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Volumn 14, Issue 2, 1997, Pages 243-255

In vitro controlled release kinetics of local anaesthetics from poly(D,L-lactide) and poly(lactide-co-glycolide) microspheres

Author keywords

Controlled release; Local anaesthetic; Microsphere; Poly(D,L lactide); Poly(lactide co glycolide)

Indexed keywords

BUPIVACAINE; ETIDOCAINE; LIDOCAINE; LOCAL ANESTHETIC AGENT; MEPIVACAINE; MICROSPHERE; POLYGLACTIN; POLYLACTIDE;

EID: 0031045570     PISSN: 02652048     EISSN: None     Source Type: Journal    
DOI: 10.3109/02652049709015336     Document Type: Article
Times cited : (60)

References (32)
  • 2
    • 0024553973 scopus 로고
    • The effect of the addition of low molecular weight poly(D,L-lactide) on drug release from biodegradable poly(D,L-lactide) drug delivery systems
    • BODMEIER, R., OH, K. H., and CHEN, H., 1989, The effect of the addition of low molecular weight poly(D,L-lactide) on drug release from biodegradable poly(D,L-lactide) drug delivery systems. International Journal of Pharmaceutics, 51, 1-8.
    • (1989) International Journal of Pharmaceutics , vol.51 , pp. 1-8
    • Bodmeier, R.1    Oh, K.H.2    Chen, H.3
  • 4
    • 0024336994 scopus 로고
    • Clinical pharmacokinetics of epidural and spinal anaesthesia
    • BURM, A. G. L., 1989, Clinical pharmacokinetics of epidural and spinal anaesthesia. Clinical Pharmacokinetics, 16, 283-311.
    • (1989) Clinical Pharmacokinetics , vol.16 , pp. 283-311
    • Burm, A.G.L.1
  • 5
    • 0024566293 scopus 로고
    • The influence of pH-adjusted 2-chloroprocaine on the quality and duration of subsequent epidural bupivacaine analgesia during labor: A randomized, double blind study
    • CHESTNUT, D. H., GEIGER, M., BATES, J. N., and CHOI, W. W., 1989, The influence of pH-adjusted 2-chloroprocaine on the quality and duration of subsequent epidural bupivacaine analgesia during labor: a randomized, double blind study. Anesthesiology, 70, 437-441.
    • (1989) Anesthesiology , vol.70 , pp. 437-441
    • Chestnut, D.H.1    Geiger, M.2    Bates, J.N.3    Choi, W.W.4
  • 9
    • 0023797362 scopus 로고
    • Topical anesthesia of the skin by liposome-encapsulated tetracaine
    • GESZTES, A., and MEZEI, M., 1988, Topical anesthesia of the skin by liposome-encapsulated tetracaine. Anesthesia Analgesia, 67, 1079-1081.
    • (1988) Anesthesia Analgesia , vol.67 , pp. 1079-1081
    • Gesztes, A.1    Mezei, M.2
  • 10
    • 0025731467 scopus 로고
    • Factors influencing the profiles of TRH release from copoly(d,1-lactide/glycolic acid) microspheres
    • HEYA, T., OKADA, H., OGAWA, Y., and TOGUCHI, H., 1991, Factors influencing the profiles of TRH release from copoly(d,1-lactide/glycolic acid) microspheres. International Journal of Pharmaceutics, 72, 199-205.
    • (1991) International Journal of Pharmaceutics , vol.72 , pp. 199-205
    • Heya, T.1    Okada, H.2    Ogawa, Y.3    Toguchi, H.4
  • 11
    • 0344893332 scopus 로고
    • Mechanism of sustained release medication
    • HIGUCHI, T., 1963, Mechanism of sustained release medication. Journal of Pharmaceutical Sciences, 52, 1145-1147.
    • (1963) Journal of Pharmaceutical Sciences , vol.52 , pp. 1145-1147
    • Higuchi, T.1
  • 12
    • 0026587501 scopus 로고
    • Release of benzocaine, procaine, 2-aminothiazole and 4-amino-4H-1,2,4-triazole from polymer carriers
    • KOLLI, M., MONTHEARD, J. P., and VERGNAUD, J. M., 1992, Release of benzocaine, procaine, 2-aminothiazole and 4-amino-4H-1,2,4-triazole from polymer carriers. International Journal of Pharmaceutics, 81, 103-110.
