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Volumn 38, Issue 2, 1997, Pages 169-174

Characterization of pulmonary and myocardial beta-adrenoceptors with S- 1'-[fluorine-18]fluorocarazolol

Author keywords

beta adrenoceptor density; fluorine 18 fluorocarazolol; PET

Indexed keywords

BETA ADRENERGIC RECEPTOR; PINDOLOL; SALBUTAMOL;

EID: 0031053257     PISSN: 01615505     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article
Times cited : (23)

References (32)
  • 3
    • 0028150716 scopus 로고
    • 18F labeling of fluorocarazolol, a high-affinity beta-adrenergic receptor antagonist
    • 18F labeling of fluorocarazolol, a high-affinity beta-adrenergic receptor antagonist. J Med Chem 1994;37:3219-3230.
    • (1994) J Med Chem , vol.37 , pp. 3219-3230
    • Zheng, L.1    Berridge, M.S.2    Ernsberger, P.3
  • 4
    • 0019976620 scopus 로고
    • The use of tritium-labeled compounds to develop gamma-emitting receptor-binding radiotracers
    • Francis BE, Eckelman WC, Grissom MP, Gibson RE, Reba RC. The use of tritium-labeled compounds to develop gamma-emitting receptor-binding radiotracers. Nucl Med Biol 1982;9:173-179.
    • (1982) Nucl Med Biol , vol.9 , pp. 173-179
    • Francis, B.E.1    Eckelman, W.C.2    Grissom, M.P.3    Gibson, R.E.4    Reba, R.C.5
  • 6
    • 0029670104 scopus 로고    scopus 로고
    • 18F]fluorocarazolol, ligands for the visualization of pulmonary β-adrenergic receptors with PET
    • 18F]fluorocarazolol, ligands for the visualization of pulmonary β-adrenergic receptors with PET. Nucl Med Biol 1996;23:159-167.
    • (1996) Nucl Med Biol , vol.23 , pp. 159-167
    • Elsinga, P.H.1    Vos, M.G.2    Van Waarde, A.3
  • 8
    • 0026874022 scopus 로고
    • A comparison of beta-adrenergic receptors and in vitro relaxant responses to isoproterenol in asthmatic airway smooth muscle
    • Bai TR, Mak JC, Barnes PJ. A comparison of beta-adrenergic receptors and in vitro relaxant responses to isoproterenol in asthmatic airway smooth muscle. Am J Respir Cell Mol Biol 1992;6:647-651.
    • (1992) Am J Respir Cell Mol Biol , vol.6 , pp. 647-651
    • Bai, T.R.1    Mak, J.C.2    Barnes, P.J.3
  • 9
    • 0025212607 scopus 로고
    • Airway beta-adrenoceptor number in cystic fibrosis and asthma
    • Sharma RK, Jeffery PK. Airway beta-adrenoceptor number in cystic fibrosis and asthma. Clin Sci 1990;78:409-417.
    • (1990) Clin Sci , vol.78 , pp. 409-417
    • Sharma, R.K.1    Jeffery, P.K.2
  • 10
    • 0023228682 scopus 로고
    • Decreased bronchiolar epithelial beta-adrenoceptor densities in patients with chronic obstructive lung disease
    • Raaijmakers JA, Beneker C, Dol R, de Ruiter Bootsma AL. Decreased bronchiolar epithelial beta-adrenoceptor densities in patients with chronic obstructive lung disease. Cell Mol Biol 1987;33:515-518.
    • (1987) Cell Mol Biol , vol.33 , pp. 515-518
    • Raaijmakers, J.A.1    Beneker, C.2    Dol, R.3    De Ruiter Bootsma, A.L.4
  • 11
    • 0022980843 scopus 로고
    • Beta-1- and beta-2-adrenergic-receptor subpopulations in nonfailing and failing human ventricular myocardium: Coupling of both receptor subtypes to muscle contraction and selective beta-1-receptor down-regulation in heart failure
    • Bristow MR, Ginsburg R, Umans V, et al. Beta-1- and beta-2-adrenergic-receptor subpopulations in nonfailing and failing human ventricular myocardium: coupling of both receptor subtypes to muscle contraction and selective beta-1-receptor down-regulation in heart failure. Circ Res 1986;59:297-309.
