메뉴 건너뛰기




Volumn 60, Issue 5-6, 1997, Pages 261-268

Estrogenic activity is increased for an antiestrogen by a natural mutation of the estrogen receptor

Author keywords

[No Author keywords available]

Indexed keywords

ANTIESTROGEN; ESTRADIOL; ESTROGEN RECEPTOR; FULVESTRANT; MESSENGER RNA; RALOXIFENE; TAMOXIFEN; TRANSCRIPTION FACTOR; TRANSFORMING GROWTH FACTOR ALPHA;

EID: 0031008040     PISSN: 09600760     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-0760(96)00184-7     Document Type: Article
Times cited : (83)

References (23)
  • 1
    • 0029073127 scopus 로고
    • Specific mutations in the estrogen receptor change the properties of an antiestrogen to full agonists
    • Mahfoudi A., Roulet E., Dauvois S., Parker M. G. and Wahli W., Specific mutations in the estrogen receptor change the properties of an antiestrogen to full agonists. Proc. Natl. Acad. Sci. U.S.A. 92 (1995) 4206-4210.
    • (1995) Proc. Natl. Acad. Sci. U.S.A. , vol.92 , pp. 4206-4210
    • Mahfoudi, A.1    Roulet, E.2    Dauvois, S.3    Parker, M.G.4    Wahli, W.5
  • 2
    • 0029616211 scopus 로고
    • Ligand-dependent, transcriptionally productive association of the amino- and carboxyl-terminal regions of a steroid hormone nuclear receptor
    • Kraus W. L., McInerney E. M. and Katzenellenbogen B. S., Ligand-dependent, transcriptionally productive association of the amino- and carboxyl-terminal regions of a steroid hormone nuclear receptor. Proc. Natl. Acad. Sci. U.S.A. 92 (1995) 12314-12318.
    • (1995) Proc. Natl. Acad. Sci. U.S.A. , vol.92 , pp. 12314-12318
    • Kraus, W.L.1    McInerney, E.M.2    Katzenellenbogen, B.S.3
  • 3
    • 0029978077 scopus 로고    scopus 로고
    • Human estrogen receptor ligand activity inversion mutants: Receptors that interpret antiestrogens as estrogens and estrogens as antiestrogens and discriminate among different antiestrogens
    • Montano M. M., Ekena K., Krueger K. D., Keller A. L. and Katzenellenbogen B. S., Human estrogen receptor ligand activity inversion mutants: receptors that interpret antiestrogens as estrogens and estrogens as antiestrogens and discriminate among different antiestrogens. Molec. Endocr. 10 (1996) 230-241.
    • (1996) Molec. Endocr. , vol.10 , pp. 230-241
    • Montano, M.M.1    Ekena, K.2    Krueger, K.D.3    Keller, A.L.4    Katzenellenbogen, B.S.5
  • 4
    • 0001559063 scopus 로고
    • A new approach to breast cancer therapy - total estrogen ablation with pure antiestrogens
    • ed. V. C. Jordan. The University of Wisconsin Press, Madison, WI
    • Wakeling A. E., A new approach to breast cancer therapy - total estrogen ablation with pure antiestrogens. In Long-term Tamoxifen Treatment for Breast Cancer, ed. V. C. Jordan. The University of Wisconsin Press, Madison, WI, 1994, pp. 219-234.
    • (1994) Long-term Tamoxifen Treatment for Breast Cancer , pp. 219-234
    • Wakeling, A.E.1
  • 5
    • 0023915865 scopus 로고
    • Contrasting action of tamoxifen on endometrial and breast tumor growth in the athymic mouse
    • Gottardis M. M., Robinson S. P., Satyaswaroop P. G. and Jordan V. C., Contrasting action of tamoxifen on endometrial and breast tumor growth in the athymic mouse. Cancer Res. 48 (1988) 812-815.
    • (1988) Cancer Res. , vol.48 , pp. 812-815
    • Gottardis, M.M.1    Robinson, S.P.2    Satyaswaroop, P.G.3    Jordan, V.C.4
  • 6
    • 0023760993 scopus 로고
    • Development of tamoxifen-stimulated growth of MCF-7 tumors in athymic mice after long-term antiestrogen administration
    • Gottardis M. M. and Jordan V. C., Development of tamoxifen-stimulated growth of MCF-7 tumors in athymic mice after long-term antiestrogen administration. Cancer Res. 48 (1988) 5183-5187.
    • (1988) Cancer Res. , vol.48 , pp. 5183-5187
    • Gottardis, M.M.1    Jordan, V.C.2
  • 9
    • 0028144926 scopus 로고
    • Characterization of tamoxifen stimulated MCF-7 tumor variants grown in athymic mice
    • Wolf D. M. and Jordan V. C., Characterization of tamoxifen stimulated MCF-7 tumor variants grown in athymic mice. Breast Cancer Res. Treat. 31 (1994) 117-127.
    • (1994) Breast Cancer Res. Treat. , vol.31 , pp. 117-127
    • Wolf, D.M.1    Jordan, V.C.2
  • 10
    • 0028093565 scopus 로고
    • The estrogen receptor from a tamoxifen stimulated MCF-7 tumor variant contains a point mutation in the ligand binding domain
    • Wolf D. M. and Jordan V. C., The estrogen receptor from a tamoxifen stimulated MCF-7 tumor variant contains a point mutation in the ligand binding domain. Breast Cancer Res. Treat. 31 (1994) 129-138.
