-
1
-
-
0029073127
-
Specific mutations in the estrogen receptor change the properties of an antiestrogen to full agonists
-
Mahfoudi A., Roulet E., Dauvois S., Parker M. G. and Wahli W., Specific mutations in the estrogen receptor change the properties of an antiestrogen to full agonists. Proc. Natl. Acad. Sci. U.S.A. 92 (1995) 4206-4210.
-
(1995)
Proc. Natl. Acad. Sci. U.S.A.
, vol.92
, pp. 4206-4210
-
-
Mahfoudi, A.1
Roulet, E.2
Dauvois, S.3
Parker, M.G.4
Wahli, W.5
-
2
-
-
0029616211
-
Ligand-dependent, transcriptionally productive association of the amino- and carboxyl-terminal regions of a steroid hormone nuclear receptor
-
Kraus W. L., McInerney E. M. and Katzenellenbogen B. S., Ligand-dependent, transcriptionally productive association of the amino- and carboxyl-terminal regions of a steroid hormone nuclear receptor. Proc. Natl. Acad. Sci. U.S.A. 92 (1995) 12314-12318.
-
(1995)
Proc. Natl. Acad. Sci. U.S.A.
, vol.92
, pp. 12314-12318
-
-
Kraus, W.L.1
McInerney, E.M.2
Katzenellenbogen, B.S.3
-
3
-
-
0029978077
-
Human estrogen receptor ligand activity inversion mutants: Receptors that interpret antiestrogens as estrogens and estrogens as antiestrogens and discriminate among different antiestrogens
-
Montano M. M., Ekena K., Krueger K. D., Keller A. L. and Katzenellenbogen B. S., Human estrogen receptor ligand activity inversion mutants: receptors that interpret antiestrogens as estrogens and estrogens as antiestrogens and discriminate among different antiestrogens. Molec. Endocr. 10 (1996) 230-241.
-
(1996)
Molec. Endocr.
, vol.10
, pp. 230-241
-
-
Montano, M.M.1
Ekena, K.2
Krueger, K.D.3
Keller, A.L.4
Katzenellenbogen, B.S.5
-
4
-
-
0001559063
-
A new approach to breast cancer therapy - total estrogen ablation with pure antiestrogens
-
ed. V. C. Jordan. The University of Wisconsin Press, Madison, WI
-
Wakeling A. E., A new approach to breast cancer therapy - total estrogen ablation with pure antiestrogens. In Long-term Tamoxifen Treatment for Breast Cancer, ed. V. C. Jordan. The University of Wisconsin Press, Madison, WI, 1994, pp. 219-234.
-
(1994)
Long-term Tamoxifen Treatment for Breast Cancer
, pp. 219-234
-
-
Wakeling, A.E.1
-
5
-
-
0023915865
-
Contrasting action of tamoxifen on endometrial and breast tumor growth in the athymic mouse
-
Gottardis M. M., Robinson S. P., Satyaswaroop P. G. and Jordan V. C., Contrasting action of tamoxifen on endometrial and breast tumor growth in the athymic mouse. Cancer Res. 48 (1988) 812-815.
-
(1988)
Cancer Res.
, vol.48
, pp. 812-815
-
-
Gottardis, M.M.1
Robinson, S.P.2
Satyaswaroop, P.G.3
Jordan, V.C.4
-
6
-
-
0023760993
-
Development of tamoxifen-stimulated growth of MCF-7 tumors in athymic mice after long-term antiestrogen administration
-
Gottardis M. M. and Jordan V. C., Development of tamoxifen-stimulated growth of MCF-7 tumors in athymic mice after long-term antiestrogen administration. Cancer Res. 48 (1988) 5183-5187.
-
(1988)
Cancer Res.
, vol.48
, pp. 5183-5187
-
-
Gottardis, M.M.1
Jordan, V.C.2
-
7
-
-
0029075872
-
Comparison of the effects of a pure steroidal antiestrogen with those of tamoxifen in a model of human breast cancer
-
Osborne C. K., Coronado-Heinsohn E. B., Hilsenbeck S. G., McCue B. L., Wakeling A. E., McClelland R. A., Manning D. L. and Nicholson R. I., Comparison of the effects of a pure steroidal antiestrogen with those of tamoxifen in a model of human breast cancer. J. Natl. Cancer Inst. 87 (1995) 746-750.
