K. Liebigs Ann. Chem., 1988, 203.
8. 8) Anderson, H. J.; Groves, J. K. Tetrahedron Let., 1971, 12, 3165.
9. 2: C: 76.90; H, 5.16; N, 17.94. Found: C, 76.74; H, 5.38; N, 17.77.