메뉴 건너뛰기




Volumn 53, Issue 5, 1997, Pages 671-676

Pseudophrynaminol: A potent noncompetitive blocker of nicotinic receptor-channels

Author keywords

acetylcholinesterase; nicotinic receptors; noncompetitive blockers; physostigmine; pseudophrynamines

Indexed keywords

NICOTINIC RECEPTOR; NICOTINIC RECEPTOR BLOCKING AGENT; PSEUDOPHRYNAMINOL; UNCLASSIFIED DRUG;

EID: 0030991757     PISSN: 00062952     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0006-2952(96)00878-7     Document Type: Article
Times cited : (16)

References (26)
  • 1
    • 0001588616 scopus 로고
    • Pseudophrynamine a: An unusual prenyl pyrrolo[2,3-b]indole ester from an Australian frog, Pseudophryne coriacea (Myobatrachidae)
    • Spande TF, Edwards MW, Pannell LK, Daly JW, Erspamer V and Melchiorri P, Pseudophrynamine A: An unusual prenyl pyrrolo[2,3-b]indole ester from an Australian frog, Pseudophryne coriacea (Myobatrachidae). J Org Chem 53: 1222-1226, 1988.
    • (1988) J Org Chem , vol.53 , pp. 1222-1226
    • Spande, T.F.1    Edwards, M.W.2    Pannell, L.K.3    Daly, J.W.4    Erspamer, V.5    Melchiorri, P.6
  • 2
    • 0025314423 scopus 로고
    • Alkaloids from Australian frogs (Myobatrachidae): Pseudophrynamines and pumiliotoxins
    • Daly JW, Garraffo HM, Pannell LK and Spande TF, Alkaloids from Australian frogs (Myobatrachidae): Pseudophrynamines and pumiliotoxins. J Nat Prod 53: 407-421, 1990.
    • (1990) J Nat Prod , vol.53 , pp. 407-421
    • Daly, J.W.1    Garraffo, H.M.2    Pannell, L.K.3    Spande, T.F.4
  • 3
    • 0000249736 scopus 로고
    • Anticholinesterase agents
    • (Eds. Gilman AG, Goodman LS, Rall TW and Murad F), Macmillan Publishing Co., New York
    • Taylor P, Anticholinesterase agents. In: The Pharmacological Basis of Therapeutics (Eds. Gilman AG, Goodman LS, Rall TW and Murad F), 110-129. Macmillan Publishing Co., New York, 1985.
    • (1985) The Pharmacological Basis of Therapeutics , pp. 110-129
    • Taylor, P.1
  • 4
    • 0022346587 scopus 로고
    • The reversible cholinesterase inhibitor physostigmine has channel-blocking and agonist effects on the acetylcholine receptor-ion channel complex
    • Shaw KP, Aracava Y, Akaike A, Daly JW, Rickett DL and Albuquerque EX, The reversible cholinesterase inhibitor physostigmine has channel-blocking and agonist effects on the acetylcholine receptor-ion channel complex. Mol Pharmacol 28: 527-538, 1985.
    • (1985) Mol Pharmacol , vol.28 , pp. 527-538
    • Shaw, K.P.1    Aracava, Y.2    Akaike, A.3    Daly, J.W.4    Rickett, D.L.5    Albuquerque, E.X.6
  • 5
    • 0027360360 scopus 로고
    • Physostigmine block of ion channels activated by acetylcholine in BC3H1 cells
    • Wachtel RE, Physostigmine block of ion channels activated by acetylcholine in BC3H1 cells. Mol Pharmacol 44: 1051-1055, 1993.
    • (1993) Mol Pharmacol , vol.44 , pp. 1051-1055
    • Wachtel, R.E.1
  • 6
    • 0001744929 scopus 로고
    • Potential anticancer agents. XXXVII. Monofunctional aziridines related to tetramin
    • Reist EJ, Junga IG and Baker BR, Potential anticancer agents. XXXVII. Monofunctional aziridines related to tetramin. J Org Chem 25: 1673-1674, 1960.
    • (1960) J Org Chem , vol.25 , pp. 1673-1674
    • Reist, E.J.1    Junga, I.G.2    Baker, B.R.3
  • 7
    • 0025785666 scopus 로고
    • Nicotinic receptor-elicited sodium-flux in rat pheochromocytoma PC12 cells: Effects of agonists, antagonists and noncompetitive blockers
    • Daly JW, Nishizawa Y, Edwards MW, Waters JA and Aronstam RS, Nicotinic receptor-elicited sodium-flux in rat pheochromocytoma PC12 cells: Effects of agonists, antagonists and noncompetitive blockers. Neurochem Res 16: 489-500, 1991.
    • (1991) Neurochem Res , vol.16 , pp. 489-500
    • Daly, J.W.1    Nishizawa, Y.2    Edwards, M.W.3    Waters, J.A.4    Aronstam, R.S.5
