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Volumn 40, Issue 1, 1997, Pages 17-34

Pharmacological profile of LY301317, a potent and selective 5-HT(1A) agonist

Author keywords

5 HT(1A); Drug discrimination; Emesis; Forced swim; Punished responding

Indexed keywords

5 HYDROXYINDOLEACETIC ACID; CISPLATIN; HISTAMINE H1 RECEPTOR; IPECAC; RECEPTOR SUBTYPE; SEROTONIN 1A AGONIST; SEROTONIN 1A RECEPTOR; SEROTONIN 1D RECEPTOR;

EID: 0031011681     PISSN: 02724391     EISSN: None     Source Type: Journal    
DOI: 10.1002/(SICI)1098-2299(199701)40:1<17::AID-DDR2>3.0.CO;2-W     Document Type: Article
Times cited : (10)

References (87)
  • 1
    • 0025917723 scopus 로고
    • 3 receptor antagonists: An overview of their present status and future potential in cancer therapy-induced emesis
    • 3 receptor antagonists: An overview of their present status and future potential in cancer therapy-induced emesis. Drugs 42:551-568.
    • (1991) Drugs , vol.42 , pp. 551-568
    • Aapro, M.1
  • 4
    • 0001331734 scopus 로고
    • The 5-hydroxytryptamine receptor antagonists as antiemetics: Preclinical evaluation and mechanisms of action
    • Andrews PLR, Bhandari P (1993): The 5-hydroxytryptamine receptor antagonists as antiemetics: Preclinical evaluation and mechanisms of action. Eur J Cancer 29A:S11-S16.
    • (1993) Eur J Cancer , vol.29 A
    • Andrews, P.L.R.1    Bhandari, P.2
  • 5
    • 0025348385 scopus 로고
    • The role of anxiety in the development of anticipatory nausea in cancer chemotherapy: A review and synthesis
    • Andrykowski M (1990): The role of anxiety in the development of anticipatory nausea in cancer chemotherapy: A review and synthesis. Psychosom Med 52:458-475.
    • (1990) Psychosom Med , vol.52 , pp. 458-475
    • Andrykowski, M.1
  • 6
    • 0001334294 scopus 로고
    • A technique for delivering shock to pigeons
    • Azrin NH (1959): A technique for delivering shock to pigeons. J Exp Anal Behav 2:161-163.
    • (1959) J Exp Anal Behav , vol.2 , pp. 161-163
    • Azrin, N.H.1
  • 8
    • 0026633686 scopus 로고
    • 1A receptor antagonists BMY 7378 and NAN-190
    • 1A receptor antagonists BMY 7378 and NAN-190. Eur J Pharmacol 217:163-171.
    • (1992) Eur J Pharmacol , vol.217 , pp. 163-171
    • Barrett, J.E.1    Gleeson, S.2
  • 10
    • 0027323919 scopus 로고
    • Antidepressant-like effect of LY228729 as measured in the rodent forced swim paradigm
    • Benvenga M, Leander JD (1993): Antidepressant-like effect of LY228729 as measured in the rodent forced swim paradigm. Eur J Pharmacol 239:249-252.
    • (1993) Eur J Pharmacol , vol.239 , pp. 249-252
    • Benvenga, M.1    Leander, J.D.2
  • 11
    • 0029073180 scopus 로고
    • Olanzapine, an atypical antipsychotic, increases rates of punished responding in pigeons
    • Benvenga MJ, Leander JD (1995): Olanzapine, an atypical antipsychotic, increases rates of punished responding in pigeons. Psychopharmacology 119:133-138.
    • (1995) Psychopharmacology , vol.119 , pp. 133-138
    • Benvenga, M.J.1    Leander, J.D.2
  • 12
    • 0030446738 scopus 로고    scopus 로고
    • 1A agnosis in pigeons are dependent on the level of response suppression
    • 1A agnosis in pigeons are dependent on the level of response suppression. Behav Pharmacol 6:540-550.
