New 2-hydrazonophenylthioacetamides intermediates in the synthesis of 6-acylamino-3,6-dihydro-2h-1,3,4-thiadiazines

Phosphorus, Sulfur and Silicon and Related Elements

Volumn 126, Issue , 1997, Pages 39-52

  Gil, M J ^a   Reliquet, A ^a   Meslin, J C ^a  

^a Centre National de la Recherche Scientifique   (France)

Author keywords

2 hydrazonophenylacetamides; 2 hydrazonophenylthioacetamides; 3,6 dihydro 2h 1,3,4 thiadiazines

Indexed keywords

EID: 0031373793     PISSN: 10426507     EISSN: None     Source Type: Journal    
DOI: 10.1080/10426509708043544     Document Type: Article

References (46)

1. A. Reliquet, M. J. Gil, F. Reliquet and J. C. Meslin, Sulfur Lett., 16, 1, (1993).
2. M. J. Gil, A. Reliquet, F. Reliquet and J. C. Meslin, Phosphorus, Sulfur and Silicon, 91, 89, (1994).
3. M. J. Gil, A. Reliquet, F. Reliquet and J. C. Meslin, Phosphorus, Sulfur and Silicon, in press.
4. A. Reliquet, R. Besbes, F. Reliquet and J.C. Meslin, Sulfur Lett., 14, 189, (1992).
5. A. Reliquet, R. Besbes, F. Reliquet and J.C. Meslin, Synthesis, 7, 543, (1991).
6. J. P. Pradère, G. Bouet and H. Quiniou, Tetrahedron Lett., 33, 3471, (1972).
7. T. Karakasa and S. Motoki, J. Org. Chem., 43, 4147, (1978).
8. J. P. Guémas, A. Reliquet, F. Reliquet and H. Quiniou, C. R. Acad. Sc. Paris, 288(C), 89, (1979).
9. I. T. Barnish, C. W. G. Fishwick, D. R. Hill and C. Jr. Szantay, Tetrahedron Lett., 33, 4449, (1989).
10. S. V. Usoltseva, G. P. Andronnikova and V. S. Mokrushin, Khimiya Geterorsikticheskikh Soedinii, 4, 435, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); P. K. Bose, Quart. J. Indian Chem. Soc., 1, 51, (1924); H. Beyer, Quart. rep. Sulfur Chem., 5, 177, (1970); A. Neugebauer and H. Fischer, Chem. Ber., 107, 717, (1974); H. Beyer, Chem. Ber., 89, 107, (1956); Y. V. Zachinaev, M. L. Petrov, A. N. Frolkov, V. N. Chistokletov and A. A. Petrov, Zhurnal Organicheskoi Khimii, 16, 938, (1980), (Engl. Transl.: JI of Organic Chem. of USSR. 818, (1980)); R. M. Mohareb, A. Habashi, E. A. Hafez and S. M. Sherif, Arch. Pharm. (Weinheim, Ger.), 320, 776, (1987); D. L. Trepanier, P. E. Krieger, J. H. Mennear and J. N. Eble, J. Med. Chem., 10, 1085, (1967); S. Tadashi and O. Masaki, Yakugaku Zasshi, 75, 1535, (1955), (Engl. Transl.: JI of the pharmaceutical society of Japan, (1955)); A. E. Baydar, G. V. Boyd and P. F. Lindley, J. Chem. Soc., Chem. Commun., 1003, (1981); D. L. Trepanier, W. Reifschneider, W. Shumaker and D. S. Tharpe, J. Org. Chem., 30, 2228, (1965); H. Kristinsson, T. Winkler and M. Mollenkopf, Helv. Chim. Acta. 66, 2714, (1983); D. M. Evans, D. R. Taylor and M. Myers, J. Chem. Soc., Chem. Commun., 1444, (1984); K. Hirai and T. Ishiba, J. Chem. Soc., Chem. Commun., 1318, (1971); P. Molina, A. Arques, I. Cartagena and J. M. Olmos, Synthesis, 518, (1989); G. Seitz, R. Mohr, W. Overheu, R. Allmann and M. Nagel, Angew. Chem. Int. Ed. Engl. 11, 890, (1984); G. Hesse and I. Jorder, Chem. Ber., 85, 924, (1952).
11. S. V. Usoltseva, G. P. Andronnikova and V. S. Mokrushin, Khimiya Geterorsikticheskikh Soedinii, 4, 435, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); P. K. Bose, Quart. J. Indian Chem. Soc., 1, 51, (1924); H. Beyer, Quart. rep. Sulfur Chem., 5, 177, (1970); A. Neugebauer and H. Fischer, Chem. Ber., 107, 717, (1974); H. Beyer, Chem. Ber., 89, 107, (1956); Y. V. Zachinaev, M. L. Petrov, A. N. Frolkov, V. N. Chistokletov and A. A. Petrov, Zhurnal Organicheskoi Khimii, 16, 938, (1980), (Engl. Transl.: JI of Organic Chem. of USSR. 818, (1980)); R. M. Mohareb, A. Habashi, E. A. Hafez and S. M. Sherif, Arch. Pharm. (Weinheim, Ger.), 320, 776, (1987); D. L. Trepanier, P. E. Krieger, J. H. Mennear and J. N. Eble, J. Med. Chem., 10, 1085, (1967); S. Tadashi and O. Masaki, Yakugaku Zasshi, 75, 1535, (1955), (Engl. Transl.: JI of the pharmaceutical society of Japan, (1955)); A. E. Baydar, G. V. Boyd and P. F. Lindley, J. Chem. Soc., Chem. Commun., 1003, (1981); D. L. Trepanier, W. Reifschneider, W. Shumaker and D. S. Tharpe, J. Org. Chem., 30, 2228, (1965); H. Kristinsson, T. Winkler and M. Mollenkopf, Helv. Chim. Acta. 66, 2714, (1983); D. M. Evans, D. R. Taylor and M. Myers, J. Chem. Soc., Chem. Commun., 1444, (1984); K. Hirai and T. Ishiba, J. Chem. Soc., Chem. Commun., 1318, (1971); P. Molina, A. Arques, I. Cartagena and J. M. Olmos, Synthesis, 518, (1989); G. Seitz, R. Mohr, W. Overheu, R. Allmann and M. Nagel, Angew. Chem. Int. Ed. Engl. 11, 890, (1984); G. Hesse and I. Jorder, Chem. Ber., 85, 924, (1952).
12. S. V. Usoltseva, G. P. Andronnikova and V. S. Mokrushin, Khimiya Geterorsikticheskikh Soedinii, 4, 435, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); P. K. Bose, Quart. J. Indian Chem. Soc., 1, 51, (1924); H. Beyer, Quart. rep. Sulfur Chem., 5, 177, (1970); A. Neugebauer and H. Fischer, Chem. Ber., 107, 717, (1974); H. Beyer, Chem. Ber., 89, 107, (1956); Y. V. Zachinaev, M. L. Petrov, A. N. Frolkov, V. N. Chistokletov and A. A. Petrov, Zhurnal Organicheskoi Khimii, 16, 938, (1980), (Engl. Transl.: JI of Organic Chem. of USSR. 818, (1980)); R. M. Mohareb, A. Habashi, E. A. Hafez and S. M. Sherif, Arch. Pharm. (Weinheim, Ger.), 320, 776, (1987); D. L. Trepanier, P. E. Krieger, J. H. Mennear and J. N. Eble, J. Med. Chem., 10, 1085, (1967); S. Tadashi and O. Masaki, Yakugaku Zasshi, 75, 1535, (1955), (Engl. Transl.: JI of the pharmaceutical society of Japan, (1955)); A. E. Baydar, G. V. Boyd and P. F. Lindley, J. Chem. Soc., Chem. Commun., 1003, (1981); D. L. Trepanier, W. Reifschneider, W. Shumaker and D. S. Tharpe, J. Org. Chem., 30, 2228, (1965); H. Kristinsson, T. Winkler and M. Mollenkopf, Helv. Chim. Acta. 66, 2714, (1983); D. M. Evans, D. R. Taylor and M. Myers, J. Chem. Soc., Chem. Commun., 1444, (1984); K. Hirai and T. Ishiba, J. Chem. Soc., Chem. Commun., 1318, (1971); P. Molina, A. Arques, I. Cartagena and J. M. Olmos, Synthesis, 518, (1989); G. Seitz, R. Mohr, W. Overheu, R. Allmann and M. Nagel, Angew. Chem. Int. Ed. Engl. 11, 890, (1984); G. Hesse and I. Jorder, Chem. Ber., 85, 924, (1952).
