Some histamine-related compounds interacting with the benzylamine-oxidizing activity of rat white adipocytes

Journal of Pharmacy and Pharmacology

Volumn 49, Issue 5, 1997, Pages 542-550

  Raimondi, Laura ^a   Conforti, Laura ^a   Banchelli, Grazia ^a   Sgromo, Lucia ^a   Pirisino, Renato ^a  

^a UNIVERSITY OF FLORENCE   (Italy)

Author keywords

[No Author keywords available]

Indexed keywords

AMINE OXIDASE (FLAVIN CONTAINING); AMTHAMINE; BENZYLAMINE; HISTAMINE DERIVATIVE; HISTAMINE RECEPTOR; LIPID; THIOUREA DERIVATIVE;

ADIPOCYTE; ANIMAL CELL; ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; DEGRADATION; ENZYME INHIBITION; LIPID METABOLISM; NONHUMAN; OXIDATION; RAT; WHITE ADIPOSE TISSUE;

EID: 0030996918     PISSN: 00223573     EISSN: None     Source Type: Journal    
DOI: 10.1111/j.2042-7158.1997.tb06839.x     Document Type: Article

References (23)

1. Bertini, V., De Munno, A., Lucchesini, F., Picci, N., Pocci, M., Buffoni, F., Bertocci, B., Banchelli, G., Raimondi, L. (1988) Aymed synthesis of selective inhibitors of copper containing amine oxidases. Pharm. Res. Comm. 20(Suppl): 163-164
2. Buffoni, F. (1966) Histaminase and related amine oxidases. Pharm. Rev. 18: 1163-1199
3. Buffoni, F. (1993) Properties, distribution and physiological role of semicarbazide-sensitive amine oxidases. Curr. Topics Pharmacol. 2: 33-50
4. Buffoni, F., Ignesti, G. (1975) Active-site titration of pig plasma benzylamine oxidase with phenylhydrazine. Biochem. J. 145: 369-372
5. Buffoni, F., Banchelli, G., Ignesti, G., Pirisino, R., Raimondi, L. (1994) The role of semicarbazide-sensitive amine oxidase with a high affinity for benzylamine (Bz.SSAO) in the catabolism of histamine in the mesenteric arterial bed of the rat. Agents Actions 42: 1-6
6. Conforti, L., Raimondi, L., Pirisino, R., Banchelli, G., Ignesti, G., Buffoni, F. (1994) The uptake of histamine by rat white adipose tissue. Br. J. Pharmacol. 111(Suppl): 328P
7. Dixon, M. (1953) The determination of enzyme inhibitor constants. Biochem. J. 55: 170-171
8. 2 receptor, explaining the activity of the different classes of histamine receptor agonists. Mol. Pharmacol. 44: 886-894
9. Leurs, R., Timmerman, H. (1995) Molecular pharmacology aspects of histamine receptors. Pharm. Ter. 66: 413-463
10. Lowry, O. H., Rosebrough, N. J., Lewis-Farr, A., Randall, R. J. (1951) Protein measurement with the Folin phenol reagent. J. Biol. Chem. 193: 265-275
11. Lyles, G. A., Marshall, C. M. S., McDonald, I. A., Bey, P., Palfreyman, M. G. (1987) Inhibition of rat aorta semicarbazide-sensitive amine oxidase by 2-phenyl-3-aloallylamines and related compounds. Biochem. Pharmacol. 36: 2872-2853
12. Matsumoto, T., Furuta, T., Nimura, Y., Suzuki, O. (1982) Increased sensitivity of the fluorimetric method of Snyder and Handley for oxidase assays. Biochem. Pharmacol. 31: 2207-2209
13. Raimondi, L., Pirisino, R., Banchelli, G., Ignesti, G., Conforti, L., Buffoni, F. (1990) Cultured preadipocytes produce a semicarbazide-sensitive amine oxidase (SSAO) activity. J. Neural Transm. 32 (Suppl): 331-336
14. Raimondi, L., Pirisino, R., Ignesti, G., Banchelli, G., Capecchi, S., Buffoni, F. (1991) Semicarbazide-sensitive amine oxidase activity (SSAO) of rat epididymal white adipose tissue. Biochem. Pharmacol. 41: 467-470
15. Raimondi, L., Pirisino, R., Banchelli, G., Ignesti, G., Conforti, L., Romanelli, E., Buffoni, F. (1992) Further studies on semicarbazide-sensitive amine oxidase activities (SSAO) of white adipose tissue. Comp. Biochem. Physiol. 102B: 953-960
16. Raimondi, L., Conforti, L., Banchelli, G., Ignesti, G., Pirisino, R., Buffon, F. (1993) Histamine lipolytic activity and semicarbazide-sensitive amine oxidase (SSAO) of rat white adipose tissue (WAT). Biochem. Pharmacol. 46: 1369-1376
17. 2-related compounds on rat adipocyte lipolysis. Pharmacol. Res. 31(Suppl.): 314
18. Rodbell, M. (1964) Metabolism of isolated fat cells. J. Biol. Chem. 239: 375-380
19. Segel, I. H. (1993) Enzyme Kinetics, John Wiley and Sons, p. 141
20. 2-receptor agonist, dimaprit. Biochem. Pharmacol. 26: 2075-2078
21. Southan, J. G., Szabò, C., Thiemermann, C. (1995) Isothioureas: potent inhibitors of nitric oxide synthases with variable isoform selectivity. Br. J. Pharmacol. 114: 510-516
22. Taylor, K. M., Snyder, S. H. (1972) Histamine methyltransferase: inhibition and potentiation by antihistamines. Mol. Pharmacol. 8: 300-310
23. Wilkinson, G. N. (1961) Statistical estimations in enzyme kinetics. Biochem. J. 80: 328-332