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Volumn 3, Issue 1, 1997, Pages 17-27

Peptomers: A versatile approach for the preparation of diverse combinatorial peptidomimetic bead libraries

Author keywords

Coding; Combinatorial peptidomimetic library; Dual color assay; Edman degradation; Insulin receptor ligands; Peptoid; Streptavidin ligands

Indexed keywords

DRUG DERIVATIVE; GLYCINE; INSULIN RECEPTOR; PEPTIDE; PEPTOID; PLANT RESIN; STREPTAVIDIN;

EID: 0031308991     PISSN: 13811991     EISSN: None     Source Type: Journal    
DOI: 10.1023/A:1009698507588     Document Type: Article
Times cited : (47)

References (44)
  • 1
    • 0026419328 scopus 로고
    • A new type of synthetic peptide library for identifying ligand-binding activity
    • Lam, K.S., Salmon, S.E., Hersh, E.M., Hruby, V.J., Kazmierski, W.M. and Knapp, R.J., A new type of synthetic peptide library for identifying ligand-binding activity, Nature, 354 (1991) 82-84.
    • (1991) Nature , vol.354 , pp. 82-84
    • Lam, K.S.1    Salmon, S.E.2    Hersh, E.M.3    Hruby, V.J.4    Kazmierski, W.M.5    Knapp, R.J.6
  • 2
    • 0025893762 scopus 로고
    • General method for rapid synthesis of multicomponent peptide mixtures
    • Furka, À., Sebestyén, F., Asgedom, M. and Dibó, G., General method for rapid synthesis of multicomponent peptide mixtures, Int. J. Pept. Protein Res., 37 (1991) 487-493.
    • (1991) Int. J. Pept. Protein Res. , vol.37 , pp. 487-493
    • Furka, À.1    Sebestyén, F.2    Asgedom, M.3    Dibó, G.4
  • 3
    • 0029074391 scopus 로고
    • Library of libraries: Approach to synthetic combinatorial library design and screening of 'pharmacophore' motifs
    • Sepetov, N.F., Krchňák, V., Stanková, M., Wade, S., Lam, K.S. and Lebl, M., Library of libraries: Approach to synthetic combinatorial library design and screening of 'pharmacophore' motifs, Proc. Natl. Acad. Sci. USA, 92 (1995) 5426-5430.
    • (1995) Proc. Natl. Acad. Sci. USA , vol.92 , pp. 5426-5430
    • Sepetov, N.F.1    Krchňák, V.2    Stanková, M.3    Wade, S.4    Lam, K.S.5    Lebl, M.6
  • 4
    • 0029896432 scopus 로고    scopus 로고
    • Identification of GIYWHHY as a novel peptide substrate for human p60c-src protein tyrosine kinase
    • Lou, Q., Leftwich, M.E. and Lam, K.S., Identification of GIYWHHY as a novel peptide substrate for human p60c-src protein tyrosine kinase, Bioorg. Med. Chem., 4 (1996) 677-682.
    • (1996) Bioorg. Med. Chem. , vol.4 , pp. 677-682
    • Lou, Q.1    Leftwich, M.E.2    Lam, K.S.3
  • 5
    • 0028556408 scopus 로고
    • Identifying substrate motifs of protein kinases by a random library approach
    • Wu, J., Ma, Q.N. and Lam, K.S., Identifying substrate motifs of protein kinases by a random library approach, Biochemistry, 33 (1994) 14825-14833.
    • (1994) Biochemistry , vol.33 , pp. 14825-14833
    • Wu, J.1    Ma, Q.N.2    Lam, K.S.3
  • 6
    • 0028264809 scopus 로고
    • Portion-mixing libraries of quenched fluorogenic substrates for complete subsite mapping of endoprotease specificity
    • Meldal, M., Svendsen, I., Breddam, K. and Auzanneau, F.-I., Portion-mixing libraries of quenched fluorogenic substrates for complete subsite mapping of endoprotease specificity, Proc. Natl. Acad. Sci. USA, 91 (1994) 3314-3318.