13. S. V. Usoltseva, G. P. Andronnikova and V. S. Mokrushin, Khimiya Geterorsikticheskikh Soedinii, 4, 435, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); P. K. Bose, Quart. J. Indian Chem. Soc., 1, 51, (1924); H. Beyer, Quart. rep. Sulfur Chem., 5, 177, (1970); A. Neugebauer and H. Fischer, Chem. Ber., 107, 717, (1974); H. Beyer, Chem. Ber., 89, 107, (1956); Y. V. Zachinaev, M. L. Petrov, A. N. Frolkov, V. N. Chistokletov and A. A. Petrov, Zhurnal Organicheskoi Khimii, 16, 938, (1980), (Engl. Transl.: JI of Organic Chem. of USSR. 818, (1980)); R. M. Mohareb, A. Habashi, E. A. Hafez and S. M. Sherif, Arch. Pharm. (Weinheim, Ger.), 320, 776, (1987); D. L. Trepanier, P. E. Krieger, J. H. Mennear and J. N. Eble, J. Med. Chem., 10, 1085, (1967); S. Tadashi and O. Masaki, Yakugaku Zasshi, 75, 1535, (1955), (Engl. Transl.: JI of the pharmaceutical society of Japan, (1955)); A. E. Baydar, G. V. Boyd and P. F. Lindley, J. Chem. Soc., Chem. Commun., 1003, (1981); D. L. Trepanier, W. Reifschneider, W. Shumaker and D. S. Tharpe, J. Org. Chem., 30, 2228, (1965); H. Kristinsson, T. Winkler and M. Mollenkopf, Helv. Chim. Acta. 66, 2714, (1983); D. M. Evans, D. R. Taylor and M. Myers, J. Chem. Soc., Chem. Commun., 1444, (1984); K. Hirai and T. Ishiba, J. Chem. Soc., Chem. Commun., 1318, (1971); P. Molina, A. Arques, I. Cartagena and J. M. Olmos, Synthesis, 518, (1989); G. Seitz, R. Mohr, W. Overheu, R. Allmann and M. Nagel, Angew. Chem. Int. Ed. Engl. 11, 890, (1984); G. Hesse and I. Jorder, Chem. Ber., 85, 924, (1952).
14. S. V. Usoltseva, G. P. Andronnikova and V. S. Mokrushin, Khimiya Geterorsikticheskikh Soedinii, 4, 435, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); P. K. Bose, Quart. J. Indian Chem. Soc., 1, 51, (1924); H. Beyer, Quart. rep. Sulfur Chem., 5, 177, (1970); A. Neugebauer and H. Fischer, Chem. Ber., 107, 717, (1974); H. Beyer, Chem. Ber., 89, 107, (1956); Y. V. Zachinaev, M. L. Petrov, A. N. Frolkov, V. N. Chistokletov and A. A. Petrov, Zhurnal Organicheskoi Khimii, 16, 938, (1980), (Engl. Transl.: JI of Organic Chem. of USSR. 818, (1980)); R. M. Mohareb, A. Habashi, E. A. Hafez and S. M. Sherif, Arch. Pharm. (Weinheim, Ger.), 320, 776, (1987); D. L. Trepanier, P. E. Krieger, J. H. Mennear and J. N. Eble, J. Med. Chem., 10, 1085, (1967); S. Tadashi and O. Masaki, Yakugaku Zasshi, 75, 1535, (1955), (Engl. Transl.: JI of the pharmaceutical society of Japan, (1955)); A. E. Baydar, G. V. Boyd and P. F. Lindley, J. Chem. Soc., Chem. Commun., 1003, (1981); D. L. Trepanier, W. Reifschneider, W. Shumaker and D. S. Tharpe, J. Org. Chem., 30, 2228, (1965); H. Kristinsson, T. Winkler and M. Mollenkopf, Helv. Chim. Acta. 66, 2714, (1983); D. M. Evans, D. R. Taylor and M. Myers, J. Chem. Soc., Chem. Commun., 1444, (1984); K. Hirai and T. Ishiba, J. Chem. Soc., Chem. Commun., 1318, (1971); P. Molina, A. Arques, I. Cartagena and J. M. Olmos, Synthesis, 518, (1989); G. Seitz, R. Mohr, W. Overheu, R. Allmann and M. Nagel, Angew. Chem. Int. Ed. Engl. 11, 890, (1984); G. Hesse and I. Jorder, Chem. Ber., 85, 924, (1952).
15. S. V. Usoltseva, G. P. Andronnikova and V. S. Mokrushin, Khimiya Geterorsikticheskikh Soedinii, 4, 435, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); P. K. Bose, Quart. J. Indian Chem. Soc., 1, 51, (1924); H. Beyer, Quart. rep. Sulfur Chem., 5, 177, (1970); A. Neugebauer and H. Fischer, Chem. Ber., 107, 717, (1974); H. Beyer, Chem. Ber., 89, 107, (1956); Y. V. Zachinaev, M. L. Petrov, A. N. Frolkov, V. N. Chistokletov and A. A. Petrov, Zhurnal Organicheskoi Khimii, 16, 938, (1980), (Engl. Transl.: JI of Organic Chem. of USSR. 818, (1980)); R. M. Mohareb, A. Habashi, E. A. Hafez and S. M. Sherif, Arch. Pharm. (Weinheim, Ger.), 320, 776, (1987); D. L. Trepanier, P. E. Krieger, J. H. Mennear and J. N. Eble, J. Med. Chem., 10, 1085, (1967); S. Tadashi and O. Masaki, Yakugaku Zasshi, 75, 1535, (1955), (Engl. Transl.: JI of the pharmaceutical society of Japan, (1955)); A. E. Baydar, G. V. Boyd and P. F. Lindley, J. Chem. Soc., Chem. Commun., 1003, (1981); D. L. Trepanier, W. Reifschneider, W. Shumaker and D. S. Tharpe, J. Org. Chem., 30, 2228, (1965); H. Kristinsson, T. Winkler and M. Mollenkopf, Helv. Chim. Acta. 66, 2714, (1983); D. M. Evans, D. R. Taylor and M. Myers, J. Chem. Soc., Chem. Commun., 1444, (1984); K. Hirai and T. Ishiba, J. Chem. Soc., Chem. Commun., 1318, (1971); P. Molina, A. Arques, I. Cartagena and J. M. Olmos, Synthesis, 518, (1989); G. Seitz, R. Mohr, W. Overheu, R. Allmann and M. Nagel, Angew. Chem. Int. Ed. Engl. 11, 890, (1984); G. Hesse and I. Jorder, Chem. Ber., 85, 924, (1952).
