Synthesis and benzodiazepine receptor binding of some imidazo-, pyrimido[2,1-b]benzoxazoles and pyrimido[1,2-a]benzimidazoles

European Journal of Medicinal Chemistry

Volumn 32, Issue 1, 1997, Pages 83-89

  Trapani, G ^c   Franco, M ^c   Latrofa, A ^c   Genchi, G ^a   Iacobazzi, V ^a   Ghiani, C A ^b   Maciocco, E ^b   Liso, G ^c  

^a UNIVERSITY OF BARI   (Italy)

^b UNIVERSITY OF CAGLIARI   (Italy)

^c NONE

Author keywords

Central benzodiazepine receptor; GABA ratio; Imidazo 2,1 b benzoxazole; Peripheral benzodiazepine receptor; Pyrimido 1,2 a benzimidazole; Pyrimido 2,1 b benzoxazole; 35S TBPS binding

Indexed keywords

4 AMINOBUTYRIC ACID RECEPTOR; 4' CHLORODIAZEPAM; BENZIMIDAZOLE DERIVATIVE; BENZODIAZEPINE RECEPTOR; BENZOXAZOLE DERIVATIVE; FLUNITRAZEPAM;

ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; BRAIN CORTEX; BRAIN HOMOGENATE; DRUG RECEPTOR BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; MOUSE; NONHUMAN; RAT;

EID: 0031028211     PISSN: 02235234     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0223-5234(97)84364-4     Document Type: Article

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