Stereoselective pharmacokinetics of bisoprolol after intravenous and oral administration in beagle dogs

Journal of Pharmaceutical Sciences

Volumn 86, Issue 5, 1997, Pages 560-564

  Horikiri, Yuji ^a   Suzuki, Takehiko ^a   Mizobe, Masakazu ^a  

^a MITSUBISHI TANABE PHARMA CORPORATION   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

BETA 1 ADRENERGIC RECEPTOR BLOCKING AGENT; BISOPROLOL;

ANIMAL EXPERIMENT; ARTICLE; CONTROLLED STUDY; DOG; DRUG BIOAVAILABILITY; DRUG BLOOD LEVEL; DRUG CLEARANCE; DRUG DISTRIBUTION; DRUG PROTEIN BINDING; ENANTIOMER; INTRAVENOUS DRUG ADMINISTRATION; MALE; NONHUMAN; ORAL DRUG ADMINISTRATION; PHARMACOKINETICS; RACEMIC MIXTURE; STEREOCHEMISTRY;

EID: 0030995437     PISSN: 00223549     EISSN: None     Source Type: Journal    
DOI: 10.1021/js960453v     Document Type: Article

References (25)

1. Manalan, A. S.; Besch, H. R.; Watanabe, A. M. Circ. Res. 1982, 49, 326-336.
2. Schliep, H.-J.; Harting, J. J. Cardiovasc. Pharmacol. 1984, 6, 1156-1160.
3. Bühring, K. U.; Sailer, H.; Faro, H.-P.; Leopold, G.; Pabst, J.; Garbe, A. J. Cardiovasc. Pharmacol. 1986, 8, S21-S28.
4. Leopold, G. J. Cardiovasc. Pharmacol. 1986, 8, S16-S20.
5. Kirch, W.; Rose, I.; Demers, H. G.; Leopold, G.; Pabst J.; Ohnhaus, E. E. Clin. Pharmacokinet. 1987, 13, 110-117.
6. Haeusler, G.; Schliep, H.-J.; Schelling, P.; Becker, K. H.; Klockow, M.; Minck, K. O.; Enenkel, H. J.; Schulze, E.; Bergmann, R.; Schmitges, C.-J.; Seyfried, C.; Harting, J. J. Cardiovasc. Pharmacol. 1986, 8, S2-S15.
7. Drayer, D. E. Clin. Pharmacol. Ther. 1986, 40, 125-133.
8. Ariëns, E. J.; Wuis, E. W. Clin Pharmacol. Ther. 1987, 42, 361-363.
9. Jamali, F.; Mehvar, R.; Pasutto, F. M. J. Pharm. Sci. 1989, 78, 695-715.
10. Lee, E. J. D.; Williams, K. M. Clin. Pharmacokinet. 1990, 18, 339-345.
11. Suzuki, T.; Horikiri, Y.; Mizobe, M.; Noda, K. J. Chromatogr. Biomed. Appl. 1993, 619, 267-273.
12. Horikiri, Y.; Suzuki, T.; Mizobe, M; Kobayashi, M; Noda, K. Biol. Pharm. Bull., in preparation.
13. Silber, B.; Holford, N. H. G.; Riegelman, S. J. Pharm. Sci. 1982, 71, 699-703.
14. Lennard, M. S.; Tucker, G. T.; Silas, J. H.; Freestone, S.; Ramsay, L. E.; Woods, H. F. Clin. Pharmacol. Ther. 1983, 34, 732-737.
15. Francis, R. J.; East, P. B.; Larmann, J. Eur. J. Clin. Pharmacol. 1982, 23, 529-533.
16. Dutta, A.; Lane, R.; Begg, E.; Robson, R.; Sia, L.; Dukart, G.; Desjardins, R.; Yacobi, A. J. Clin. Pharmacol. 1994, 34, 829-836.
17. Vagelgesang, B.; Echizen, H.; Schmidt, E.; Eichlbaum, M. Br. J. Clin. Pharmacol. 1984, 18, 733-740.
18. Lee, E. J. D.; Williams, K.; Day, R.; Graham, G.; Champion, D. Br. J. Clin. Pharmacol. 1985, 19, 669-674.
19. Williams, K.; Lee, E. Drugs 1985, 30, 333-354.
20. Carr, R. A.; Pasutto, F. M.; Foster, R. T. Biopharm. Drug Dispos. 1994, 15, 109-120.
21. Masubuchi, Y.; Yamamoto, L. A.; Uesaka, M.; Fujita, S.; Narimatsu, S.; Suzuki, T. Biochem. Pharmacol. 1993. 46, 1759-1765.
22. Kushiya, M. M.; Okada, S.; Kimura, T.; Hasegawa, R. J. Pharm. Pharmacol. 1993, 45, 225-228.
23. Kimura, K.; Mizuno, Y.; Sugihara, K.; Ohbe, Y. Xenobiotic Metabolism and Disposition; Kato, R.; Estabrook, R. W.; Cayen M. N., Eds.; Taylor and Francis: London, 1989; pp 185-192.
24. Hsyu, P. H.; Giacomini, K. H. J. Clin. Invest. 1985, 76, 1720-1726.
25. Yamada, Y.; Nakahara, M.; Naito, K.; Kohno, M.; Otsuka, M.; Takaichi, O. Xenobiot. Metab. Dispos. 1989, 4, 149-164.