    • (1992) International Journal of Pharmaceutics , vol.81 , pp. 103-110
    • Kolli, M.1    Montheard, J.P.2    Vergnaud, J.M.3
  • 14
    • 84950232819 scopus 로고
    • Polymeric delivery systems for controlled drug release
    • LANGER, R., 1980, Polymeric delivery systems for controlled drug release. Chemical Engineering Communications, 6, 1-48.
    • (1980) Chemical Engineering Communications , vol.6 , pp. 1-48
    • Langer, R.1
  • 15
    • 0025906215 scopus 로고
    • Spinal anesthesia: Significant prolongation of the pharmacologic effect of tetracaine with lipid solution of the agent
    • LANGERMAN, L., GOLOMB, E., and BENITA, S., 1991, Spinal anesthesia: significant prolongation of the pharmacologic effect of tetracaine with lipid solution of the agent. Anesthesiology, 74, 105-107.
    • (1991) Anesthesiology , vol.74 , pp. 105-107
    • Langerman, L.1    Golomb, E.2    Benita, S.3
  • 16
    • 0026795752 scopus 로고
    • Prolongation of spinal anesthesia: Differential action of a lipid drug carrier on tetracaine, lidocaine and procaine
    • LANGERMAN, L., GRANT, G. J., ZAKOWSKI, M., RAMANATHAN, S., and TURNDORF, H., 1992, Prolongation of spinal anesthesia: differential action of a lipid drug carrier on tetracaine, lidocaine and procaine. Anesthesiology, 77, 475-481.
    • (1992) Anesthesiology , vol.77 , pp. 475-481
    • Langerman, L.1    Grant, G.J.2    Zakowski, M.3    Ramanathan, S.4    Turndorf, H.5
  • 17
    • 0028285190 scopus 로고
    • Preparation and characterization of bupivacaine-loaded polylactide and polylactide-co-glycolide microspheres
    • LE CORRE, P., LE GUEVELLO, P., GAJAN, V., CHEVANNE, F., and LE VERGE, R., 1994, Preparation and characterization of bupivacaine-loaded polylactide and polylactide-co-glycolide microspheres. International Journal of Pharmaceutics, 107, 41-49.
    • (1994) International Journal of Pharmaceutics , vol.107 , pp. 41-49
    • Le Corre, P.1    Le Guevello, P.2    Gajan, V.3    Chevanne, F.4    Le Verge, R.5
  • 19
    • 0029163511 scopus 로고
    • Motor and blood pressure effects of epidural sustained release bupivacaine from polymer microspheres: A dose-response study in rabbits
    • MALINOWSKI, J. M., BERNARD, J. M., LE CORRE, P., DUMAND, J. B., LEPAGE, J. Y., LE VERGE, R., and SOURON, R., 1995, Motor and blood pressure effects of epidural sustained release bupivacaine from polymer microspheres: a dose-response study in rabbits. Anesthesia Analgesia, 81, 519-524.
    • (1995) Anesthesia Analgesia , vol.81 , pp. 519-524
    • Malinowski, J.M.1    Bernard, J.M.2    Le Corre, P.3    Dumand, J.B.4    Lepage, J.Y.5    Le Verge, R.6    Souron, R.7
  • 20
    • 0011831666 scopus 로고
    • Influence of different liposomal formulations on pharmacokinetics of encapsulated bupivacaine
    • LEGROS, F., LUO, H., BOURGEOIS, P., LAFANT, N., and BOOGAERTS, J., 1990, Influence of different liposomal formulations on pharmacokinetics of encapsulated bupivacaine. Anesthesiology, 73, A849.
    • (1990) Anesthesiology , vol.73
    • Legros, F.1    Luo, H.2    Bourgeois, P.3    Lafant, N.4    Boogaerts, J.5
  • 23
    • 0027496079 scopus 로고
    • Sustained local anesthetic release from bioerodible polymer matrices: A potential method for prolonged regional anesthesia
    • MASTERS, D. B., BERDE, C. B., DUTTA, S., TUREK, T., and LANGER, R., 1993, Sustained local anesthetic release from bioerodible polymer matrices: a potential method for prolonged regional anesthesia. Pharmaceutical Research, 10, 1527-1532.
