Inhibition of dipeptidyl peptidase IV (CD26) by peptide boronic acid dipeptides

Journal of Enzyme Inhibition

Volumn 11, Issue 3, 1997, Pages 151-169

  Pargellis, Christopher A ^a   Campbell, Scot J ^a   Pav, Susan ^a   Graham, Edward T ^a   Pitner, T Phil ^a  

^a BOEHRINGER INGELHEIM PHARMACEUTICALS INC   (United States)

Author keywords

CD26; Dipeptidyl peptidase IV; DPPIV; Peptide boronates; Val boroPro

Indexed keywords

BORONIC ACID DERIVATIVE; DIPEPTIDE; DIPEPTIDYL PEPTIDASE IV; RECOMBINANT ENZYME;

ANIMAL CELL; ARTICLE; CONTROLLED STUDY; DISSOCIATION; ENZYME BINDING; ENZYME INHIBITION; HALF LIFE TIME; NONHUMAN; PH; PRIORITY JOURNAL;

EID: 0031026598     PISSN: 87555093     EISSN: None     Source Type: Journal    
DOI: 10.3109/14756369709027647     Document Type: Article

References (26)

1. David, F., Bernard, A.-M., Pierres, M. and Marguet, D. (1993). J. Biol. Chem., 268, 17247-17252.
2. Darmoul, D., Lacasa, M., Baricault, L, Marguet, D., Sapin, C., Trotot, P., Barbat, A. and Trugnan, G. (1992). J. Biol. Chem., 267, 4824-4833.
3. Dang, N.H., Torimoto, Y., Shimamura, K., Tanaka, T., Daley, J.F., Schlossman, S.F. and Morimoto, C. (1991). J. Immunol., 147, 2825-2832.
4. Hegen, M., Neidobitek, G., Klein, C.E., Stein, H. and Fleischer, B. (1990). J. Immunol., 144, 2908-2914.
5. Tanaka, T., Kameoka, J., Yaron, A., Schlossman, S.F. and Morimoto, C. (1993). Proc. Natl. Acad. Sci. USA, 90, 4586-4590.
6. Hegen, M., Mittrücker, H.-W., Hug, R., Demuth, H.-U., Neubert, K., Barth, A. and Fleischer, B. (1993). Immunobiol., 189, 483-493.
7. Flentke, G.R., Munoz, E., Huber, B.T., Plaut, A.G., Kettner, C.A. and Bachovchin, W.W. (1991). Proc. Natl. Acad. Sci. USA, 88, 1556-1559.
8. Kubota, T., Flentke, G.R., Bachovchin, W.W. and Stollar, B.D. (1992). Clin. Exp. Immunol., 89, 192-197.
9. Gutheil, W.G. and Bachovchin, W.W. (1993). Biochemistry, 32, 8723-8731.
10. Bartlett, P.A., Hanson, J.E. and Giannousis, P.P. (1990). J. Org. Chem., 55, 6268-6274.
11. Hanson, J.E., Kaplan, A.P. and Bartlett, P.A. (1989). Biochemistry, 28, 6294-6305.
12. Yoshioka, M., Erickson, R.H., Matsumoto, H., Gum, E. and Kim, Y.S. (1991). Int. J. Cancer, 47, 916-921.
13. Hong, W., Piaza, G.A., Hixson, D.C. and Doyle, D. (1989). Biochemistry, 28, 8474-8479.
14. Snow, R.J., Bachovchin, W.W., Barton, R.W., Campbell, S.J., Coutts, S.J , Freeman, D.M., Kelly, T.A., Kennedy, C.A., Krolikowski, D.A., Leonard, S.F., Pargellis, C.A., Tong, L. and Adams, J. (1994) J. Am. Chem. Soc., 116, 10860-10869.
15. Kelly, T.A., Adams, J., Bachovchin, W.W., Barton, R.W., Campbell, S.J., Coutts, S.J., Kennedy, C.A. and Snow, R.J. (1993). J. Am. Chem. Soc., 115, 12637-12638.
16. Frieden, C., Kurz, L.C and Gilbert, H.R. (1980). Biochemistry, 19, 5303-5309.
17. Pargellis, C.A , Morelock, M.M., Graham, E.T., Kinkade, P., Pav, S., Lubbe, K., Lamarre, D. and Anderson, P.C. (1994). Biochemistry, 33, 12527-12534.
18. Smith, R.E. and Van Frank, R.M. (1975). In Frontiers of Biology Volume 43: Lysosomes in Biology and Pathology (Neuberger, A., Tatum, E.L. (Eds )) pp. 193-249, Amsterdam: North Holland.
19. Matayoshi, E.D., Wang, G T., Krafft, G.A. and Erickson, J. (1990). Science, 247, 954-958.
20. Glasoe, P.K. and Long, F A. (1960). J Phys. Chem., 64, 188-191.
21. Rule, C.K. and LaMer, V.K. (1938) J. Am. Chem. Soc., 60, 1974-1981
22. Cha, S. (1980). Biochem. Pharmacol., 29, 1779-1789.
23. Williams, J.W. and Morrison, J.F (1979) Meth. Enzymol., 63, 437-467
24. Weber, P.C., Lee, S.L., Lewandowski, F.A., Schadt, M.C., Chang, C W. and Kettner, C.A. (1995). Biochemistry, 34, 3750-3757.
25. Morrison, J.F. and Walsh, C.T. (1988). Adv. Enzymol., 61, 201-301.
26. Williams, J.W , Morrison, J.F and Duggleby, R.G. (1979). Biochemistry, 18, 2567-2573.