    • (1996) Behav Pharmacol , vol.6 , pp. 540-550
    • Benvenga, M.1    Leander, J.D.2
  • 17
    • 0023481665 scopus 로고
    • Conditioned side effects induced by cancer chemotherapy: Prevention through behavioral treatment
    • Burish TG, Carey MP, Krozely MG, Greco FA (1987): Conditioned side effects induced by cancer chemotherapy: Prevention through behavioral treatment. J Consult Clin Psychol 55:42-18.
    • (1987) J Consult Clin Psychol , vol.55 , pp. 42-118
    • Burish, T.G.1    Carey, M.P.2    Krozely, M.G.3    Greco, F.A.4
  • 18
    • 0017165533 scopus 로고
    • Beta adrenergic receptor binding in membrane preparations from mammalian brain
    • Bylund D, Snyder S (1976): Beta adrenergic receptor binding in membrane preparations from mammalian brain. Mol Pharmacol 12:568-580.
    • (1976) Mol Pharmacol , vol.12 , pp. 568-580
    • Bylund, D.1    Snyder, S.2
  • 23
    • 0022390340 scopus 로고
    • A stimulator of laboratory studies of motion sickness in cats
    • Crampton GH, Lucot JB (1985): A stimulator of laboratory studies of motion sickness in cats. Aviat Space Environ Med 56:462-465.
    • (1985) Aviat Space Environ Med , vol.56 , pp. 462-465
    • Crampton, G.H.1    Lucot, J.B.2
  • 25
    • 0025613807 scopus 로고
    • Serotonin and appetite
    • Curzon G (1990): Serotonin and appetite. Ann NY Acad Sci 600:521-531.
    • (1990) Ann NY Acad Sci , vol.600 , pp. 521-531
    • Curzon, G.1
  • 26
    • 0027166318 scopus 로고
    • 1A agonists in anxiety and depression
    • 1A agonists in anxiety and depression. J Psychopharmocol 7:283-289.
    • (1993) J Psychopharmocol , vol.7 , pp. 283-289
    • Deakin, J.F.W.1
  • 28
    • 0028990742 scopus 로고
    • 1A receptor agonists: Recent developments and controversial issues
    • 1A receptor agonists: Recent developments and controversial issues. Psychopharmacology 121:1-26.
    • (1995) Psychopharmacology , vol.121 , pp. 1-26
    • De Vry, J.1
  • 31
    • 13344283445 scopus 로고    scopus 로고
    • Serotonin receptors involved in regulation of pituitary-adrenocortical function in rats
    • Fuller RW (1996): Serotonin receptors involved in regulation of pituitary-adrenocortical function in rats. Behav Brain Res 73:215-219.
    • (1996) Behav Brain Res , vol.73 , pp. 215-219
    • Fuller, R.W.1
  • 32
    • 0024560609 scopus 로고
    • Effects of buspirone and its metabolite, 1-(2-pyrimidinyl)piperazine, on brain monoamines and their metabolites in rats
    • Fuller RW, Perry KW (1989): Effects of buspirone and its metabolite, 1-(2-pyrimidinyl)piperazine, on brain monoamines and their metabolites in rats. J Pharmacol Exp Ther 248:50-56.
    • (1989) J Pharmacol Exp Ther , vol.248 , pp. 50-56
    • Fuller, R.W.1    Perry, K.W.2
  • 33
    • 0024992869 scopus 로고
    • Serotonin receptor subtypes involved in the elevation of serum corticosterone concentration in rats by direct- And indirect acting serotonin agonists
    • Fuller RW, Snoddy HD (1990): Serotonin receptor subtypes involved in the elevation of serum corticosterone concentration in rats by direct-and indirect acting serotonin agonists. Neuroendocrinology 52:206-211.
