Identification of a loop outside the active site cavity of the human immunodeficiency virus proteases which confers inhibitor specificity

Biochemistry

Volumn 36, Issue 17, 1997, Pages 5128-5133

  Towler, Eric M ^a,b   Thompson, Scott K ^a   Tomaszek, Thaddeus ^a   Debouck, Christine ^a  

^a GLAXOSMITHKLINE   (United Kingdom)

^b SAIC FREDERICK INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

PROTEINASE; VIRUS ENZYME;

ARTICLE; BINDING AFFINITY; ENZYME ACTIVE SITE; ENZYME SPECIFICITY; ENZYME STRUCTURE; HUMAN; HUMAN CELL; HUMAN IMMUNODEFICIENCY VIRUS; INHIBITION KINETICS; MOLECULAR GENETICS; PRIORITY JOURNAL; PROTEIN DOMAIN; STRUCTURE ANALYSIS; VIRUS INHIBITION;

AMINO ACID SEQUENCE; HIV PROTEASE; HIV PROTEASE INHIBITORS; HIV-1; HIV-2; HUMANS; MODELS, MOLECULAR; MOLECULAR SEQUENCE DATA; STRUCTURE-ACTIVITY RELATIONSHIP;

HUMAN IMMUNODEFICIENCY VIRUS;

EID: 0031006664     PISSN: 00062960     EISSN: None     Source Type: Journal    
DOI: 10.1021/bi962729j     Document Type: Article

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