    • (1994) Proc. Natl. Acad. Sci. USA , vol.91 , pp. 3314-3318
    • Meldal, M.1    Svendsen, I.2    Breddam, K.3    Auzanneau, F.-I.4
  • 7
    • 0030252966 scopus 로고    scopus 로고
    • High-volume cellular screening for anticancer agents with combinatorial chemical libraries: A new methodology
    • Salmon, S.E., Liu-Stevens, R.H., Zhao, Y., Lebl, M., Krchňák, V., Wertman, K., Sepetov, N. and Lam, K.S., High-volume cellular screening for anticancer agents with combinatorial chemical libraries: A new methodology, Mol. Div., 2 (1996) 57-63.
    • (1996) Mol. Div. , vol.2 , pp. 57-63
    • Salmon, S.E.1    Liu-Stevens, R.H.2    Zhao, Y.3    Lebl, M.4    Krchňák, V.5    Wertman, K.6    Sepetov, N.7    Lam, K.S.8
  • 8
    • 0028318863 scopus 로고
    • Applications of combinatorial technologies to drug discovery. 2. Combinatorial organic synthesis, library screening strategies, and future directions
    • Gordon, E.M., Barrett, R.W., Dower, W.J., Fodor, S.RA. and Gallop, M.A., Applications of combinatorial technologies to drug discovery. 2. Combinatorial organic synthesis, library screening strategies, and future directions, J. Med. Chem., 37 (1994) 1385-1401.
    • (1994) J. Med. Chem. , vol.37 , pp. 1385-1401
    • Gordon, E.M.1    Barrett, R.W.2    Dower, W.J.3    Fodor, S.R.A.4    Gallop, M.A.5
  • 9
    • 0026419319 scopus 로고
    • Generation and use of synthetic peptide combinatorial libraries for basic research and drug discovery
    • Houghten, R.A., Pinilla, C., Blondelle, S.E., Appel, J.R., Dooley, C.T. and Cuervo, J.H., Generation and use of synthetic peptide combinatorial libraries for basic research and drug discovery, Nature, 354 (1991) 84-86.
    • (1991) Nature , vol.354 , pp. 84-86
    • Houghten, R.A.1    Pinilla, C.2    Blondelle, S.E.3    Appel, J.R.4    Dooley, C.T.5    Cuervo, J.H.6
  • 10
    • 0027052983 scopus 로고
    • Rapid identification of high affinity peptide ligands using positional scanning synthetic peptide combinatorial libraries
    • Pinilla, C., Appel, J.R., Blanc, P. and Houghten, R.A., Rapid identification of high affinity peptide ligands using positional scanning synthetic peptide combinatorial libraries, BioTechniques, 13 (1992) 901-905.
    • (1992) BioTechniques , vol.13 , pp. 901-905
    • Pinilla, C.1    Appel, J.R.2    Blanc, P.3    Houghten, R.A.4
  • 11
    • 0343986261 scopus 로고
    • A comparison of combinatorial library approaches for the study of opioid compounds
    • Dooley, C.T. and Houghten, R.A., A comparison of combinatorial library approaches for the study of opioid compounds, Perspect. Drug Discov. Design, 2 (1994) 287-304.
    • (1994) Perspect. Drug Discov. Design , vol.2 , pp. 287-304
    • Dooley, C.T.1    Houghten, R.A.2
  • 12
    • 0028173391 scopus 로고
    • 'Libraries from libraries': Chemical transformation of combinatorial libraries to extend the range and repertoire of chemical diversity
    • Ostresh, J.M., Husar, G.M., Blondelle, S.E., Dörner, B., Weber, P.A. and Houghten, R.A., 'Libraries from libraries': Chemical transformation of combinatorial libraries to extend the range and repertoire of chemical diversity, Proc. Natl. Acad. Sci. USA, 91 (1994) 11138-11142.
    • (1994) Proc. Natl. Acad. Sci. USA , vol.91 , pp. 11138-11142
    • Ostresh, J.M.1    Husar, G.M.2    Blondelle, S.E.3    Dörner, B.4    Weber, P.A.5    Houghten, R.A.6
  • 14
    • 84989568285 scopus 로고
    • Synthetic methods for the implementation of encoded combinatorial chemistry
    • Nielsen, J., Brenner, S. and Janda, K.D., Synthetic methods for the implementation of encoded combinatorial chemistry, J. Am. Chem. Soc., 115 (1993) 9812-9813.