    • (1994) Breast Cancer Res. Treat. , vol.31 , pp. 129-138
    • Wolf, D.M.1    Jordan, V.C.2
  • 11
    • 0029154750 scopus 로고
    • A naturally occurring estrogen receptor mutation results in increased estrogenicity of a tamoxifen analogue
    • Catherino W. H., Wolf D. M. and Jordan V. C., A naturally occurring estrogen receptor mutation results in increased estrogenicity of a tamoxifen analogue. Molec. Endocr. 9 (1995) 1053-1063.
    • (1995) Molec. Endocr. , vol.9 , pp. 1053-1063
    • Catherino, W.H.1    Wolf, D.M.2    Jordan, V.C.3
  • 12
    • 0029017926 scopus 로고
    • Transforming growth factor α: Expression, regulation, and biological activities
    • Lee D. C., Fenton S. E., Berkowitz E. A. and Hissong M. A., Transforming growth factor α: expression, regulation, and biological activities. Pharmacol. Rev. 47 (1995) 51-85.
    • (1995) Pharmacol. Rev. , vol.47 , pp. 51-85
    • Lee, D.C.1    Fenton, S.E.2    Berkowitz, E.A.3    Hissong, M.A.4
  • 13
    • 0027946822 scopus 로고
    • Inhibition of estrogen-induced breast cancer cell proliferation by reduction in autocrine transforming growth factor alpha expression
    • Reddy K. B., Yee D., Hilsenbeck S. G., Coffey R. J. and Osborne C. K., Inhibition of estrogen-induced breast cancer cell proliferation by reduction in autocrine transforming growth factor alpha expression. Cell Growth Differen. 5 (1994) 1275-1282.
    • (1994) Cell Growth Differen. , vol.5 , pp. 1275-1282
    • Reddy, K.B.1    Yee, D.2    Hilsenbeck, S.G.3    Coffey, R.J.4    Osborne, C.K.5
  • 14
    • 0028558331 scopus 로고
    • Transfection of human estrogen receptor (ER) cDNA into ER-negative mammalian cell lines
    • Levenson A. S. and Jordan V. C., Transfection of human estrogen receptor (ER) cDNA into ER-negative mammalian cell lines. J. Steroid Biochem. Molec. Biol 51 (1994) 229-239.
    • (1994) J. Steroid Biochem. Molec. Biol , vol.51 , pp. 229-239
    • Levenson, A.S.1    Jordan, V.C.2
  • 15
    • 0026520381 scopus 로고
    • Growth regulation of estrogen receptor-negative breast cancer cells transfected with complementary DNAs for estrogen receptor
    • Jiang S. Y. and Jordan V. C., Growth regulation of estrogen receptor-negative breast cancer cells transfected with complementary DNAs for estrogen receptor. J. Natl. Cancer Inst. 84 (1992) 580-591.
    • (1992) J. Natl. Cancer Inst. , vol.84 , pp. 580-591
    • Jiang, S.Y.1    Jordan, V.C.2
  • 16
    • 0018850985 scopus 로고
    • A simple, rapid, and sensitive DNA assay procedure
    • LaBarca C. and Paigen K., A simple, rapid, and sensitive DNA assay procedure. Analyt. Biochem. 102 (1980) 344-352.
    • (1980) Analyt. Biochem. , vol.102 , pp. 344-352
    • LaBarca, C.1    Paigen, K.2
  • 17
    • 0028128432 scopus 로고
    • Paradoxical regulation of estrogen-dependent growth factor gene expression in estrogen receptor (ER) negative human breast cancer cells stably expressing ER
    • Jeng M. H., Jiang S. Y. and Jordan V. C., Paradoxical regulation of estrogen-dependent growth factor gene expression in estrogen receptor (ER) negative human breast cancer cells stably expressing ER. Cancer Lett. 82 (1994) 123-128.
    • (1994) Cancer Lett. , vol.82 , pp. 123-128
    • Jeng, M.H.1    Jiang, S.Y.2    Jordan, V.C.3
  • 19
    • 0020694796 scopus 로고
    • Antagonism of estrogen action with a new benzothiophene derived antiestrogen
    • Black L. J., Jones C. D. and Falcone J. F., Antagonism of estrogen action with a new benzothiophene derived antiestrogen. Life Sci. 32 (1993) 1031-1036.
    • (1993) Life Sci. , vol.32 , pp. 1031-1036
    • Black, L.J.1    Jones, C.D.2    Falcone, J.F.3
  • 20
    • 0029074473 scopus 로고
    • Use of pure antiestrogens to elucidate the mode of action of estrogens
    • Wakeling A. E., Use of pure antiestrogens to elucidate the mode of action of estrogens. Biochem. Pharmacol 49 (1995) 1545-1549.
    • (1995) Biochem. Pharmacol , vol.49 , pp. 1545-1549
    • Wakeling, A.E.1
  • 22
    • 0023712331 scopus 로고
    • The hormone-binding domains of the estrogen and glucocorticoid receptors contain an inducible transcription activation function
    • Webster N. J., Green S., Jin J. R. and Chambon P., The hormone-binding domains of the estrogen and glucocorticoid receptors contain an inducible transcription activation function. Cell 54 (1988) 199-207.
    • (1988) Cell , vol.54 , pp. 199-207
    • Webster, N.J.1    Green, S.2    Jin, J.R.3    Chambon, P.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.