16. S. V. Usoltseva, G. P. Andronnikova and V. S. Mokrushin, Khimiya Geterorsikticheskikh Soedinii, 4, 435, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); P. K. Bose, Quart. J. Indian Chem. Soc., 1, 51, (1924); H. Beyer, Quart. rep. Sulfur Chem., 5, 177, (1970); A. Neugebauer and H. Fischer, Chem. Ber., 107, 717, (1974); H. Beyer, Chem. Ber., 89, 107, (1956); Y. V. Zachinaev, M. L. Petrov, A. N. Frolkov, V. N. Chistokletov and A. A. Petrov, Zhurnal Organicheskoi Khimii, 16, 938, (1980), (Engl. Transl.: JI of Organic Chem. of USSR. 818, (1980)); R. M. Mohareb, A. Habashi, E. A. Hafez and S. M. Sherif, Arch. Pharm. (Weinheim, Ger.), 320, 776, (1987); D. L. Trepanier, P. E. Krieger, J. H. Mennear and J. N. Eble, J. Med. Chem., 10, 1085, (1967); S. Tadashi and O. Masaki, Yakugaku Zasshi, 75, 1535, (1955), (Engl. Transl.: JI of the pharmaceutical society of Japan, (1955)); A. E. Baydar, G. V. Boyd and P. F. Lindley, J. Chem. Soc., Chem. Commun., 1003, (1981); D. L. Trepanier, W. Reifschneider, W. Shumaker and D. S. Tharpe, J. Org. Chem., 30, 2228, (1965); H. Kristinsson, T. Winkler and M. Mollenkopf, Helv. Chim. Acta. 66, 2714, (1983); D. M. Evans, D. R. Taylor and M. Myers, J. Chem. Soc., Chem. Commun., 1444, (1984); K. Hirai and T. Ishiba, J. Chem. Soc., Chem. Commun., 1318, (1971); P. Molina, A. Arques, I. Cartagena and J. M. Olmos, Synthesis, 518, (1989); G. Seitz, R. Mohr, W. Overheu, R. Allmann and M. Nagel, Angew. Chem. Int. Ed. Engl. 11, 890, (1984); G. Hesse and I. Jorder, Chem. Ber., 85, 924, (1952).
17. S. V. Usoltseva, G. P. Andronnikova and V. S. Mokrushin, Khimiya Geterorsikticheskikh Soedinii, 4, 435, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); P. K. Bose, Quart. J. Indian Chem. Soc., 1, 51, (1924); H. Beyer, Quart. rep. Sulfur Chem., 5, 177, (1970); A. Neugebauer and H. Fischer, Chem. Ber., 107, 717, (1974); H. Beyer, Chem. Ber., 89, 107, (1956); Y. V. Zachinaev, M. L. Petrov, A. N. Frolkov, V. N. Chistokletov and A. A. Petrov, Zhurnal Organicheskoi Khimii, 16, 938, (1980), (Engl. Transl.: JI of Organic Chem. of USSR. 818, (1980)); R. M. Mohareb, A. Habashi, E. A. Hafez and S. M. Sherif, Arch. Pharm. (Weinheim, Ger.), 320, 776, (1987); D. L. Trepanier, P. E. Krieger, J. H. Mennear and J. N. Eble, J. Med. Chem., 10, 1085, (1967); S. Tadashi and O. Masaki, Yakugaku Zasshi, 75, 1535, (1955), (Engl. Transl.: JI of the pharmaceutical society of Japan, (1955)); A. E. Baydar, G. V. Boyd and P. F. Lindley, J. Chem. Soc., Chem. Commun., 1003, (1981); D. L. Trepanier, W. Reifschneider, W. Shumaker and D. S. Tharpe, J. Org. Chem., 30, 2228, (1965); H. Kristinsson, T. Winkler and M. Mollenkopf, Helv. Chim. Acta. 66, 2714, (1983); D. M. Evans, D. R. Taylor and M. Myers, J. Chem. Soc., Chem. Commun., 1444, (1984); K. Hirai and T. Ishiba, J. Chem. Soc., Chem. Commun., 1318, (1971); P. Molina, A. Arques, I. Cartagena and J. M. Olmos, Synthesis, 518, (1989); G. Seitz, R. Mohr, W. Overheu, R. Allmann and M. Nagel, Angew. Chem. Int. Ed. Engl. 11, 890, (1984); G. Hesse and I. Jorder, Chem. Ber., 85, 924, (1952).
18. S. V. Usoltseva, G. P. Andronnikova and V. S. Mokrushin, Khimiya Geterorsikticheskikh Soedinii, 4, 435, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); P. K. Bose, Quart. J. Indian Chem. Soc., 1, 51, (1924); H. Beyer, Quart. rep. Sulfur Chem., 5, 177, (1970); A. Neugebauer and H. Fischer, Chem. Ber., 107, 717, (1974); H. Beyer, Chem. Ber., 89, 107, (1956); Y. V. Zachinaev, M. L. Petrov, A. N. Frolkov, V. N. Chistokletov and A. A. Petrov, Zhurnal Organicheskoi Khimii, 16, 938, (1980), (Engl. Transl.: JI of Organic Chem. of USSR. 818, (1980)); R. M. Mohareb, A. Habashi, E. A. Hafez and S. M. Sherif, Arch. Pharm. (Weinheim, Ger.), 320, 776, (1987); D. L. Trepanier, P. E. Krieger, J. H. Mennear and J. N. Eble, J. Med. Chem., 10, 1085, (1967); S. Tadashi and O. Masaki, Yakugaku Zasshi, 75, 1535, (1955), (Engl. Transl.: JI of the pharmaceutical society of Japan, (1955)); A. E. Baydar, G. V. Boyd and P. F. Lindley, J. Chem. Soc., Chem. Commun., 1003, (1981); D. L. Trepanier, W. Reifschneider, W. Shumaker and D. S. Tharpe, J. Org. Chem., 30, 2228, (1965); H. Kristinsson, T. Winkler and M. Mollenkopf, Helv. Chim. Acta. 66, 2714, (1983); D. M. Evans, D. R. Taylor and M. Myers, J. Chem. Soc., Chem. Commun., 1444, (1984); K. Hirai and T. Ishiba, J. Chem. Soc., Chem. Commun., 1318, (1971); P. Molina, A. Arques, I. Cartagena and J. M. Olmos, Synthesis, 518, (1989); G. Seitz, R. Mohr, W. Overheu, R. Allmann and M. Nagel, Angew. Chem. Int. Ed. Engl. 11, 890, (1984); G. Hesse and I. Jorder, Chem. Ber., 85, 924, (1952).
19. S. V. Usoltseva, G. P. Andronnikova and V. S. Mokrushin, Khimiya Geterorsikticheskikh Soedinii, 4, 435, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); P. K. Bose, Quart. J. Indian Chem. Soc., 1, 51, (1924); H. Beyer, Quart. rep. Sulfur Chem., 5, 177, (1970); A. Neugebauer and H. Fischer, Chem. Ber., 107, 717, (1974); H. Beyer, Chem. Ber., 89, 107, (1956); Y. V. Zachinaev, M. L. Petrov, A. N. Frolkov, V. N. Chistokletov and A. A. Petrov, Zhurnal Organicheskoi Khimii, 16, 938, (1980), (Engl. Transl.: JI of Organic Chem. of USSR. 818, (1980)); R. M. Mohareb, A. Habashi, E. A. Hafez and S. M. Sherif, Arch. Pharm. (Weinheim, Ger.), 320, 776, (1987); D. L. Trepanier, P. E. Krieger, J. H. Mennear and J. N. Eble, J. Med. Chem., 10, 1085, (1967); S. Tadashi and O. Masaki, Yakugaku Zasshi, 75, 1535, (1955), (Engl. Transl.: JI of the pharmaceutical society of Japan, (1955)); A. E. Baydar, G. V. Boyd and P. F. Lindley, J. Chem. Soc., Chem. Commun., 1003, (1981); D. L. Trepanier, W. Reifschneider, W. Shumaker and D. S. Tharpe, J. Org. Chem., 30, 2228, (1965); H. Kristinsson, T. Winkler and M. Mollenkopf, Helv. Chim. Acta. 66, 2714, (1983); D. M. Evans, D. R. Taylor and M. Myers, J. Chem. Soc., Chem. Commun., 1444, (1984); K. Hirai and T. Ishiba, J. Chem. Soc., Chem. Commun., 1318, (1971); P. Molina, A. Arques, I. Cartagena and J. M. Olmos, Synthesis, 518, (1989); G. Seitz, R. Mohr, W. Overheu, R. Allmann and M. Nagel, Angew. Chem. Int. Ed. Engl. 11, 890, (1984); G. Hesse and I. Jorder, Chem. Ber., 85, 924, (1952).