    • (1986) Circ Res , vol.59 , pp. 297-309
    • Bristow, M.R.1    Ginsburg, R.2    Umans, V.3
  • 12
    • 0025851462 scopus 로고
    • Beta1- and beta2-adrenoceptors in the human heart: Properties, function and alterations in chronic heart failure
    • Brodde OE. Beta1- and beta2-adrenoceptors in the human heart: properties, function and alterations in chronic heart failure. Pharmacol Rev 1991;43:203-242.
    • (1991) Pharmacol Rev , vol.43 , pp. 203-242
    • Brodde, O.E.1
  • 13
    • 0026090589 scopus 로고
    • Lung beta-adrenoceptors in pulmonary hypertension. a study of biopsy specimens in children with congenital heart disease
    • Lopes AA, Liberato MH, Brentani MM, Aiello VD, Riso AA, Ebaid M. Lung beta-adrenoceptors in pulmonary hypertension. A study of biopsy specimens in children with congenital heart disease. Chest 1991;99:637-641.
    • (1991) Chest , vol.99 , pp. 637-641
    • Lopes, A.A.1    Liberato, M.H.2    Brentani, M.M.3    Aiello, V.D.4    Riso, A.A.5    Ebaid, M.6
  • 14
    • 33544473721 scopus 로고
    • Suitability of CGP12177 and CGP26505 for quantitative imaging of beta-adrenoceptors
    • Van Waarde A, Meeder JG, Blanksma PK, et al. Suitability of CGP12177 and CGP26505 for quantitative imaging of beta-adrenoceptors. Nucl Med Biol 1992;19: 711-718.
    • (1992) Nucl Med Biol , vol.19 , pp. 711-718
    • Van Waarde, A.1    Meeder, J.G.2    Blanksma, P.K.3
  • 15
    • 0026447602 scopus 로고
    • Uptake of radioligands by rat heart and lung in vivo: CGP12177 does and CGP26505 does not reflect binding to β-adrenoceptors
    • Van Waarde A, Meeder JG, Blanksma PK, et al. Uptake of radioligands by rat heart and lung in vivo: CGP12177 does and CGP26505 does not reflect binding to β-adrenoceptors. Eur J Pharmacol 1992;222:107-112.
    • (1992) Eur J Pharmacol , vol.222 , pp. 107-112
    • Van Waarde, A.1    Meeder, J.G.2    Blanksma, P.K.3
  • 16
    • 0027320592 scopus 로고
    • Demonstration of the suitability of CGP 12177 for in vivo studies of β-adrenoceptors
    • Law MP. Demonstration of the suitability of CGP 12177 for in vivo studies of β-adrenoceptors. Br J Pharmacol 1993;109:1101-1109.
    • (1993) Br J Pharmacol , vol.109 , pp. 1101-1109
    • Law, M.P.1
  • 17
    • 0027401947 scopus 로고
    • 11C CGP-12177 to assess beta-adrenergic receptor concentration in idiopathic dilated cardiomyopathy
    • 11C CGP-12177 to assess beta-adrenergic receptor concentration in idiopathic dilated cardiomyopathy. Circulation 1993;87:1169-1178.
    • (1993) Circulation , vol.87 , pp. 1169-1178
    • Merlet, P.1    Delforge, J.2    Syrota, A.3
  • 19
    • 0025762367 scopus 로고
    • Cardiac beta-adrenergic receptor density measured in vivo using PET, CGP 12177 and a new graphical method
    • Delforge J, Syrota A, Lançon JP, et al. Cardiac beta-adrenergic receptor density measured in vivo using PET, CGP 12177 and a new graphical method. J Nucl Med 1991;32:739-748.
    • (1991) J Nucl Med , vol.32 , pp. 739-748
    • Delforge, J.1    Syrota, A.2    Lançon, J.P.3
  • 20
  • 22
    • 0027462811 scopus 로고
    • Airway responsiveness: Standardized challenge testing with pharmacological, physical and sensitizing stimuli in adults
    • Sterk PJ, Fabbri LM, Quanjer PH, et al. Airway responsiveness: Standardized challenge testing with pharmacological, physical and sensitizing stimuli in adults. Eur Respir J 1993;6(suppl. 16):53-83.