    • (1990) Neuroendocrinology , vol.52 , pp. 206-211
    • Fuller, R.W.1    Snoddy, H.D.2
  • 34
    • 0012297220 scopus 로고
    • Characterization of the 5-HT receptor subtype mediating ACTH release in the rat
    • Gilbert F, Stahl Sm, Tricklebank MD (1987): Characterization of the 5-HT receptor subtype mediating ACTH release in the rat. Br J Pharmacol 91:495P.
    • (1987) Br J Pharmacol , vol.91
    • Gilbert, F.1    Stahl, Sm.2    Tricklebank, M.D.3
  • 35
    • 0025232511 scopus 로고
    • Serotonin receptors: Clinical implications
    • Glennon RA (1990): Serotonin receptors: Clinical implications. Neurosci Biobehav Rev 14:35-47.
    • (1990) Neurosci Biobehav Rev , vol.14 , pp. 35-47
    • Glennon, R.A.1
  • 36
    • 0018332473 scopus 로고
    • 3H]prazosin to rat brain alpha adrenergic receptors
    • 3H]prazosin to rat brain alpha adrenergic receptors. Eur J Pharmacol 55:323-328.
    • (1979) Eur J Pharmacol , vol.55 , pp. 323-328
    • Greengrass, P.1    Bremner, R.2
  • 40
    • 0021956188 scopus 로고
    • Hypothermia in the rat induced by the potent serotonergic agent, 8-OH-DPAT
    • Hjorth S (1985): Hypothermia in the rat induced by the potent serotonergic agent, 8-OH-DPAT. J Neural Transm 62:131-135.
    • (1985) J Neural Transm , vol.62 , pp. 131-135
    • Hjorth, S.1
  • 41
    • 0019936569 scopus 로고
    • Buspirone: Effects on central monoaminergic transmission - Possible relevance to animal experimental and clinical findings
    • Hjorth S, Carlsson A (1982): Buspirone: Effects on central monoaminergic transmission - possible relevance to animal experimental and clinical findings. Eur J Pharmacol 83:299-303.
    • (1982) Eur J Pharmacol , vol.83 , pp. 299-303
    • Hjorth, S.1    Carlsson, A.2
  • 42
    • 0024203466 scopus 로고
    • 1A receptor agonist, 8-OH-DPAT, preferentially activates cell body autoreceptors in rat brain in vivo
    • 1A receptor agonist, 8-OH-DPAT, preferentially activates cell body autoreceptors in rat brain in vivo. Naunyn Schmeidbergs Arch Pharmacol 338:463-471.
    • (1988) Naunyn Schmeidbergs Arch Pharmacol , vol.338 , pp. 463-471
    • Hjorth, S.1    Magnusson, T.2
  • 49
    • 0025236582 scopus 로고
    • Animal studies in the study of vomiting
    • King GL (1990): Animal studies in the study of vomiting. Can J Pharmacol 68:260-268.
    • (1990) Can J Pharmacol , vol.68 , pp. 260-268
    • King, G.L.1
  • 51
    • 0024478025 scopus 로고
    • 3 receptors prevents cisplatin-induced but not motion- or xylazine-induced emesis in the cat
    • 3 receptors prevents cisplatin-induced but not motion-or xylazine-induced emesis in the cat. Pharmacol Biochem Behav 32:207-210.
    • (1989) Pharmacol Biochem Behav , vol.32 , pp. 207-210
    • Lucot, J.B.1
  • 52
    • 0028009855 scopus 로고
    • Antiemetic effects of flesinoxin in cats: Comparisons with 8-hydroxy-2-(di-n-propylamino)tetralin
    • Lucot J (1994): Antiemetic effects of flesinoxin in cats: Comparisons with 8-hydroxy-2-(di-n-propylamino)tetralin. Eur J Pharmacol 253:53-60.
    • (1994) Eur J Pharmacol , vol.253 , pp. 53-60
    • Lucot, J.1
  • 53
    • 0024455229 scopus 로고
    • 8-OH-DPAT suppresses vomiting in the cat elicited by motion, cisplatin, or xylazine
    • Lucot J, Crampton G (1989): 8-OH-DPAT suppresses vomiting in the cat elicited by motion, cisplatin, or xylazine. Pharmacol Biochem Behav 33:627-631.
