Syntheses and biological activities of joro spider toxin analogs to spidamine and joramine

Chemical and Pharmaceutical Bulletin

Volumn 45, Issue 1, 1997, Pages 93-100

  Chiba, Tadashige ^a   Akizawa, Toshifumi ^a   Matsukawa, Motomi ^a   Kawai, Nobufumi ^b   Kono, Yoshiaki ^c   Yoshioka, Masanori ^a  

^a SETSUNAN UNIVERSITY   (Japan)

^b Department of Physiology   (Japan)

^c NATIONAL INSTITUTE OF INFECTIOUS DISEASES   (Japan)

Author keywords

excitatory post synaptic potential; insect; joramine; spidamine; spider toxin; synthetic analog

Indexed keywords

GLUTAMATE RECEPTOR; INSECTICIDE; JORAMINE DERIVATIVE; SPIDAMINE DERIVATIVE; SPIDER VENOM; UNCLASSIFIED DRUG;

ARTICLE; BIOASSAY; COCKROACH; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; INSECT CONTROL; LOBSTER; MOSQUITO; NEUROMUSCULAR SYNAPSE; NONHUMAN; SPIDER; STRUCTURE ACTIVITY RELATION;

EID: 0031021640     PISSN: 00092363     EISSN: None     Source Type: Journal    
DOI: 10.1248/cpb.45.93     Document Type: Article

References (24)

1. Chiba T., Akizawa T., Matsukawa M., Nishi M., Kawai N., Yoshioka M., Chem. Pharm. Bull., 44, 972-979 (1996).
2. Teshima T., Matsumoto T., Wakamiya T., Shiba T., Nakajima T., Kawai N., Tetrahedron, 46, 3813-3818 (1990).
3. Kawai N., Nakajima T., J. Toxicol., 9, 203-223 (1990).
4. Chiba T., Akizawa T., Matsukawa M., Pan-Hou H., Yoshioka M., Chem. Pharm. Bull., 42, 1964-1969 (1994).
5. Chiba T., Akizawa T., Matsukawa M., Pan-Hou H., Kawai N., Yoshioka M., Chem. Pharm. Bull., 43, 2177-2181 (1995).
6. Nakanishi K., Goodnow R., Konno K., Niwa M., Bukownik R., Kallimopoulos T. A., Usherwood P., Eldefrawi A. T., Eldefrawi M. E., Pure & Appl. Chem., 62, 1223-1230 (1990).
7. Goodnow R., Konno K., Niwa M., Kallimopoulos T., Bukownik R., Lenares D., Nakanishi K., Tetrahedron, 46, 3267-3286 (1990).
8. Choi S. K., Goodnow R. A., Kalivretenos A., Chiles G. W., Fushiya S., Nakanishi K., Tetrahedron, 48, 4793-4822 (1992).
9. Choi S. K., Nakanishi K., Usherwood P. N. R., Tetrahedron, 49, 5777-5790 (1993).
10. Kalivretenos A. G., Nakanishi K., J. Org. Chem., 58, 6596-6608 (1993).
11. Nakanishi K., Choi S. K., Hwang D., Lerro K., Orlando M., Kalivretenos A. G., Eldefrawi A., Eldefrawi M., Usherwood P. N. R., Pure & Appl. Chem., 66, 671-678 (1994).
12. Choi S. K., Kalivretenos A. G., Usherwood P. N. R., Nakanishi K., Chemistry & Biology, 2, 23-27 (1995).
13. Kono Y., Narai N., Numata M., Yoshioka M., Appl. Ent. Zool., 22, 392-394 (1987).
14. Miyashita M., Matsushita M., Sato H., Toki T., Nakajima T., Irie H., Chem. Lett., 929-932 (1993).
15. Miyashita M., Sato H., Yoshikishi A., Toki T., Matsushita M., Irie H., Yanami T., Kikuchi Y., Takasaki C., Nakajima T., Tetrahedron Lett., 33, 2833-2836 (1992).
16. Miyashita M., Sato H., Matsushita M., Kusumegi Y., Toki T., Yoshikishi A., Yanami T., Kikuchi Y., Takasaki C., Nakajima T., Irie H., Tetrahedron Lett., 33, 2837-2840 (1992).
17. Bycroft B. W., Chan W. C., Hone N. D., Millington S., Nash I. A., J. Am. Chem. Soc., 116, 7415-7416 (1994).
18. Matsushita M., Kanemura T., Hatakeyama S., Irie H., Toki T., Miyashita M., Tetrahedron, 51, 10687-10698 (1995).
19. Matsushita M., Kanemura T., Hatakeyama S., Irie H., Toki T., Miyashita M., Tetrahedron Lett., 36, 5231-5234 (1995).
20. Houssin R., Bernier J. L., Henichart J. P., Synthesis, 1988, 259-261.
21. Mattingly P. G., Synthesis, 1990, 366-368.
22. Atwell G. J., Denny W. A., Synthesis, 1984, 1032-1033.
23. Teshima T., Wakamiya T., Aramaki Y., Nakajima T., Kawai N., Shiba T., Tetrahedron Lett., 28, 3509-3510 (1987).
24. Yoshioka M., Narai N., Kawai N., Numata M., Nakajima T., Biog. Amines, 7, 375-384 (1990).