Pharmacological profiles of a new antiulcer agent, SWR-215

Biological and Pharmaceutical Bulletin

Volumn 20, Issue 1, 1997, Pages 28-35

  Kataoka, Hirohumi ^a   Isoi, Takashi ^a   Kiso, Tatsuya ^a   Tanaka, Chizu ^a   Shinkawa, Ranjun ^a   Kakita, Takao ^a   Shogaki, Takeshi ^a   Furukawa, Masumi ^a   Ohtsubo, Yoshikazu ^a  

^a SAWAI PHARMACEUTICAL CO LTD   (Japan)

Author keywords

gastric acid secretion; H2 receptor antagonist; histamine; mucosal protective effect; roxatidine acetate hydrochloride; SWR 215

Indexed keywords

ALCOHOL; ANTIULCER AGENT; EPIRIZOLE; HISTAMINE; INDOMETACIN; PROSTAGLANDIN; ROXATIDINE; SWR 215; UNCLASSIFIED DRUG; [[(1,2 DIHYDRO 2 OXO 4 QUINOLINYL)METHYL]THIO] N [[[4 (1 PIPERIDINYLMETHYL) 2 PYRIDINYL]OXY] 2 BUTENYL]ACETAMIDE;

ANIMAL CELL; ANIMAL MODEL; ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; DOG; DOSE RESPONSE; DRUG POTENCY; FEMALE; GUINEA PIG; HISTAMINE METABOLISM; MALE; NONHUMAN; ORAL DRUG ADMINISTRATION; PEPTIC ULCER; PROSTAGLANDIN SYNTHESIS; RAT; RECEPTOR BLOCKING; STOMACH ACID SECRETION; STOMACH PROTECTION; ULCER HEALING;

EID: 0031012487     PISSN: 09186158     EISSN: None     Source Type: Journal    
DOI: 10.1248/bpb.20.28     Document Type: Article

References (34)

1. Charlet N., Gallo Torres H. E., Bounameaux Y., Wills R. J., J. Clin. Pharmacol., 25, 564-582 (1985).
2. Ganellin C. R., "Pharmacology of Histamine Receptors," ed. by Ganellin C. R., Parsons M. E., Wright, PSG, Bristol, 1982, pp. 10-102.
3. Bertaccini G., Coruzzi G., Atlas Sci. Pharmacol., 1, 181-186 (1987).
4. Pounder R.E., Pharmacol. Ther., 26, 221-234 (1984).
5. Nakagawa K., Murakami N., Yoshizaki S., Tominaga M., Mori H., Yabuuchi Y., Shintani S., J. Med. Chem., 17, 529-533 (1974).
6. Yoshizaki S., Tanimura K., Tamada S., Yabuuchi Y., Nakagawa K., J. Med. Chem., 19, 1138-1142 (1976).
7. Uchida M., Tabusa F., Komatsu M., Morita S., Kanbe T., Nakagawa K., Chem. Pharm. Bull., 33, 3775-3786 (1985).
8. Yamasaki K., Ishiyama H., Imaizumi T., Kanbe T., Yabuuchi Y., Jpn. J. Pharmacol., 49, 441-448 (1989).
9. Reinhardt D., Wagner J., Schumann H. J., Agents Actions, 4, 217-221 (1974).
10. Arunlakshana O., Schild H. O., Br. J. Pharmacol., 14, 48-58 (1959).
11. Okabe S., Takagi K., Igata H., Kato S., Shimosako K., Yamaji Y., Seiki M., Jpn. J. Pharmacol., 59, 275-289 (1992).
12. Robert V. D., Henry N. H., J. Appl. Physiol., 14, 138-139 (1959).
13. Hung C. R., Okabe S., Kasuya Y., Jpn. J. Pharmacol., 29, 147-150 (1979).
14. Takagi K., Kasuya Y., Watanabe K., Chem. Pharm. Bull., 12, 465-472 (1964).
15. Urushidani T., Okabe S., Takeuchi K., Takagi K., Jpn. J. Pharmacol., 27, 316-319 (1977).
16. Mizui T., Doteuchi M., Jpn. J. Pharmacol., 33, 939-945 (1983).
17. Okabe S., Ishihara Y., Inoo H., Tanaka H., Dig. Dis. Sci., 27, 242-249 (1982).
18. Robert A., Nezamis J. E., Lancaster C., Davis J. P., Field S. O., Hanchar A. J., Am. J. Physiol., 245, G113-G121 (1983).
19. Guddum J., Hameed K. A., Hathway D. E., Stephens F. F., Q. J. Exp. Physiol., 40, 49-74 (1955).
20. Torchiana M. L., Pendleton R. G., Cook P. G., Hanson C. A., Clineschmidt B. V., J. Pharmacol. Exp. Ther., 224, 514-519 (1983).
21. Buyniski J. P., Cavanagh R. L., Pircio A. W., Algieri A. A., Crenshaw R. R., "Highlight in Receptor Chemistry," ed. by Melchiorre C., Giannella M., Elsevier Science Publishers, Amsterdam, 1984, pp. 195-215.
22. Muramatsu M., Hirose-Kijima H., Aihara H., Otomo S., Jpn. J. Pharmacol., 57, 13-23 (1991).
23. Inaba N., Shibata M., Onodera S., Tanaka M., Suzuki T., Yamaura T., Ohnishi H., Folia. Pharmacol. Jpn., 105, 231-241 (1995).
24. Yuki H., Kamato T., Nishida A., Fujihara A., Takeda M., Miyata K., Jpn. J. Pharmacol., 63, 345-351 (1993).
25. Katz L. B., Scott C. K., Shriver D. A., J. Pharmacol. Exp. Ther., 238, 587-593 (1986).
26. Katz L. B., Tobia A. J., Shriver D. A., J. Pharmacol. Exp. Ther., 242, 437-442 (1987).
27. Bertaccini G., Coruzzi G., Poli E., Adami M., Agents Actions, 19, 180-187 (1986).
28. Hayase M., Takeuchi K., Dig. Dis. Sci., 31, 166-171 (1986).
29. Arai I., Hirose H., Muramatsu M., Aihara H., Physiology Behavior, 40, 357-361 (1987).
30. Ishihara Y., Yamada Y., Hata Y., Okabe S., Dig. Dis. Sci., 28, 552-558 (1983).
31. Tanaka H., Ueki S., Ohno T., Takeuchi K., Okabe S., Jpn. J. Pharmacol., 42, 383-396 (1986).
32. Okada M., Niida H., Takeuchi K., Okabe S., Dig. Dis. Sci., 34, 694-702 (1989).
33. Ueki S., Takeuchi K., Okabe S., Dig. Dis. Sci., 33, 209-216 (1988).
34. Hui W. M., Chen B. W., Cho C. H., Luk C. T., Lam S. K., Digestion, 48, 113-120 (1991).