    • (1993) J. Am. Chem. Soc. , vol.115 , pp. 9812-9813
    • Nielsen, J.1    Brenner, S.2    Janda, K.D.3
  • 16
    • 0000772738 scopus 로고
    • Encoded combinatorial peptide libraries containing non-natural amino acids
    • Kerr, J.M., Banville, S.C. and Zuckermann, R.N., Encoded combinatorial peptide libraries containing non-natural amino acids, J. Am. Chem. Soc., 115 (1993) 2529-2531.
    • (1993) J. Am. Chem. Soc. , vol.115 , pp. 2529-2531
    • Kerr, J.M.1    Banville, S.C.2    Zuckermann, R.N.3
  • 17
    • 0030072692 scopus 로고
    • A new combination of protecting groups and links for encoded synthetic libraries suited for consecutive tests on solid phase and in solution
    • Felder, E.R., Heizmann, G., Matthews, I.T., Rink, H. and Spieser, E., A new combination of protecting groups and links for encoded synthetic libraries suited for consecutive tests on solid phase and in solution, Mol. Div., 1 (1995) 109-112.
    • (1995) Mol. Div. , vol.1 , pp. 109-112
    • Felder, E.R.1    Heizmann, G.2    Matthews, I.T.3    Rink, H.4    Spieser, E.5
  • 18
    • 0029328482 scopus 로고
    • Linear presentation of variable side-chain spacing in a highly diverse combinatorial library
    • Krchňák, V., Weichsel, A.S., Cabel, D. and Lebl, M., Linear presentation of variable side-chain spacing in a highly diverse combinatorial library, Pept. Res., 8 (1995) 198-205.
    • (1995) Pept. Res. , vol.8 , pp. 198-205
    • Krchňák, V.1    Weichsel, A.S.2    Cabel, D.3    Lebl, M.4
  • 19
    • 0027597947 scopus 로고
    • Peptide-encoding for structure determination of nonsequenceable polymers within libraries synthesized and tested on solid-phase supports
    • Nikolaiev, V., Stierandová, A., Krchňák, V., Seligmann, B., Lam, K.S., Salmon, S.E. and Lebl, M., Peptide-encoding for structure determination of nonsequenceable polymers within libraries synthesized and tested on solid-phase supports, Pept. Res., 6 (1993) 161-170.
    • (1993) Pept. Res. , vol.6 , pp. 161-170
    • Nikolaiev, V.1    Stierandová, A.2    Krchňák, V.3    Seligmann, B.4    Lam, K.S.5    Salmon, S.E.6    Lebl, M.7
  • 20
    • 0028327679 scopus 로고
    • Synthetic receptor binding elucidated with an encoded combinatorial library
    • Borchardt, A. and Still, W.C., Synthetic receptor binding elucidated with an encoded combinatorial library, J. Am. Chem. Soc., 116 (1994) 373-374.
    • (1994) J. Am. Chem. Soc. , vol.116 , pp. 373-374
    • Borchardt, A.1    Still, W.C.2
  • 22
  • 23
    • 0028815228 scopus 로고
    • Radio frequency tag encoded combinatorial library method for the discovery of tripeptide-substituted cinnamic acid inhibitors of the protein tyrosine phosphatase PTP1B
    • Moran, E.J., Sarshar, S., Cargill, J.F., Shabbaz, M.M., Lio, A., Mjalli, A.M.M. and Armstrong, R.W., Radio frequency tag encoded combinatorial library method for the discovery of tripeptide-substituted cinnamic acid inhibitors of the protein tyrosine phosphatase PTP1B, J. Am. Chem. Soc., 117 (1995) 10787-10788.
    • (1995) J. Am. Chem. Soc. , vol.117 , pp. 10787-10788
    • Moran, E.J.1    Sarshar, S.2    Cargill, J.F.3    Shabbaz, M.M.4    Lio, A.5    Mjalli, A.M.M.6    Armstrong, R.W.7
  • 25
    • 0028153337 scopus 로고
    • Application of one-bead one structure approach to identification of nonpeptidic ligands
    • Stanková, M., Issakova, O., Sepetov, N.F., Krchňák, V., Lam, K.S. and Lebl, M., Application of one-bead one structure approach to identification of nonpeptidic ligands, Drug Dev. Res., 33 (1994) 146-156.
