Amino diol based asymmetric syntheses of a fused benzazepine as a selective D1 dopamine receptor

Organic Process Research and Development

Volumn 1, Issue 5, 1997, Pages 359-364

  Wu, Guangzhong ^a  

^a MERCK RESEARCH LABORATORIES   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 0031484346     PISSN: 10836160     EISSN: None     Source Type: Journal    
DOI: 10.1021/op970105v     Document Type: Article

References (10)

1. (a) Berger, J. G.; Chang, W. K.; Clader, J. W.; Hou, D.; Chipkin, R. E.; McPhail, A. T. J. Med. Chem. 1989, 32, 1913.
2. (b) Chumpradit, S.; Kung, M.; Billings, J. J.; Kung, H. F. J. Med. Chem. 1991, 34, 877.
3. (c) Chipkin, R. E.; Iorio, L. C.; Coffin, V. L.; Mcquade, R. D.; Berger, J. G.; Barnett, A. J. Pharmacol. 1988, 24, 1093.
4. (a) Sedvall, G.; Farde, L.; Stone-Elander, S.; Halldin, C. In Neurobiology of Central D-1 Dopamine receptors; Breese, G. R., Creese, I., Eds.; Plenum Press: New York, 1991; p 1.
5. (b) Stoof, J. C.; Kebabian, J. W. Life Sci. 1984, 35, 2281.
6. Umino, N.; Iwakuma, T.; Itoh, N. Tetrahedron Lett. 1976, 763.
7. Schumacher, D. P.; Murphy, B. L.; Clark, J. E.; Tahbaz, P.; Mann, T. A. J. Org. Chem. 1989, 54, 2242.
8. Coote, S. J.; Davies, S. G.; Middlemiss, D.; Naylor, A. Tetrahedron: Asymmetry 1990, I, 33.
9. Kikugawa, Y.; Ogawa, Y. Chem. Pharm. Bull. 1979, 27, 2405.
10. Munavalli, S.; Bhat, G. A.; Viel, C. Bull. Soc. Chim. Fr. 1966, 10, 3311.