20. S. V. Usoltseva, G. P. Andronnikova and V. S. Mokrushin, Khimiya Geterorsikticheskikh Soedinii, 4, 435, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); P. K. Bose, Quart. J. Indian Chem. Soc., 1, 51, (1924); H. Beyer, Quart. rep. Sulfur Chem., 5, 177, (1970); A. Neugebauer and H. Fischer, Chem. Ber., 107, 717, (1974); H. Beyer, Chem. Ber., 89, 107, (1956); Y. V. Zachinaev, M. L. Petrov, A. N. Frolkov, V. N. Chistokletov and A. A. Petrov, Zhurnal Organicheskoi Khimii, 16, 938, (1980), (Engl. Transl.: JI of Organic Chem. of USSR. 818, (1980)); R. M. Mohareb, A. Habashi, E. A. Hafez and S. M. Sherif, Arch. Pharm. (Weinheim, Ger.), 320, 776, (1987); D. L. Trepanier, P. E. Krieger, J. H. Mennear and J. N. Eble, J. Med. Chem., 10, 1085, (1967); S. Tadashi and O. Masaki, Yakugaku Zasshi, 75, 1535, (1955), (Engl. Transl.: JI of the pharmaceutical society of Japan, (1955)); A. E. Baydar, G. V. Boyd and P. F. Lindley, J. Chem. Soc., Chem. Commun., 1003, (1981); D. L. Trepanier, W. Reifschneider, W. Shumaker and D. S. Tharpe, J. Org. Chem., 30, 2228, (1965); H. Kristinsson, T. Winkler and M. Mollenkopf, Helv. Chim. Acta. 66, 2714, (1983); D. M. Evans, D. R. Taylor and M. Myers, J. Chem. Soc., Chem. Commun., 1444, (1984); K. Hirai and T. Ishiba, J. Chem. Soc., Chem. Commun., 1318, (1971); P. Molina, A. Arques, I. Cartagena and J. M. Olmos, Synthesis, 518, (1989); G. Seitz, R. Mohr, W. Overheu, R. Allmann and M. Nagel, Angew. Chem. Int. Ed. Engl. 11, 890, (1984); G. Hesse and I. Jorder, Chem. Ber., 85, 924, (1952).
21. S. V. Usoltseva, G. P. Andronnikova and V. S. Mokrushin, Khimiya Geterorsikticheskikh Soedinii, 4, 435, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); P. K. Bose, Quart. J. Indian Chem. Soc., 1, 51, (1924); H. Beyer, Quart. rep. Sulfur Chem., 5, 177, (1970); A. Neugebauer and H. Fischer, Chem. Ber., 107, 717, (1974); H. Beyer, Chem. Ber., 89, 107, (1956); Y. V. Zachinaev, M. L. Petrov, A. N. Frolkov, V. N. Chistokletov and A. A. Petrov, Zhurnal Organicheskoi Khimii, 16, 938, (1980), (Engl. Transl.: JI of Organic Chem. of USSR. 818, (1980)); R. M. Mohareb, A. Habashi, E. A. Hafez and S. M. Sherif, Arch. Pharm. (Weinheim, Ger.), 320, 776, (1987); D. L. Trepanier, P. E. Krieger, J. H. Mennear and J. N. Eble, J. Med. Chem., 10, 1085, (1967); S. Tadashi and O. Masaki, Yakugaku Zasshi, 75, 1535, (1955), (Engl. Transl.: JI of the pharmaceutical society of Japan, (1955)); A. E. Baydar, G. V. Boyd and P. F. Lindley, J. Chem. Soc., Chem. Commun., 1003, (1981); D. L. Trepanier, W. Reifschneider, W. Shumaker and D. S. Tharpe, J. Org. Chem., 30, 2228, (1965); H. Kristinsson, T. Winkler and M. Mollenkopf, Helv. Chim. Acta. 66, 2714, (1983); D. M. Evans, D. R. Taylor and M. Myers, J. Chem. Soc., Chem. Commun., 1444, (1984); K. Hirai and T. Ishiba, J. Chem. Soc., Chem. Commun., 1318, (1971); P. Molina, A. Arques, I. Cartagena and J. M. Olmos, Synthesis, 518, (1989); G. Seitz, R. Mohr, W. Overheu, R. Allmann and M. Nagel, Angew. Chem. Int. Ed. Engl. 11, 890, (1984); G. Hesse and I. Jorder, Chem. Ber., 85, 924, (1952).
22. S. V. Usoltseva, G. P. Andronnikova and V. S. Mokrushin, Khimiya Geterorsikticheskikh Soedinii, 4, 435, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); P. K. Bose, Quart. J. Indian Chem. Soc., 1, 51, (1924); H. Beyer, Quart. rep. Sulfur Chem., 5, 177, (1970); A. Neugebauer and H. Fischer, Chem. Ber., 107, 717, (1974); H. Beyer, Chem. Ber., 89, 107, (1956); Y. V. Zachinaev, M. L. Petrov, A. N. Frolkov, V. N. Chistokletov and A. A. Petrov, Zhurnal Organicheskoi Khimii, 16, 938, (1980), (Engl. Transl.: JI of Organic Chem. of USSR. 818, (1980)); R. M. Mohareb, A. Habashi, E. A. Hafez and S. M. Sherif, Arch. Pharm. (Weinheim, Ger.), 320, 776, (1987); D. L. Trepanier, P. E. Krieger, J. H. Mennear and J. N. Eble, J. Med. Chem., 10, 1085, (1967); S. Tadashi and O. Masaki, Yakugaku Zasshi, 75, 1535, (1955), (Engl. Transl.: JI of the pharmaceutical society of Japan, (1955)); A. E. Baydar, G. V. Boyd and P. F. Lindley, J. Chem. Soc., Chem. Commun., 1003, (1981); D. L. Trepanier, W. Reifschneider, W. Shumaker and D. S. Tharpe, J. Org. Chem., 30, 2228, (1965); H. Kristinsson, T. Winkler and M. Mollenkopf, Helv. Chim. Acta. 66, 2714, (1983); D. M. Evans, D. R. Taylor and M. Myers, J. Chem. Soc., Chem. Commun., 1444, (1984); K. Hirai and T. Ishiba, J. Chem. Soc., Chem. Commun., 1318, (1971); P. Molina, A. Arques, I. Cartagena and J. M. Olmos, Synthesis, 518, (1989); G. Seitz, R. Mohr, W. Overheu, R. Allmann and M. Nagel, Angew. Chem. Int. Ed. Engl. 11, 890, (1984); G. Hesse and I. Jorder, Chem. Ber., 85, 924, (1952).
