Synthesis and conformational analysis of peptide inhibitors of farnesyltransferase

Bioorganic and Medicinal Chemistry

Volumn 5, Issue 1, 1997, Pages 115-124

  Byk, Gerardo ^a   Lelievre, Yves ^b   Duchesne, Marc ^b   Clerc, François F ^b   Scherman, Daniel ^a   Guitton, Jean Dominique ^b  

^a SANOFI   (France)

^b Biotechnology Department   (France)

Author keywords

[No Author keywords available]

Indexed keywords

ANTINEOPLASTIC AGENT; PROTEIN FARNESYLTRANSFERASE; TRANSFERASE INHIBITOR;

CELL PROLIFERATION; CONFERENCE PAPER; ENZYME INHIBITION; MOLECULAR DYNAMICS; ONCOGENE RAS; PEPTIDE SYNTHESIS; STRUCTURE ACTIVITY RELATION;

ALKYL AND ARYL TRANSFERASES; ENZYME INHIBITORS; FARNESYLTRANSTRANSFERASE; MAGNETIC RESONANCE SPECTROSCOPY; MASS SPECTROMETRY; PEPTIDES; STRUCTURE-ACTIVITY RELATIONSHIP; TRANSFERASES;

EID: 0031031030     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0968-0896(96)00210-6     Document Type: Conference Paper

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