    • (1994) Drug Dev. Res. , vol.33 , pp. 146-156
    • Stanková, M.1    Issakova, O.2    Sepetov, N.F.3    Krchňák, V.4    Lam, K.S.5    Lebl, M.6
  • 26
    • 0028229329 scopus 로고
    • Microchemical structural determination of a peptoid bound to a polymeric bead by matrix-assisted laser desorption ionization time-of-flight spectrometry
    • Zambias, R.A., Boulton, D.A. and Griffin, P.R., Microchemical structural determination of a peptoid bound to a polymeric bead by matrix-assisted laser desorption ionization time-of-flight spectrometry, Tetrahedron Lett., 35 (1994) 4283-4286.
    • (1994) Tetrahedron Lett. , vol.35 , pp. 4283-4286
    • Zambias, R.A.1    Boulton, D.A.2    Griffin, P.R.3
  • 27
    • 23444457432 scopus 로고
    • A mass spectrometric solution to the address problem of combinatorial libraries
    • Brummel, C.L., Lee, I.N.W., Zhou, Y., Benkovic, S.J. and Winograd, N., A mass spectrometric solution to the address problem of combinatorial libraries, Science, 264 (1994) 399-402.
    • (1994) Science , vol.264 , pp. 399-402
    • Brummel, C.L.1    Lee, I.N.W.2    Zhou, Y.3    Benkovic, S.J.4    Winograd, N.5
  • 28
    • 0027972778 scopus 로고
    • Matrix-assisted laser desorption ionization for rapid determination of the sequences of biologically active peptides isolated from support-bound combinatorial peptide libraries
    • Youngquist, R.S., Fuentes, G.R., Lacey, M.P. and Keough, T., Matrix-assisted laser desorption ionization for rapid determination of the sequences of biologically active peptides isolated from support-bound combinatorial peptide libraries, Rapid Commun. Mass Spectrom., 8 (1994) 77-81.
    • (1994) Rapid Commun. Mass Spectrom. , vol.8 , pp. 77-81
    • Youngquist, R.S.1    Fuentes, G.R.2    Lacey, M.P.3    Keough, T.4
  • 30
    • 0025449880 scopus 로고
    • Color-monitored solid-phase multiple peptide synthesis under low-pressure continuous flow conditions
    • Krchňák, V. and Vagner, J., Color-monitored solid-phase multiple peptide synthesis under low-pressure continuous flow conditions, Pept. Res., 3 (1990) 182-193.
    • (1990) Pept. Res. , vol.3 , pp. 182-193
    • Krchňák, V.1    Vagner, J.2
  • 32
    • 0000908874 scopus 로고
    • Efficient method for the preparation of peptoids [oligo(N-substituted glycines)] by submonomer solid-phase synthesis
    • Zuckermann, R.N., Kerr, J.M., Kent, S.B.H. and Moos, W.H., Efficient method for the preparation of peptoids [oligo(N-substituted glycines)] by submonomer solid-phase synthesis, J. Am. Chem. Soc., 114 (1992) 10646-10647.
    • (1992) J. Am. Chem. Soc. , vol.114 , pp. 10646-10647
    • Zuckermann, R.N.1    Kerr, J.M.2    Kent, S.B.H.3    Moos, W.H.4
  • 33
    • 12044258245 scopus 로고
    • 1-Hydroxy-7-azabenzotriazole. An efficient peptide coupling additive
    • Carpino, L.A., 1-Hydroxy-7-azabenzotriazole. An efficient peptide coupling additive, J. Am. Chem. Soc., 115 (1993) 4397-4398.
    • (1993) J. Am. Chem. Soc. , vol.115 , pp. 4397-4398
    • Carpino, L.A.1
  • 34
    • 0031088571 scopus 로고    scopus 로고
    • Synthesis and screening of an indexed motif-library containing nonproteinogenic amino acids
    • Østergaard, S. and Holm, A., Synthesis and screening of an indexed motif-library containing nonproteinogenic amino acids, J. Pept. Sci., 3 (1997) 123-132.