    • (1993) Eur Respir J , vol.6 , Issue.16 SUPPL. , pp. 53-83
    • Sterk, P.J.1    Fabbri, L.M.2    Quanjer, P.H.3
  • 24
    • 1842400095 scopus 로고
    • Quantification of beta-adrenergic receptor concentration in human with positron emission tomography
    • Merlet P, Delforge J, Syrota A, et al. Quantification of beta-adrenergic receptor concentration in human with positron emission tomography [Abstract]. J Nucl Med 1991;32:989.
    • (1991) J Nucl Med , vol.32 , pp. 989
    • Merlet, P.1    Delforge, J.2    Syrota, A.3
  • 25
    • 23544436817 scopus 로고
    • Myocardial beta-adrenoceptor density is reduced in hypertrophic cardiomyopathy
    • Lefroy DC, De Silva R, Choudhury L, et al. Myocardial beta-adrenoceptor density is reduced in hypertrophic cardiomyopathy [Abstract]. Circulation 1992;86:I-246.
    • (1992) Circulation , vol.86
    • Lefroy, D.C.1    De Silva, R.2    Choudhury, L.3
  • 26
    • 0023195974 scopus 로고
    • Beta-adrenoceptors in human tracheal smooth muscle: Characteristics of binding and relaxation
    • van Koppen CJ, Hermanussen MW, Verrijp KN, et al. Beta-adrenoceptors in human tracheal smooth muscle: characteristics of binding and relaxation. Life Sci 1987;40: 2561-2570.
    • (1987) Life Sci , vol.40 , pp. 2561-2570
    • Van Koppen, C.J.1    Hermanussen, M.W.2    Verrijp, K.N.3
  • 27
    • 0021784714 scopus 로고
    • Autoradiographic visualization of beta-adrenoceptor subtypes in human lung
    • Carstairs JR, Nimmo AJ, Barnes PJ. Autoradiographic visualization of beta-adrenoceptor subtypes in human lung. Am Rev Respir Dis 1985;132:541-547.
    • (1985) Am Rev Respir Dis , vol.132 , pp. 541-547
    • Carstairs, J.R.1    Nimmo, A.J.2    Barnes, P.J.3
  • 28
    • 0030081109 scopus 로고    scopus 로고
    • Optimal experiment design for PET quantification of receptor concentration
    • Muzic RF, Nelson AD, Saidel GM, Miraldi F. Optimal experiment design for PET quantification of receptor concentration. IEEE Trans Med Imag 1996;15:2-12.
    • (1996) IEEE Trans Med Imag , vol.15 , pp. 2-12
    • Muzic, R.F.1    Nelson, A.D.2    Saidel, G.M.3    Miraldi, F.4
  • 29
    • 0020523811 scopus 로고
    • CGP-12177. a hydrophilic beta-adrenergic receptor radioligand reveals high affinity binding of agonists to intact cells
    • Staehelin M, Simons P, Jaeggi K, Wigger N. CGP-12177. A hydrophilic beta-adrenergic receptor radioligand reveals high affinity binding of agonists to intact cells. J Biol Chem 1983;258:3496-3502.
    • (1983) J Biol Chem , vol.258 , pp. 3496-3502
    • Staehelin, M.1    Simons, P.2    Jaeggi, K.3    Wigger, N.4
  • 31
    • 0028985330 scopus 로고
    • Quantification of a carbon-11-labeled β-adrenoceptor ligand, S-(-)-CGP 12177, in plasma of humans and rats
    • Van Waarde A, Anthonio RL, Visser TJ, et al. Quantification of a carbon-11-labeled β-adrenoceptor ligand, S-(-)-CGP 12177, in plasma of humans and rats. J Chromatogr 1995;B 663:361-369.
    • (1995) J Chromatogr , vol.663 B , pp. 361-369
    • Van Waarde, A.1    Anthonio, R.L.2    Visser, T.J.3
  • 32
    • 0000102055 scopus 로고
    • 11C]-CGP12177 metabolism in rat, dog and man using solid phase extraction and HPLC
    • 11C]-CGP12177 metabolism in rat, dog and man using solid phase extraction and HPLC. J Lab Compd Radiopharm 1992;31:518-520.
    • (1992) J Lab Compd Radiopharm , vol.31 , pp. 518-520
    • Luthra, S.K.1    Osman, S.2    Steel, C.J.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.