    • (1993) Pharmaceutical Research , vol.10 , pp. 1527-1532
    • Masters, D.B.1    Berde, C.B.2    Dutta, S.3    Turek, T.4    Langer, R.5
  • 24
    • 0025079173 scopus 로고
    • Controlled release of local anesthetic agents from liquid-solid emulsion gels
    • MHANDO, J. R., and LI WAN PO, A., 1990, Controlled release of local anesthetic agents from liquid-solid emulsion gels. International Journal of Pharmaceutics, 62, 249-258.
    • (1990) International Journal of Pharmaceutics , vol.62 , pp. 249-258
    • Mhando, J.R.1    Li Wan Po, A.2
  • 26
    • 0026571139 scopus 로고
    • The influence of polymer glass transition temperature and molecular weight on drug release from tablets containing poly(D,L-lactic acid)
    • OMELCZUK, M. O., and MCGINITY, J. W., 1992, The influence of polymer glass transition temperature and molecular weight on drug release from tablets containing poly(D,L-lactic acid). Pharmaceutical Research, 9, 26-32.
    • (1992) Pharmaceutical Research , vol.9 , pp. 26-32
    • Omelczuk, M.O.1    Mcginity, J.W.2
  • 27
    • 0027400066 scopus 로고
    • pH-dependent solubility and dissolution of bupivacaine and its relevance to the formulation of a controlled release system
    • SHAH, J. C., and MANIAR, M., 1993, pH-dependent solubility and dissolution of bupivacaine and its relevance to the formulation of a controlled release system. Journal of Controlled Release, 23, 261-270.
    • (1993) Journal of Controlled Release , vol.23 , pp. 261-270
    • Shah, J.C.1    Maniar, M.2
  • 28
    • 0028258955 scopus 로고
    • Topical liposome system bearing local anesthetic lignocaine: Preparation and evaluation
    • SHARMA, B. B., JAIN, S. K., and VYAS, S. P., 1994, Topical liposome system bearing local anesthetic lignocaine: preparation and evaluation. Journal of Microencapsulation, 11, 279-286.
    • (1994) Journal of Microencapsulation , vol.11 , pp. 279-286
    • Sharma, B.B.1    Jain, S.K.2    Vyas, S.P.3
  • 29
    • 0025202543 scopus 로고
    • Fundamental properties of local anesthetics. II. Measured octanol buffer partition coefficients and pKa values of clinically used drugs
    • STRICHARTZ, G. R., SANCHEZ, V., ARTHUR, R., CHAFETZ, R., and MARTIN, D., 1990, Fundamental properties of local anesthetics. II. Measured octanol buffer partition coefficients and pKa values of clinically used drugs. Anesthesia Analgesia, 71, 158-170.
    • (1990) Anesthesia Analgesia , vol.71 , pp. 158-170
    • Strichartz, G.R.1    Sanchez, V.2    Arthur, R.3    Chafetz, R.4    Martin, D.5
  • 30
    • 0015949763 scopus 로고
    • Quantitative analytical method for determination of drugs dispersed in polymers using differential scanning calorimetry
    • THEEUWES, F., HUSSAIN, A., and HIGUCHI, T., 1974, Quantitative analytical method for determination of drugs dispersed in polymers using differential scanning calorimetry. Journal of Pharmaceutical Sciences, 63, 427-429.
    • (1974) Journal of Pharmaceutical Sciences , vol.63 , pp. 427-429
    • Theeuwes, F.1    Hussain, A.2    Higuchi, T.3
  • 31
    • 0020353252 scopus 로고
    • Preparation and evaluation in vitro and in vivo of polylactic acid microspheres containing dibucaine
    • WAKIYAMA, N., JUNI, K., and NAKANO, M., 1982, Preparation and evaluation in vitro and in vivo of polylactic acid microspheres containing dibucaine. Chemical and Pharmaceutical Bulletin, 30, 3719-3727.
    • (1982) Chemical and Pharmaceutical Bulletin , vol.30 , pp. 3719-3727
    • Wakiyama, N.1    Juni, K.2    Nakano, M.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.