-
(1995)
J. Natl. Cancer Inst.
, vol.87
, pp. 746-750
-
-
Osborne, C.K.1
Coronado-Heinsohn, E.B.2
Hilsenbeck, S.G.3
McCue, B.L.4
Wakeling, A.E.5
McClelland, R.A.6
Manning, D.L.7
Nicholson, R.I.8
-
8
-
-
0030203362
-
An analysis of tamoxifen-stimulated human carcinomas for mutations in the AF-2 region of the estrogen receptor
-
Bilimoria M. M., Assikis V. J., Muenzner H. D., Wolf D. M., Satyaswaroop P. G. and Jordan V. C., An analysis of tamoxifen-stimulated human carcinomas for mutations in the AF-2 region of the estrogen receptor. J. Steroid Biochem. Molec. Biol. 58 (1996) 479-488.
-
(1996)
J. Steroid Biochem. Molec. Biol.
, vol.58
, pp. 479-488
-
-
Bilimoria, M.M.1
Assikis, V.J.2
Muenzner, H.D.3
Wolf, D.M.4
Satyaswaroop, P.G.5
Jordan, V.C.6
-
9
-
-
0028144926
-
Characterization of tamoxifen stimulated MCF-7 tumor variants grown in athymic mice
-
Wolf D. M. and Jordan V. C., Characterization of tamoxifen stimulated MCF-7 tumor variants grown in athymic mice. Breast Cancer Res. Treat. 31 (1994) 117-127.
-
(1994)
Breast Cancer Res. Treat.
, vol.31
, pp. 117-127
-
-
Wolf, D.M.1
Jordan, V.C.2
-
10
-
-
0028093565
-
The estrogen receptor from a tamoxifen stimulated MCF-7 tumor variant contains a point mutation in the ligand binding domain
-
Wolf D. M. and Jordan V. C., The estrogen receptor from a tamoxifen stimulated MCF-7 tumor variant contains a point mutation in the ligand binding domain. Breast Cancer Res. Treat. 31 (1994) 129-138.
-
(1994)
Breast Cancer Res. Treat.
, vol.31
, pp. 129-138
-
-
Wolf, D.M.1
Jordan, V.C.2
-
11
-
-
0029154750
-
A naturally occurring estrogen receptor mutation results in increased estrogenicity of a tamoxifen analogue
-
Catherino W. H., Wolf D. M. and Jordan V. C., A naturally occurring estrogen receptor mutation results in increased estrogenicity of a tamoxifen analogue. Molec. Endocr. 9 (1995) 1053-1063.
-
(1995)
Molec. Endocr.
, vol.9
, pp. 1053-1063
-
-
Catherino, W.H.1
Wolf, D.M.2
Jordan, V.C.3
-
12
-
-
0029017926
-
Transforming growth factor α: Expression, regulation, and biological activities
-
Lee D. C., Fenton S. E., Berkowitz E. A. and Hissong M. A., Transforming growth factor α: expression, regulation, and biological activities. Pharmacol. Rev. 47 (1995) 51-85.
-
(1995)
Pharmacol. Rev.
, vol.47
, pp. 51-85
-
-
Lee, D.C.1
Fenton, S.E.2
Berkowitz, E.A.3
Hissong, M.A.4
-
13
-
-
0027946822
-
Inhibition of estrogen-induced breast cancer cell proliferation by reduction in autocrine transforming growth factor alpha expression
-
Reddy K. B., Yee D., Hilsenbeck S. G., Coffey R. J. and Osborne C. K., Inhibition of estrogen-induced breast cancer cell proliferation by reduction in autocrine transforming growth factor alpha expression. Cell Growth Differen. 5 (1994) 1275-1282.
-
(1994)
Cell Growth Differen.
, vol.5
, pp. 1275-1282
-
-
Reddy, K.B.1
Yee, D.2
Hilsenbeck, S.G.3
Coffey, R.J.4
Osborne, C.K.5
-
14
-
-
0028558331
-
Transfection of human estrogen receptor (ER) cDNA into ER-negative mammalian cell lines
-
Levenson A. S. and Jordan V. C., Transfection of human estrogen receptor (ER) cDNA into ER-negative mammalian cell lines. J. Steroid Biochem. Molec. Biol 51 (1994) 229-239.
-
(1994)
J. Steroid Biochem. Molec. Biol
, vol.51
, pp. 229-239
-
-
Levenson, A.S.1
Jordan, V.C.2
-
15
-
-
0026520381
-
Growth regulation of estrogen receptor-negative breast cancer cells transfected with complementary DNAs for estrogen receptor
-
Jiang S. Y. and Jordan V. C., Growth regulation of estrogen receptor-negative breast cancer cells transfected with complementary DNAs for estrogen receptor. J. Natl. Cancer Inst. 84 (1992) 580-591.
