Quantitative structure-activity studies of octopaminergic 2-(arylimino)thiazolidines and oxazolidines against the nervous system of Periplaneta americana L.

Bioorganic and Medicinal Chemistry

Volumn 5, Issue 12, 1997, Pages 2121-2128

  Hirashima, Akinori ^a   Tomita, Jun ^a   Pan, Canping ^a   Taniguchi, Eiji ^a   Eto, Morifusa ^b  

^a KYUSHU UNIVERSITY   (Japan)

^b MIYAKONOJO NATIONAL COLLEGE OF TECHNOLOGY   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

2 (ARYLIMINO)THIAZOLIDINE DERIVATIVE; OCTOPAMINE; THIAZOLIDINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL MODIFICATION; COCKROACH; DRUG CONFORMATION; ENZYME ACTIVATION; NONHUMAN; PARASITOSIS; QUANTITATIVE STRUCTURE ACTIVITY RELATION; REGRESSION ANALYSIS;

ANIMALS; COMPUTER SIMULATION; ENZYME ACTIVATION; IMINES; KINETICS; MODELS, MOLECULAR; NERVOUS SYSTEM; OCTOPAMINE; OXAZOLES; PERIPLANETA; STRUCTURE-ACTIVITY RELATIONSHIP; THIAZOLES;

EID: 0031450773     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0968-0896(97)00136-3     Document Type: Article

References (25)

1. Hirashima, A.; Yoshii, Y.; Eto, M. Agric. Biol. Chem. 1991, 55, 2537.
2. Hirashima, A.; Yoshii, Y.; Eto, M. Pestic. Biochem. Physiol. 1992, 44, 101.
3. Hirashima, A.; Yoshii, Y.; Eto, M. Biosci. Biotech. Biochem. 1992, 56, 1062.
4. Hirashima, A.; Taniguchi, E.; Eto, M. Pestic. Sci. 1995, 43, 311.
5. Hirashima, A.; Tarui, H.; Eto, M. Biosci. Biochem. Biotech. 1994, 55, 1206.
6. Hirashima, A.; Tarui, H.; Taniguchi, E.; Eto, M. Pestic. Biochem. Physiol. 1994, 50, 83.
7. Hirashima, A.; Pan, P.; Katafuchi, Y.; Taniguchi, E.; Eto, M. Nihon Noyaku Gakkaishi (J. Pestic. Sci.) 1996, 21, 329.
8. Stähle, H. In Chronicles of Drug Discovery; Bindra, J. S.; Lednicer, D., Eds.; John Wiley: New York, 1982; Vol. I, pp 87-111.
9. Kamoshita, K. Ph.D. thesis, Faculty of Agriculture 1980, Kyoto University, Japan, 1980.
10. Hansch, C.; Rockwell, S. D.; Jow, P. Y. C.; Leo, A.; Steller, E. E. J. Med. Chem. 1977, 20, 304.
11. Hansch, C.; Leo, A.; Unger, S. H.; Kim, K.-H.; Nikaitani, D.; Lien, E. J. J. Med. Chem. 1973, 16, 1207.
12. Taft, Jr. R. W. In Steric Effects in Organic Chemistry; Newman, M. S., Ed.; John Wiley: New York, 1956; pp 556-675.
13. Unger, S. H.; Hansch, C. Prog. Phys. Org. Chem. 1976, 12, 91.
14. Hancock, C. K.; Meyers, E. A.; Yager, B. J. J. Amer. Chem. Soc. 1961, 83, 4211.
15. Swain, C. G.; Lupton, E. C. J. Amer. Chem. Soc. 1968, 90, 4328.
16. Verloop, A. In Pesticide Chemistry, Human Welfare and the Environment; Miyamoto, J.; Kearney, P. C., Eds.; Pergamon: Oxford, 1983; Vol. 1, pp 339-344.
17. Charton, M. Prog. Phys. Org. Chem. 1981, 13, 119.
18. Taft, Jr. R. W.; Lewis, I. C. J. Amer. Chem. Soc. 1958, 80, 2436.
19. Harmar, A. J.; Horn, A. S. Molec. Pharmacol. 1977, 13, 512.
20. Dekeyser, M. A.; Harrison W. A. Pestic. Sci. 1993, 38, 309.
21. Dekeyser, M. A.; Harrison, W. A.; Taylor, N. J.; Downer, R. G. H. Can. J. Chem. 1995, 73, 853.
22. Hirashima, A.; Pan, C.; Tomita, J.; Kuwano, E.; Taniguchi, E.; Eto, M. Pestic. Biochem. Physiol. 1997, in press.
23. Kahn, S. D., Hehre, W. J. J. Amer. Chem. Soc., 1987, 109, 663.
24. Kearsley, S. K.; Smith, G. M. Tetrahed. Comp. Method. 1992, 3, 615.
25. Masek, B.; Merchant, A.; Matthews, J. J. Med. Chem. 1993, 36, 1230