23. S. V. Usoltseva, G. P. Andronnikova and V. S. Mokrushin, Khimiya Geterorsikticheskikh Soedinii, 4, 435, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); P. K. Bose, Quart. J. Indian Chem. Soc., 1, 51, (1924); H. Beyer, Quart. rep. Sulfur Chem., 5, 177, (1970); A. Neugebauer and H. Fischer, Chem. Ber., 107, 717, (1974); H. Beyer, Chem. Ber., 89, 107, (1956); Y. V. Zachinaev, M. L. Petrov, A. N. Frolkov, V. N. Chistokletov and A. A. Petrov, Zhurnal Organicheskoi Khimii, 16, 938, (1980), (Engl. Transl.: JI of Organic Chem. of USSR. 818, (1980)); R. M. Mohareb, A. Habashi, E. A. Hafez and S. M. Sherif, Arch. Pharm. (Weinheim, Ger.), 320, 776, (1987); D. L. Trepanier, P. E. Krieger, J. H. Mennear and J. N. Eble, J. Med. Chem., 10, 1085, (1967); S. Tadashi and O. Masaki, Yakugaku Zasshi, 75, 1535, (1955), (Engl. Transl.: JI of the pharmaceutical society of Japan, (1955)); A. E. Baydar, G. V. Boyd and P. F. Lindley, J. Chem. Soc., Chem. Commun., 1003, (1981); D. L. Trepanier, W. Reifschneider, W. Shumaker and D. S. Tharpe, J. Org. Chem., 30, 2228, (1965); H. Kristinsson, T. Winkler and M. Mollenkopf, Helv. Chim. Acta. 66, 2714, (1983); D. M. Evans, D. R. Taylor and M. Myers, J. Chem. Soc., Chem. Commun., 1444, (1984); K. Hirai and T. Ishiba, J. Chem. Soc., Chem. Commun., 1318, (1971); P. Molina, A. Arques, I. Cartagena and J. M. Olmos, Synthesis, 518, (1989); G. Seitz, R. Mohr, W. Overheu, R. Allmann and M. Nagel, Angew. Chem. Int. Ed. Engl. 11, 890, (1984); G. Hesse and I. Jorder, Chem. Ber., 85, 924, (1952).
24. S. V. Usoltseva, G. P. Andronnikova and V. S. Mokrushin, Khimiya Geterorsikticheskikh Soedinii, 4, 435, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); P. K. Bose, Quart. J. Indian Chem. Soc., 1, 51, (1924); H. Beyer, Quart. rep. Sulfur Chem., 5, 177, (1970); A. Neugebauer and H. Fischer, Chem. Ber., 107, 717, (1974); H. Beyer, Chem. Ber., 89, 107, (1956); Y. V. Zachinaev, M. L. Petrov, A. N. Frolkov, V. N. Chistokletov and A. A. Petrov, Zhurnal Organicheskoi Khimii, 16, 938, (1980), (Engl. Transl.: JI of Organic Chem. of USSR. 818, (1980)); R. M. Mohareb, A. Habashi, E. A. Hafez and S. M. Sherif, Arch. Pharm. (Weinheim, Ger.), 320, 776, (1987); D. L. Trepanier, P. E. Krieger, J. H. Mennear and J. N. Eble, J. Med. Chem., 10, 1085, (1967); S. Tadashi and O. Masaki, Yakugaku Zasshi, 75, 1535, (1955), (Engl. Transl.: JI of the pharmaceutical society of Japan, (1955)); A. E. Baydar, G. V. Boyd and P. F. Lindley, J. Chem. Soc., Chem. Commun., 1003, (1981); D. L. Trepanier, W. Reifschneider, W. Shumaker and D. S. Tharpe, J. Org. Chem., 30, 2228, (1965); H. Kristinsson, T. Winkler and M. Mollenkopf, Helv. Chim. Acta. 66, 2714, (1983); D. M. Evans, D. R. Taylor and M. Myers, J. Chem. Soc., Chem. Commun., 1444, (1984); K. Hirai and T. Ishiba, J. Chem. Soc., Chem. Commun., 1318, (1971); P. Molina, A. Arques, I. Cartagena and J. M. Olmos, Synthesis, 518, (1989); G. Seitz, R. Mohr, W. Overheu, R. Allmann and M. Nagel, Angew. Chem. Int. Ed. Engl. 11, 890, (1984); G. Hesse and I. Jorder, Chem. Ber., 85, 924, (1952).
25. S. V. Usoltseva, G. P. Andronnikova and V. S. Mokrushin, Khimiya Geterorsikticheskikh Soedinii, 4, 435, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); P. K. Bose, Quart. J. Indian Chem. Soc., 1, 51, (1924); H. Beyer, Quart. rep. Sulfur Chem., 5, 177, (1970); A. Neugebauer and H. Fischer, Chem. Ber., 107, 717, (1974); H. Beyer, Chem. Ber., 89, 107, (1956); Y. V. Zachinaev, M. L. Petrov, A. N. Frolkov, V. N. Chistokletov and A. A. Petrov, Zhurnal Organicheskoi Khimii, 16, 938, (1980), (Engl. Transl.: JI of Organic Chem. of USSR. 818, (1980)); R. M. Mohareb, A. Habashi, E. A. Hafez and S. M. Sherif, Arch. Pharm. (Weinheim, Ger.), 320, 776, (1987); D. L. Trepanier, P. E. Krieger, J. H. Mennear and J. N. Eble, J. Med. Chem., 10, 1085, (1967); S. Tadashi and O. Masaki, Yakugaku Zasshi, 75, 1535, (1955), (Engl. Transl.: JI of the pharmaceutical society of Japan, (1955)); A. E. Baydar, G. V. Boyd and P. F. Lindley, J. Chem. Soc., Chem. Commun., 1003, (1981); D. L. Trepanier, W. Reifschneider, W. Shumaker and D. S. Tharpe, J. Org. Chem., 30, 2228, (1965); H. Kristinsson, T. Winkler and M. Mollenkopf, Helv. Chim. Acta. 66, 2714, (1983); D. M. Evans, D. R. Taylor and M. Myers, J. Chem. Soc., Chem. Commun., 1444, (1984); K. Hirai and T. Ishiba, J. Chem. Soc., Chem. Commun., 1318, (1971); P. Molina, A. Arques, I. Cartagena and J. M. Olmos, Synthesis, 518, (1989); G. Seitz, R. Mohr, W. Overheu, R. Allmann and M. Nagel, Angew. Chem. Int. Ed. Engl. 11, 890, (1984); G. Hesse and I. Jorder, Chem. Ber., 85, 924, (1952).
26. S. V. Usoltseva, G. P. Andronnikova and V. S. Mokrushin, Khimiya Geterorsikticheskikh Soedinii, 4, 435, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); P. K. Bose, Quart. J. Indian Chem. Soc., 1, 51, (1924); H. Beyer, Quart. rep. Sulfur Chem., 5, 177, (1970); A. Neugebauer and H. Fischer, Chem. Ber., 107, 717, (1974); H. Beyer, Chem. Ber., 89, 107, (1956); Y. V. Zachinaev, M. L. Petrov, A. N. Frolkov, V. N. Chistokletov and A. A. Petrov, Zhurnal Organicheskoi Khimii, 16, 938, (1980), (Engl. Transl.: JI of Organic Chem. of USSR. 818, (1980)); R. M. Mohareb, A. Habashi, E. A. Hafez and S. M. Sherif, Arch. Pharm. (Weinheim, Ger.), 320, 776, (1987); D. L. Trepanier, P. E. Krieger, J. H. Mennear and J. N. Eble, J. Med. Chem., 10, 1085, (1967); S. Tadashi and O. Masaki, Yakugaku Zasshi, 75, 1535, (1955), (Engl. Transl.: JI of the pharmaceutical society of Japan, (1955)); A. E. Baydar, G. V. Boyd and P. F. Lindley, J. Chem. Soc., Chem. Commun., 1003, (1981); D. L. Trepanier, W. Reifschneider, W. Shumaker and D. S. Tharpe, J. Org. Chem., 30, 2228, (1965); H. Kristinsson, T. Winkler and M. Mollenkopf, Helv. Chim. Acta. 66, 2714, (1983); D. M. Evans, D. R. Taylor and M. Myers, J. Chem. Soc., Chem. Commun., 1444, (1984); K. Hirai and T. Ishiba, J. Chem. Soc., Chem. Commun., 1318, (1971); P. Molina, A. Arques, I. Cartagena and J. M. Olmos, Synthesis, 518, (1989); G. Seitz, R. Mohr, W. Overheu, R. Allmann and M. Nagel, Angew. Chem. Int. Ed. Engl. 11, 890, (1984); G. Hesse and I. Jorder, Chem. Ber., 85, 924, (1952).