    • (1989) Pharmacol Biochem Behav , vol.33 , pp. 627-631
    • Lucot, J.1    Crampton, G.2
  • 54
    • 0028027657 scopus 로고
    • 1A receptor-mediated regulation of plasma neuroendocrine hormones
    • 1A receptor-mediated regulation of plasma neuroendocrine hormones. J Pharmacol Exp Ther 271:1246-1252.
    • (1994) J Pharmacol Exp Ther , vol.271 , pp. 1246-1252
    • Meller, E.1    Bohmaker, K.2
  • 56
    • 0025697462 scopus 로고
    • Role of serotonin in depression
    • Meltzer HY (1990): Role of serotonin in depression. Ann NY Acad Sci 600:486-500.
    • (1990) Ann NY Acad Sci , vol.600 , pp. 486-500
    • Meltzer, H.Y.1
  • 58
    • 0027486344 scopus 로고
    • Induction of hypothermia as a model of 5-hydroxytryptamine receptor-mediated activity in the rat: A pharmacological characterization of the actions of novel agonists and antagonists
    • Millan MJ, Rivet J-M, Canton H, Le Marouille-Girardon S, Gober A (1993): Induction of hypothermia as a model of 5-hydroxytryptamine receptor-mediated activity in the rat: A pharmacological characterization of the actions of novel agonists and antagonists. J Pharmacol Exp Ther 264:1364-1376.
    • (1993) J Pharmacol Exp Ther , vol.264 , pp. 1364-1376
    • Millan, M.J.1    Rivet, J.-M.2    Canton, H.3    Le Marouille-Girardon, S.4    Gober, A.5
  • 60
    • 0019061918 scopus 로고
    • Ligand: A versatile computerized approach for characterization of ligand-binding systems
    • Munson PJ, Rodbard JD (1980): Ligand: A versatile computerized approach for characterization of ligand-binding systems. Anal Biochem 107:220-239.
    • (1980) Anal Biochem , vol.107 , pp. 220-239
    • Munson, P.J.1    Rodbard, J.D.2
  • 62
    • 0028913581 scopus 로고
    • 3 receptor antagonists for chemotherapy-induced emesis
    • 3 receptor antagonists for chemotherapy-induced emesis. J Clin Oncol 13:1036-1043.
    • (1995) J Clin Oncol , vol.13 , pp. 1036-1043
    • Perez, E.A.1
  • 63
    • 0017618768 scopus 로고
    • Depression: A new animal model sensitive to antidepressant treatments
    • Porsolt RD, LePichon MMJ (1977): Depression: A new animal model sensitive to antidepressant treatments. Nature 266:730.
    • (1977) Nature , vol.266 , pp. 730
    • Porsolt, R.D.1    LePichon, M.M.J.2
  • 65
    • 0004679802 scopus 로고
    • The effect of "broad spectrum" antiemetic drugs on nicotine-induced emesis in the Suncus murinus
    • Rudd JA, Naylor RJ (1995): The effect of "broad spectrum" antiemetic drugs on nicotine-induced emesis in the Suncus murinus. Br J Pharmacol 114:385.
    • (1995) Br J Pharmacol , vol.114 , pp. 385
    • Rudd, J.A.1    Naylor, R.J.2
  • 66
    • 0000718648 scopus 로고
    • The effect of 8-OH-DPAT on drug-induced emesis in the ferret
    • Rudd JR, Bunce KT, Naylor RJ (1992): The effect of 8-OH-DPAT on drug-induced emesis in the ferret. Br J Pharmacol 106:101.