-
(1992)
J. Natl. Cancer Inst.
, vol.84
, pp. 580-591
-
-
Jiang, S.Y.1
Jordan, V.C.2
-
16
-
-
0018850985
-
A simple, rapid, and sensitive DNA assay procedure
-
LaBarca C. and Paigen K., A simple, rapid, and sensitive DNA assay procedure. Analyt. Biochem. 102 (1980) 344-352.
-
(1980)
Analyt. Biochem.
, vol.102
, pp. 344-352
-
-
LaBarca, C.1
Paigen, K.2
-
17
-
-
0028128432
-
Paradoxical regulation of estrogen-dependent growth factor gene expression in estrogen receptor (ER) negative human breast cancer cells stably expressing ER
-
Jeng M. H., Jiang S. Y. and Jordan V. C., Paradoxical regulation of estrogen-dependent growth factor gene expression in estrogen receptor (ER) negative human breast cancer cells stably expressing ER. Cancer Lett. 82 (1994) 123-128.
-
(1994)
Cancer Lett.
, vol.82
, pp. 123-128
-
-
Jeng, M.H.1
Jiang, S.Y.2
Jordan, V.C.3
-
18
-
-
0028167482
-
Raloxifene (LY 139481HCL) prevents bone loss and reduces serum cholesterol without causing uterine hypertrophy in ovariectomized rats
-
Black L. J., Sato M., Rowley E. R., Magee D. E., Bekele A., Williams D. C., Cullinan G. L., Bendele R., Kauffman R. F., Bensch W. R., Frolik C. A., Termine J. D. and Bryant H. U., Raloxifene (LY 139481HCL) prevents bone loss and reduces serum cholesterol without causing uterine hypertrophy in ovariectomized rats. J. Clin. Invest. 93 (1994) 63-69.
-
(1994)
J. Clin. Invest.
, vol.93
, pp. 63-69
-
-
Black, L.J.1
Sato, M.2
Rowley, E.R.3
Magee, D.E.4
Bekele, A.5
Williams, D.C.6
Cullinan, G.L.7
Bendele, R.8
Kauffman, R.F.9
Bensch, W.R.10
Frolik, C.A.11
Termine, J.D.12
Bryant, H.U.13
-
19
-
-
0020694796
-
Antagonism of estrogen action with a new benzothiophene derived antiestrogen
-
Black L. J., Jones C. D. and Falcone J. F., Antagonism of estrogen action with a new benzothiophene derived antiestrogen. Life Sci. 32 (1993) 1031-1036.
-
(1993)
Life Sci.
, vol.32
, pp. 1031-1036
-
-
Black, L.J.1
Jones, C.D.2
Falcone, J.F.3
-
20
-
-
0029074473
-
Use of pure antiestrogens to elucidate the mode of action of estrogens
-
Wakeling A. E., Use of pure antiestrogens to elucidate the mode of action of estrogens. Biochem. Pharmacol 49 (1995) 1545-1549.
-
(1995)
Biochem. Pharmacol
, vol.49
, pp. 1545-1549
-
-
Wakeling, A.E.1
-
21
-
-
0023663885
-
Functional domains of the human estrogen receptor
-
Kumar V., Green S., Stack G., Berry M., Jin J. R. and Chambon P., Functional domains of the human estrogen receptor. Cell 51 (1987) 941-951.
-
(1987)
Cell
, vol.51
, pp. 941-951
-
-
Kumar, V.1
Green, S.2
Stack, G.3
Berry, M.4
Jin, J.R.5
Chambon, P.6
-
22
-
-
0023712331
-
The hormone-binding domains of the estrogen and glucocorticoid receptors contain an inducible transcription activation function
-
Webster N. J., Green S., Jin J. R. and Chambon P., The hormone-binding domains of the estrogen and glucocorticoid receptors contain an inducible transcription activation function. Cell 54 (1988) 199-207.
-
(1988)
Cell
, vol.54
, pp. 199-207
-
-
Webster, N.J.1
Green, S.2
Jin, J.R.3
Chambon, P.4
-
23
-
-
0026591464
-
Mechanisms of antihormone action
-
Gronemeyer H., Benhamou B., Berry M., Bocquel M. T., Gofflo D., Garcia T., Lerouge T., Metzger D., Meyer M. E., Tora L., Vergezac A. and Chambon P., Mechanisms of antihormone action. J. Steroid Biochem. Molec. Biol. 41 (1992) 217-221.
-
(1992)
J. Steroid Biochem. Molec. Biol.
, vol.41
, pp. 217-221
-
-
Gronemeyer, H.1
Benhamou, B.2
Berry, M.3
Bocquel, M.T.4
Gofflo, D.5
Garcia, T.6
Lerouge, T.7
Metzger, D.8
Meyer, M.E.9
Tora, L.10
Vergezac, A.11
Chambon, P.12
|