27. S. V. Usoltseva, G. P. Andronnikova and V. S. Mokrushin, Khimiya Geterorsikticheskikh Soedinii, 4, 435, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); P. K. Bose, Quart. J. Indian Chem. Soc., 1, 51, (1924); H. Beyer, Quart. rep. Sulfur Chem., 5, 177, (1970); A. Neugebauer and H. Fischer, Chem. Ber., 107, 717, (1974); H. Beyer, Chem. Ber., 89, 107, (1956); Y. V. Zachinaev, M. L. Petrov, A. N. Frolkov, V. N. Chistokletov and A. A. Petrov, Zhurnal Organicheskoi Khimii, 16, 938, (1980), (Engl. Transl.: JI of Organic Chem. of USSR. 818, (1980)); R. M. Mohareb, A. Habashi, E. A. Hafez and S. M. Sherif, Arch. Pharm. (Weinheim, Ger.), 320, 776, (1987); D. L. Trepanier, P. E. Krieger, J. H. Mennear and J. N. Eble, J. Med. Chem., 10, 1085, (1967); S. Tadashi and O. Masaki, Yakugaku Zasshi, 75, 1535, (1955), (Engl. Transl.: JI of the pharmaceutical society of Japan, (1955)); A. E. Baydar, G. V. Boyd and P. F. Lindley, J. Chem. Soc., Chem. Commun., 1003, (1981); D. L. Trepanier, W. Reifschneider, W. Shumaker and D. S. Tharpe, J. Org. Chem., 30, 2228, (1965); H. Kristinsson, T. Winkler and M. Mollenkopf, Helv. Chim. Acta. 66, 2714, (1983); D. M. Evans, D. R. Taylor and M. Myers, J. Chem. Soc., Chem. Commun., 1444, (1984); K. Hirai and T. Ishiba, J. Chem. Soc., Chem. Commun., 1318, (1971); P. Molina, A. Arques, I. Cartagena and J. M. Olmos, Synthesis, 518, (1989); G. Seitz, R. Mohr, W. Overheu, R. Allmann and M. Nagel, Angew. Chem. Int. Ed. Engl. 11, 890, (1984); G. Hesse and I. Jorder, Chem. Ber., 85, 924, (1952).
28. S. V. Usoltseva, G. P. Andronnikova and V. S. Mokrushin, Khimiya Geterorsikticheskikh Soedinii, 4, 435, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); P. K. Bose, Quart. J. Indian Chem. Soc., 1, 51, (1924); H. Beyer, Quart. rep. Sulfur Chem., 5, 177, (1970); A. Neugebauer and H. Fischer, Chem. Ber., 107, 717, (1974); H. Beyer, Chem. Ber., 89, 107, (1956); Y. V. Zachinaev, M. L. Petrov, A. N. Frolkov, V. N. Chistokletov and A. A. Petrov, Zhurnal Organicheskoi Khimii, 16, 938, (1980), (Engl. Transl.: JI of Organic Chem. of USSR. 818, (1980)); R. M. Mohareb, A. Habashi, E. A. Hafez and S. M. Sherif, Arch. Pharm. (Weinheim, Ger.), 320, 776, (1987); D. L. Trepanier, P. E. Krieger, J. H. Mennear and J. N. Eble, J. Med. Chem., 10, 1085, (1967); S. Tadashi and O. Masaki, Yakugaku Zasshi, 75, 1535, (1955), (Engl. Transl.: JI of the pharmaceutical society of Japan, (1955)); A. E. Baydar, G. V. Boyd and P. F. Lindley, J. Chem. Soc., Chem. Commun., 1003, (1981); D. L. Trepanier, W. Reifschneider, W. Shumaker and D. S. Tharpe, J. Org. Chem., 30, 2228, (1965); H. Kristinsson, T. Winkler and M. Mollenkopf, Helv. Chim. Acta. 66, 2714, (1983); D. M. Evans, D. R. Taylor and M. Myers, J. Chem. Soc., Chem. Commun., 1444, (1984); K. Hirai and T. Ishiba, J. Chem. Soc., Chem. Commun., 1318, (1971); P. Molina, A. Arques, I. Cartagena and J. M. Olmos, Synthesis, 518, (1989); G. Seitz, R. Mohr, W. Overheu, R. Allmann and M. Nagel, Angew. Chem. Int. Ed. Engl. 11, 890, (1984); G. Hesse and I. Jorder, Chem. Ber., 85, 924, (1952).
29. S. V. Usoltseva, G. P. Andronnikova and V. S. Mokrushin, Khimiya Geterorsikticheskikh Soedinii, 4, 435, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); P. K. Bose, Quart. J. Indian Chem. Soc., 1, 51, (1924); H. Beyer, Quart. rep. Sulfur Chem., 5, 177, (1970); A. Neugebauer and H. Fischer, Chem. Ber., 107, 717, (1974); H. Beyer, Chem. Ber., 89, 107, (1956); Y. V. Zachinaev, M. L. Petrov, A. N. Frolkov, V. N. Chistokletov and A. A. Petrov, Zhurnal Organicheskoi Khimii, 16, 938, (1980), (Engl. Transl.: JI of Organic Chem. of USSR. 818, (1980)); R. M. Mohareb, A. Habashi, E. A. Hafez and S. M. Sherif, Arch. Pharm. (Weinheim, Ger.), 320, 776, (1987); D. L. Trepanier, P. E. Krieger, J. H. Mennear and J. N. Eble, J. Med. Chem., 10, 1085, (1967); S. Tadashi and O. Masaki, Yakugaku Zasshi, 75, 1535, (1955), (Engl. Transl.: JI of the pharmaceutical society of Japan, (1955)); A. E. Baydar, G. V. Boyd and P. F. Lindley, J. Chem. Soc., Chem. Commun., 1003, (1981); D. L. Trepanier, W. Reifschneider, W. Shumaker and D. S. Tharpe, J. Org. Chem., 30, 2228, (1965); H. Kristinsson, T. Winkler and M. Mollenkopf, Helv. Chim. Acta. 66, 2714, (1983); D. M. Evans, D. R. Taylor and M. Myers, J. Chem. Soc., Chem. Commun., 1444, (1984); K. Hirai and T. Ishiba, J. Chem. Soc., Chem. Commun., 1318, (1971); P. Molina, A. Arques, I. Cartagena and J. M. Olmos, Synthesis, 518, (1989); G. Seitz, R. Mohr, W. Overheu, R. Allmann and M. Nagel, Angew. Chem. Int. Ed. Engl. 11, 890, (1984); G. Hesse and I. Jorder, Chem. Ber., 85, 924, (1952).