    • (1992) Br J Pharmacol , vol.106 , pp. 101
    • Rudd, J.R.1    Bunce, K.T.2    Naylor, R.J.3
  • 68
    • 0027277135 scopus 로고
    • 1A receptor ligands in animal models of anxiety, impulsivity and depression: Multiple mechanisms of action?
    • 1A receptor ligands in animal models of anxiety, impulsivity and depression: Multiple mechanisms of action? Pro Neuro Psychopharmacol Biol Psychiatry 17:87-104.
    • (1993) Pro Neuro Psychopharmacol Biol Psychiatry , vol.17 , pp. 87-104
    • Schreiber, R.1    De Vry, J.2
  • 69
    • 0027136728 scopus 로고
    • 1A receptor agonists 8-OH-DPAT and ipsapirone in the rat forced swimming test
    • 1A receptor agonists 8-OH-DPAT and ipsapirone in the rat forced swimming test. Behav Pharmacol 4:625-636.
    • (1993) Behav Pharmacol , vol.4 , pp. 625-636
    • Schreiber, R.1    De Vry, J.2
  • 73
    • 7144227374 scopus 로고    scopus 로고
    • Serotonergic control of the organization of feeding and satiety
    • Simansky KJ (1996): Serotonergic control of the organization of feeding and satiety. Behav Brain Res 73:37-42.
    • (1996) Behav Brain Res , vol.73 , pp. 37-42
    • Simansky, K.J.1
  • 75
    • 1842334586 scopus 로고
    • An evaluation of a method for determination of free corticosteroids in minute quantities of mouse plasma
    • Solem JH, Brink-Johnsen (1965): An evaluation of a method for determination of free corticosteroids in minute quantities of mouse plasma. Scand J Clin Invest 17(Suppl 80):1-14.
    • (1965) Scand J Clin Invest , vol.17 , Issue.80 SUPPL. , pp. 1-14
    • Solem, J.H.1    Brink-Johnsen2
  • 77
    • 0025693902 scopus 로고
    • Serotonergic agents in anxiety
    • Taylor DP (1990): Serotonergic agents in anxiety. Ann NY Acad Sci 600:545-557.
    • (1990) Ann NY Acad Sci , vol.600 , pp. 545-557
    • Taylor, D.P.1
  • 80
    • 0025296047 scopus 로고
    • 1A agonists measured with the forced swim assay
    • 1A agonists measured with the forced swim assay. Psychopharmacology 101:497-504.
    • (1990) Psychopharmacology , vol.101 , pp. 497-504
    • Wieland, S.1    Lucki, I.2
  • 81
    • 0018332925 scopus 로고
    • 3]muscimol, a potent gamma aminobutyric acid agonist, to rat brain synaptosomal membranes using liltration assay
    • 3]muscimol, a potent gamma aminobutyric acid agonist, to rat brain synaptosomal membranes using liltration assay. J Neurochem 32:713-718.
    • (1979) J Neurochem , vol.32 , pp. 713-718
    • Williams, M.1    Risley, E.2
  • 82
    • 0021348560 scopus 로고
    • The validity of animal models of depression
    • Willner P (1984): The validity of animal models of depression. Psychopharmacology 83:1-16.
    • (1984) Psychopharmacology , vol.83 , pp. 1-16
    • Willner, P.1
  • 85
    • 1842301210 scopus 로고    scopus 로고
    • 1A selective compounds with mixed agonist/antagonist properties
    • 1A selective compounds with mixed agonist/antagonist properties. Soc Neurosci Abst 22:1586.
    • (1996) Soc Neurosci Abst , vol.22 , pp. 1586
    • Wolff, M.C.1    Leander, J.D.2
  • 87
    • 0016159582 scopus 로고
    • Muscarinic cholinergic binding in rat brain
    • Yamamura H, Snyder S (1974): Muscarinic cholinergic binding in rat brain. Proc Natl Acad Sci USA 71:1725-1729.
    • (1974) Proc Natl Acad Sci USA , vol.71 , pp. 1725-1729
    • Yamamura, H.1    Snyder, S.2


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