Acyl amino acid derivatives as novel inhibitors of influenza neuraminidase

Bioscience, Biotechnology and Biochemistry

Volumn 61, Issue 5, 1997, Pages 870-874

  Kondoh, Mitsuyo ^a   Furutani, Toshiyuki ^a,b   Azuma, Masayuki ^a   Ooshima, Hiroshi ^a   Kato, Jyoji ^a  

^a Osaka Prefecture University   (Japan)

^b MITSUBISHI TANABE PHARMA CORPORATION   (Japan)

Author keywords

Acyl amino acid derivatives; Influenza neuraminidase; Noncompetitive inhibitor

Indexed keywords

AMINO ACID; ENZYME INHIBITOR; N ACETYLNEURAMINIC ACID; SIALIDASE;

ACYLATION; ANIMAL; ARTICLE; DRUG ANTAGONISM; ENZYMOLOGY; HUMAN; KINETICS; ORTHOMYXOVIRUS; RAT; WISTAR RAT;

ACYLATION; AMINO ACIDS; ANIMALS; ENZYME INHIBITORS; HUMANS; KINETICS; N-ACETYLNEURAMINIC ACID; NEURAMINIDASE; ORTHOMYXOVIRIDAE; RATS; RATS, WISTAR;

ANIMALIA; ORTHOMYXOVIRIDAE;

EID: 0031148043     PISSN: 09168451     EISSN: 13476947     Source Type: Journal    
DOI: 10.1271/bbb.61.870     Document Type: Article

References (19)

1. P. M. Colman, Protein Sei., 3, 1687-1696 (1994).
2. C. Liu, M. C. Eichelberger, R. W. Compans, and G. M. Air, J. ViroL, 69, 1099-1106 (1995).
3. A. Puri, S. Grimaldi, and R. Blumenthal, Biochemistry, 31, 10108-10113 (1992).
4. P. Palese and R. W. Compans, J. Gen. Virol., 33, 159-163 (1976).
5. I. A. Griffin, S. Basak, and R. W. Compans, Virology, 125, 324-334 (1983).
6. S. Shibata, F. Y. Goshima, K. Maeo, T. Hanaichi, Y. Fujita, K. Nakajima, M. Imai, T. Komatsu, and S. Sugiura, J. Virol., 67, 3264-3273 (1993).
7. M. J. Bamford, J. Enzyme Inhibition, 10, 1-16 (1995).
8. T. Furutani, M. Furui, H. Ooshima, and J. Kato, Enzyme Microb. Technol, 19, 578-584 (1996).
9. T. Miyagi, J. Sagawa, K. Konno, and S. Tsuiki, J. Biochem., 107, 794-798 (1990).
10. T. Nagai, Y. Miyaichi, T. Tomimori, Y. Suzuki, and H. Yamada, Antiviral Res., 19, 207-217 (1992).
11. T. Nagai and H. Yamada, Chem. Pharm. Bull., 36, 4008-4018 (1988).
12. O. H. Lowry, N. J. Rosebrough, A. L. Farr, and R. J. Randall, J. Biol. Chem., 193, 265-275 (1951).
13. C. T. Holzer, M. Itzstein, B. Jin, M. S. Pegg, W. P. Stewart, and W. Y. Wu, GlycoconjugateJ., 10, 40-44 (1993).
14. M. Itzstein, W. Y. Wu, G. B. Kok, M. S. Pegg, J. C. Dyason, B. Jin, T. V. Phan, M. L. Smythe, H. F. White, S. W. Oliver, P. M. Colman, J. N. Varghese, D. M. Ryan, J. M. Woods, R. C. Bethell, V. J. Hotham, J. M. Cameron, and C. R. Penn, Nature, 363, 418-423 (1993).
15. S. Singh, M. J. Jedrzejas, G. M. Air, M. Luo, W. G. Laver, and W. J. Brouillette, J. Med. Chem., 38, 3217-3225 (1995).
16. F. G. Hayden, J. J. Treanor, R. F. Betts, M. Lobo, J. D. Esinhart, and E. K. Hussey, JAMA, 275, 295-299 (1996).
17. J. C. Wu, G. W. Peet, S. J. Coutts, R. J. Eckner, J. A. Griffin, and P. R. Farina, Biochemistry, 34, 7154-7160 (1995).
18. A. Gottschalk, Adv. Enzymol, 20, 135-145 (1958).
19. L. V. Gubareva, R. Bethell, G. J. Hart, K. G. Murti, C. R. Penn, and R. G. Webster, J. Virol., 70, 1818-1827 (1996).