30. Y. Kamitori, M. Hojo, R. Masuda, Y. Kawamura and T. Numai, Synthesis, 491, (1990).
31. A. P. Novikova, N. M. Perova and O. N. Chupakhin, Khimiya Geterotsiklicheskikh Soedinii, 11, 1443, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); D. Brown, R. B. Hargreaves, B. J. Mc Loughlin and S. D. Mills, Eur. Pat. 80,296, CA, 100, 22672, (1984); N. Yoshida, K. Tanaka, Y. Iizuka, K. Wachi, T. Nishimura and H. Yasuda, (Sankyo Co., Ltd), Jpn. Kokai Tokkyo Koho JP 7,488,889, CA, 82, 57744, (1975); J. Dizon and D. H. Robinson, (Fisons PLC), Brit. UK Pat. Appl. GB 2,179,655, CA, 108, 37839, (1988); W. Thorwart, U. Gebert, R. Schleyerbach and R. Bartlett, (Hoechst A.-G.), Ger. Offen. DE. 3,702,757, CA, 110, 8223, (1988); W. Thorwart, U. Gebert, R. Schleyerbach and R. Barlett, (Hoechst A.-G.), Ger. Offen. DE. 3,702,756, CA, 109, 170466, (1988); W. D. Jones and F. P. Miller, (Richardson-Merrell Inc.), Ger. Offen. DE. 3,031,703,
32. A. P. Novikova, N. M. Perova and O. N. Chupakhin, Khimiya Geterotsiklicheskikh Soedinii, 11, 1443, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); D. Brown, R. B. Hargreaves, B. J. Mc Loughlin and S. D. Mills, Eur. Pat. 80,296, CA, 100, 22672, (1984); N. Yoshida, K. Tanaka, Y. Iizuka, K. Wachi, T. Nishimura and H. Yasuda, (Sankyo Co., Ltd), Jpn. Kokai Tokkyo Koho JP 7,488,889, CA, 82, 57744, (1975); J. Dizon and D. H. Robinson, (Fisons PLC), Brit. UK Pat. Appl. GB 2,179,655, CA, 108, 37839, (1988); W. Thorwart, U. Gebert, R. Schleyerbach and R. Bartlett, (Hoechst A.-G.), Ger. Offen. DE. 3,702,757, CA, 110, 8223, (1988); W. Thorwart, U. Gebert, R. Schleyerbach and R. Barlett, (Hoechst A.-G.), Ger. Offen. DE. 3,702,756, CA, 109, 170466, (1988); W. D. Jones and F. P. Miller, (Richardson-Merrell Inc.), Ger. Offen. DE. 3,031,703,
33. A. P. Novikova, N. M. Perova and O. N. Chupakhin, Khimiya Geterotsiklicheskikh Soedinii, 11, 1443, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); D. Brown, R. B. Hargreaves, B. J. Mc Loughlin and S. D. Mills, Eur. Pat. 80,296, CA, 100, 22672, (1984); N. Yoshida, K. Tanaka, Y. Iizuka, K. Wachi, T. Nishimura and H. Yasuda, (Sankyo Co., Ltd), Jpn. Kokai Tokkyo Koho JP 7,488,889, CA, 82, 57744, (1975); J. Dizon and D. H. Robinson, (Fisons PLC), Brit. UK Pat. Appl. GB 2,179,655, CA, 108, 37839, (1988); W. Thorwart, U. Gebert, R. Schleyerbach and R. Bartlett, (Hoechst A.-G.), Ger. Offen. DE. 3,702,757, CA, 110, 8223, (1988); W. Thorwart, U. Gebert, R. Schleyerbach and R. Barlett, (Hoechst A.-G.), Ger. Offen. DE. 3,702,756, CA, 109, 170466, (1988); W. D. Jones and F. P. Miller, (Richardson-Merrell Inc.), Ger. Offen. DE. 3,031,703,
34. A. P. Novikova, N. M. Perova and O. N. Chupakhin, Khimiya Geterotsiklicheskikh Soedinii, 11, 1443, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); D. Brown, R. B. Hargreaves, B. J. Mc Loughlin and S. D. Mills, Eur. Pat. 80,296, CA, 100, 22672, (1984); N. Yoshida, K. Tanaka, Y. Iizuka, K. Wachi, T. Nishimura and H. Yasuda, (Sankyo Co., Ltd), Jpn. Kokai Tokkyo Koho JP 7,488,889, CA, 82, 57744, (1975); J. Dizon and D. H. Robinson, (Fisons PLC), Brit. UK Pat. Appl. GB 2,179,655, CA, 108, 37839, (1988); W. Thorwart, U. Gebert, R. Schleyerbach and R. Bartlett, (Hoechst A.-G.), Ger. Offen. DE. 3,702,757, CA, 110, 8223, (1988); W. Thorwart, U. Gebert, R. Schleyerbach and R. Barlett, (Hoechst A.-G.), Ger. Offen. DE. 3,702,756, CA, 109, 170466, (1988); W. D. Jones and F. P. Miller, (Richardson-Merrell Inc.), Ger. Offen. DE. 3,031,703,
35. A. P. Novikova, N. M. Perova and O. N. Chupakhin, Khimiya Geterotsiklicheskikh Soedinii, 11, 1443, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); D. Brown, R. B. Hargreaves, B. J. Mc Loughlin and S. D. Mills, Eur. Pat. 80,296, CA, 100, 22672, (1984); N. Yoshida, K. Tanaka, Y. Iizuka, K. Wachi, T. Nishimura and H. Yasuda, (Sankyo Co., Ltd), Jpn. Kokai Tokkyo Koho JP 7,488,889, CA, 82, 57744, (1975); J. Dizon and D. H. Robinson, (Fisons PLC), Brit. UK Pat. Appl. GB 2,179,655, CA, 108, 37839, (1988); W. Thorwart, U. Gebert, R. Schleyerbach and R. Bartlett, (Hoechst A.-G.), Ger. Offen. DE. 3,702,757, CA, 110, 8223, (1988); W. Thorwart, U. Gebert, R. Schleyerbach and R. Barlett, (Hoechst A.-G.), Ger. Offen. DE. 3,702,756, CA, 109, 170466, (1988); W. D. Jones and F. P. Miller, (Richardson-Merrell Inc.), Ger. Offen. DE. 3,031,703,
36. A. P. Novikova, N. M. Perova and O. N. Chupakhin, Khimiya Geterotsiklicheskikh Soedinii, 11, 1443, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); D. Brown, R. B. Hargreaves, B. J. Mc Loughlin and S. D. Mills, Eur. Pat. 80,296, CA, 100, 22672, (1984); N. Yoshida, K. Tanaka, Y. Iizuka, K. Wachi, T. Nishimura and H. Yasuda, (Sankyo Co., Ltd), Jpn. Kokai Tokkyo Koho JP 7,488,889, CA, 82, 57744, (1975); J. Dizon and D. H. Robinson, (Fisons PLC), Brit. UK Pat. Appl. GB 2,179,655, CA, 108, 37839, (1988); W. Thorwart, U. Gebert, R. Schleyerbach and R. Bartlett, (Hoechst A.-G.), Ger. Offen. DE. 3,702,757, CA, 110, 8223, (1988); W. Thorwart, U. Gebert, R. Schleyerbach and R. Barlett, (Hoechst A.-G.), Ger. Offen. DE. 3,702,756, CA, 109, 170466, (1988); W. D. Jones and F. P. Miller, (Richardson-Merrell Inc.), Ger. Offen. DE. 3,031,703,
37. A. P. Novikova, N. M. Perova and O. N. Chupakhin, Khimiya Geterotsiklicheskikh Soedinii, 11, 1443, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); D. Brown, R. B. Hargreaves, B. J. Mc Loughlin and S. D. Mills, Eur. Pat. 80,296, CA, 100, 22672, (1984); N. Yoshida, K. Tanaka, Y. Iizuka, K. Wachi, T. Nishimura and H. Yasuda, (Sankyo Co., Ltd), Jpn. Kokai Tokkyo Koho JP 7,488,889, CA, 82, 57744, (1975); J. Dizon and D. H. Robinson, (Fisons PLC), Brit. UK Pat. Appl. GB 2,179,655, CA, 108, 37839, (1988); W. Thorwart, U. Gebert, R. Schleyerbach and R. Bartlett, (Hoechst A.-G.), Ger. Offen. DE. 3,702,757, CA, 110, 8223, (1988); W. Thorwart, U. Gebert, R. Schleyerbach and R. Barlett, (Hoechst A.-G.), Ger. Offen. DE. 3,702,756, CA, 109, 170466, (1988); W. D. Jones and F. P. Miller, (Richardson-Merrell Inc.), Ger. Offen. DE. 3,031,703,