    • (1997) J. Pept. Sci. , vol.3 , pp. 123-132
    • Østergaard, S.1    Holm, A.2
  • 35
    • 0025004285 scopus 로고
    • Random peptide libraries: A source of specific protein binding molecules
    • Devlin, J.J., Panganiban, L.C. and Devlin, P.E., Random peptide libraries: A source of specific protein binding molecules, Science, 249 (1990) 404-406.
    • (1990) Science , vol.249 , pp. 404-406
    • Devlin, J.J.1    Panganiban, L.C.2    Devlin, P.E.3
  • 36
    • 0026807019 scopus 로고
    • Crystal structure and ligand-binding studies of a screened peptide completed with streptavidin
    • Weber, P.C., Pantoliano, M.W. and Thompson, L.D., Crystal structure and ligand-binding studies of a screened peptide completed with streptavidin, Biochemistry, 31 (1992) 9350-9354.
    • (1992) Biochemistry , vol.31 , pp. 9350-9354
    • Weber, P.C.1    Pantoliano, M.W.2    Thompson, L.D.3
  • 37
    • 0028914195 scopus 로고
    • Application of a dual color detection scheme in the screening of a random combinatorial peptide library
    • Lam, K.S., Wade, S., Abdul-Latif, F. and Lebl, M., Application of a dual color detection scheme in the screening of a random combinatorial peptide library, J. Immunol. Methods, 180 (1994) 219-223.
    • (1994) J. Immunol. Methods , vol.180 , pp. 219-223
    • Lam, K.S.1    Wade, S.2    Abdul-Latif, F.3    Lebl, M.4
  • 40
    • 0343010435 scopus 로고    scopus 로고
    • The synthesis of peptidomimetic combinatorial libraries through successive amide alkylations
    • Dörner, B., Husar, G.M., Ostresh, J.M. and Houghten, R.A., The synthesis of peptidomimetic combinatorial libraries through successive amide alkylations, Bioorg. Med. Chem., 4 (1996) 709-715.
    • (1996) Bioorg. Med. Chem. , vol.4 , pp. 709-715
    • Dörner, B.1    Husar, G.M.2    Ostresh, J.M.3    Houghten, R.A.4
  • 41
    • 2342514048 scopus 로고    scopus 로고
    • The use of soluble polyamine combinatorial libraries for the identification of potent opioid receptor active compounds
    • Kaumaya, P.T.P. and Hodges, R.S. (Eds.) Mayflower Scientific, Kingswinford
    • Houghten, R.A., Dooley, C.T. and Ostresh, J.M., The use of soluble polyamine combinatorial libraries for the identification of potent opioid receptor active compounds, In Kaumaya, P.T.P. and Hodges, R.S. (Eds.) Peptides: Chemistry, Structure and Biology, Mayflower Scientific, Kingswinford, 1996, pp. 278-280.
    • (1996) Peptides: Chemistry, Structure and Biology , pp. 278-280
    • Houghten, R.A.1    Dooley, C.T.2    Ostresh, J.M.3
  • 42
    • 0029988589 scopus 로고    scopus 로고
    • Azatides: Solution and liquid phase synthesis of a new peptidomimetic
    • Han, H. and Janda, K.D., Azatides: Solution and liquid phase synthesis of a new peptidomimetic, J. Am. Chem. Soc., 118 (1996) 2539-2544.
    • (1996) J. Am. Chem. Soc. , vol.118 , pp. 2539-2544
    • Han, H.1    Janda, K.D.2
  • 44
    • 0028833961 scopus 로고
    • Reductive alkylation on a solid-phase: Synthesis of a piperazinedione combinatorial library
    • Gordon, D.W. and Steele, J., Reductive alkylation on a solid-phase: Synthesis of a piperazinedione combinatorial library, Bioorg. Med. Chem. Lett., 5 (1995) 47-50.
    • (1995) Bioorg. Med. Chem. Lett. , vol.5 , pp. 47-50
    • Gordon, D.W.1    Steele, J.2


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