38. A. P. Novikova, N. M. Perova and O. N. Chupakhin, Khimiya Geterotsiklicheskikh Soedinii, 11, 1443, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); D. Brown, R. B. Hargreaves, B. J. Mc Loughlin and S. D. Mills, Eur. Pat. 80,296, CA, 100, 22672, (1984); N. Yoshida, K. Tanaka, Y. Iizuka, K. Wachi, T. Nishimura and H. Yasuda, (Sankyo Co., Ltd), Jpn. Kokai Tokkyo Koho JP 7,488,889, CA, 82, 57744, (1975); J. Dizon and D. H. Robinson, (Fisons PLC), Brit. UK Pat. Appl. GB 2,179,655, CA, 108, 37839, (1988); W. Thorwart, U. Gebert, R. Schleyerbach and R. Bartlett, (Hoechst A.-G.), Ger. Offen. DE. 3,702,757, CA, 110, 8223, (1988); W. Thorwart, U. Gebert, R. Schleyerbach and R. Barlett, (Hoechst A.-G.), Ger. Offen. DE. 3,702,756, CA, 109, 170466, (1988); W. D. Jones and F. P. Miller, (Richardson-Merrell Inc.), Ger. Offen. DE. 3,031,703,
39. A. P. Novikova, N. M. Perova and O. N. Chupakhin, Khimiya Geterotsiklicheskikh Soedinii, 11, 1443, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); D. Brown, R. B. Hargreaves, B. J. Mc Loughlin and S. D. Mills, Eur. Pat. 80,296, CA, 100, 22672, (1984); N. Yoshida, K. Tanaka, Y. Iizuka, K. Wachi, T. Nishimura and H. Yasuda, (Sankyo Co., Ltd), Jpn. Kokai Tokkyo Koho JP 7,488,889, CA, 82, 57744, (1975); J. Dizon and D. H. Robinson, (Fisons PLC), Brit. UK Pat. Appl. GB 2,179,655, CA, 108, 37839, (1988); W. Thorwart, U. Gebert, R. Schleyerbach and R. Bartlett, (Hoechst A.-G.), Ger. Offen. DE. 3,702,757, CA, 110, 8223, (1988); W. Thorwart, U. Gebert, R. Schleyerbach and R. Barlett, (Hoechst A.-G.), Ger. Offen. DE. 3,702,756, CA, 109, 170466, (1988); W. D. Jones and F. P. Miller, (Richardson-Merrell Inc.), Ger. Offen. DE. 3,031,703,
40. A. P. Novikova, N. M. Perova and O. N. Chupakhin, Khimiya Geterotsiklicheskikh Soedinii, 11, 1443, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); D. Brown, R. B. Hargreaves, B. J. Mc Loughlin and S. D. Mills, Eur. Pat. 80,296, CA, 100, 22672, (1984); N. Yoshida, K. Tanaka, Y. Iizuka, K. Wachi, T. Nishimura and H. Yasuda, (Sankyo Co., Ltd), Jpn. Kokai Tokkyo Koho JP 7,488,889, CA, 82, 57744, (1975); J. Dizon and D. H. Robinson, (Fisons PLC), Brit. UK Pat. Appl. GB 2,179,655, CA, 108, 37839, (1988); W. Thorwart, U. Gebert, R. Schleyerbach and R. Bartlett, (Hoechst A.-G.), Ger. Offen. DE. 3,702,757, CA, 110, 8223, (1988); W. Thorwart, U. Gebert, R. Schleyerbach and R. Barlett, (Hoechst A.-G.), Ger. Offen. DE. 3,702,756, CA, 109, 170466, (1988); W. D. Jones and F. P. Miller, (Richardson-Merrell Inc.), Ger. Offen. DE. 3,031,703,
41. A. P. Novikova, N. M. Perova and O. N. Chupakhin, Khimiya Geterotsiklicheskikh Soedinii, 11, 1443, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); D. Brown, R. B. Hargreaves, B. J. Mc Loughlin and S. D. Mills, Eur. Pat. 80,296, CA, 100, 22672, (1984); N. Yoshida, K. Tanaka, Y. Iizuka, K. Wachi, T. Nishimura and H. Yasuda, (Sankyo Co., Ltd), Jpn. Kokai Tokkyo Koho JP 7,488,889, CA, 82, 57744, (1975); J. Dizon and D. H. Robinson, (Fisons PLC), Brit. UK Pat. Appl. GB 2,179,655, CA, 108, 37839, (1988); W. Thorwart, U. Gebert, R. Schleyerbach and R. Bartlett, (Hoechst A.-G.), Ger. Offen. DE. 3,702,757, CA, 110, 8223, (1988); W. Thorwart, U. Gebert, R. Schleyerbach and R. Barlett, (Hoechst A.-G.), Ger. Offen. DE. 3,702,756, CA, 109, 170466, (1988); W. D. Jones and F. P. Miller, (Richardson-Merrell Inc.), Ger. Offen. DE. 3,031,703,
42. A. P. Novikova, N. M. Perova and O. N. Chupakhin, Khimiya Geterotsiklicheskikh Soedinii, 11, 1443, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); D. Brown, R. B. Hargreaves, B. J. Mc Loughlin and S. D. Mills, Eur. Pat. 80,296, CA, 100, 22672, (1984); N. Yoshida, K. Tanaka, Y. Iizuka, K. Wachi, T. Nishimura and H. Yasuda, (Sankyo Co., Ltd), Jpn. Kokai Tokkyo Koho JP 7,488,889, CA, 82, 57744, (1975); J. Dizon and D. H. Robinson, (Fisons PLC), Brit. UK Pat. Appl. GB 2,179,655, CA, 108, 37839, (1988); W. Thorwart, U. Gebert, R. Schleyerbach and R. Bartlett, (Hoechst A.-G.), Ger. Offen. DE. 3,702,757, CA, 110, 8223, (1988); W. Thorwart, U. Gebert, R. Schleyerbach and R. Barlett, (Hoechst A.-G.), Ger. Offen. DE. 3,702,756, CA, 109, 170466, (1988); W. D. Jones and F. P. Miller, (Richardson-Merrell Inc.), Ger. Offen. DE. 3,031,703,
43. A. P. Novikova, N. M. Perova and O. N. Chupakhin, Khimiya Geterotsiklicheskikh Soedinii, 11, 1443, (1991), (Engl. Transl.: Chem. Heterocycl. Comp., (1991)); D. Brown, R. B. Hargreaves, B. J. Mc Loughlin and S. D. Mills, Eur. Pat. 80,296, CA, 100, 22672, (1984); N. Yoshida, K. Tanaka, Y. Iizuka, K. Wachi, T. Nishimura and H. Yasuda, (Sankyo Co., Ltd), Jpn. Kokai Tokkyo Koho JP 7,488,889, CA, 82, 57744, (1975); J. Dizon and D. H. Robinson, (Fisons PLC), Brit. UK Pat. Appl. GB 2,179,655, CA, 108, 37839, (1988); W. Thorwart, U. Gebert, R. Schleyerbach and R. Bartlett, (Hoechst A.-G.), Ger. Offen. DE. 3,702,757, CA, 110, 8223, (1988); W. Thorwart, U. Gebert, R. Schleyerbach and R. Barlett, (Hoechst A.-G.), Ger. Offen. DE. 3,702,756, CA, 109, 170466, (1988); W. D. Jones and F. P. Miller, (Richardson-Merrell Inc.), Ger. Offen. DE. 3,031,703,
44. CA, 95, 81033, (1981);
45. F. P. Miller and W. D. Jones, (Richardson-Merrell Inc.), Belgian Pat. 884,990,
46. CA, 95, 62276, (1981).