  • 8
    • 0023165023 scopus 로고
    • 3H](-)-nicotine label the same recognition site in rat brain
    • 3H](-)-nicotine label the same recognition site in rat brain. Mol Pharmacol 31: 169-174, 1986.
    • (1986) Mol Pharmacol , vol.31 , pp. 169-174
    • Martino-Garrows, A.M.1    Kellar, K.J.2
  • 9
    • 0023029997 scopus 로고
    • Nicotine binding sites in rat and mouse brain: Comparison of acetylcholine, nicotine and α-bungarotoxin
    • Marks MJ, Stitzel JA, Romm E, Wehner JM and Collins AC, Nicotine binding sites in rat and mouse brain: Comparison of acetylcholine, nicotine and α-bungarotoxin. Mol Pharmacol 30: 427-436, 1986.
    • (1986) Mol Pharmacol , vol.30 , pp. 427-436
    • Marks, M.J.1    Stitzel, J.A.2    Romm, E.3    Wehner, J.M.4    Collins, A.C.5
  • 10
    • 0022260733 scopus 로고
    • Biochemical characterization of a filtered synaptoneurosome preparation from guinea pig cerebral cortex: Cyclic adenosine 3′:5′-monophosphate-generating systems, receptors, and enzymes
    • Hollingsworth EB, McNeal ET, Burton JL, Williams RJ, Daly JW and Creveling CR, Biochemical characterization of a filtered synaptoneurosome preparation from guinea pig cerebral cortex: Cyclic adenosine 3′:5′-monophosphate-generating systems, receptors, and enzymes. J Neurosci 5: 2240-2253, 1985.
    • (1985) J Neurosci , vol.5 , pp. 2240-2253
    • Hollingsworth, E.B.1    McNeal, E.T.2    Burton, J.L.3    Williams, R.J.4    Daly, J.W.5    Creveling, C.R.6
  • 11
    • 0023470574 scopus 로고
    • Stimulation of phosphoinositide breakdown in brain synaptoneurosomes by agents that activate sodium influx: Antagonism by tetrodotoxin, saxitoxin and cadmium
    • Gusovsky F, McNeal ET and Daly JW, Stimulation of phosphoinositide breakdown in brain synaptoneurosomes by agents that activate sodium influx: Antagonism by tetrodotoxin, saxitoxin and cadmium. Mol Pharmacol 32: 479-487, 1987.
    • (1987) Mol Pharmacol , vol.32 , pp. 479-487
    • Gusovsky, F.1    McNeal, E.T.2    Daly, J.W.3
  • 13
    • 0024500536 scopus 로고
    • Comparative inhibitory effects of various physostigmine analogs against acetyl- and butyrylcholinesterase
    • Atack JR, Yu QS, Soncrant TT, Brossi A and Rapoport S, Comparative inhibitory effects of various physostigmine analogs against acetyl- and butyrylcholinesterase. J Pharmacol Exp Ther 249: 194-202, 1989.
    • (1989) J Pharmacol Exp Ther , vol.249 , pp. 194-202
    • Atack, J.R.1    Yu, Q.S.2    Soncrant, T.T.3    Brossi, A.4    Rapoport, S.5
  • 14
    • 0342573730 scopus 로고
    • The anatomy of a receptor
    • Karlin A, The anatomy of a receptor. Neurosci Commen 1: 111-123, 1983.
    • (1983) Neurosci Commen , vol.1 , pp. 111-123
    • Karlin, A.1
  • 16
    • 0020068128 scopus 로고
    • Actions of the histrionicotoxins at the ion channel of the nicotinic acetyl-choline receptor and at the voltage-sensitive channels of muscle membranes
    • Spivak CE, Maleque MA, Oliveira AC, Masukawa LM, Tokuyama T, Daly JW and Albuquerque EX, Actions of the histrionicotoxins at the ion channel of the nicotinic acetyl-choline receptor and at the voltage-sensitive channels of muscle membranes. Mol Pharmacol 21: 351-361, 1982.
    • (1982) Mol Pharmacol , vol.21 , pp. 351-361
    • Spivak, C.E.1    Maleque, M.A.2    Oliveira, A.C.3    Masukawa, L.M.4    Tokuyama, T.5    Daly, J.W.6    Albuquerque, E.X.7
  • 17
    • 0022551675 scopus 로고
    • Interaction of gephyrotoxin and indolizidine alkaloids with the nicotinic acetylcholine receptor-ion channel complex of Torpedo electroplax
    • Aronstam RS, Daly JW, Spande TF, Narayanan TK and Albuquerque EX, Interaction of gephyrotoxin and indolizidine alkaloids with the nicotinic acetylcholine receptor-ion channel complex of Torpedo electroplax. Neurochem Res 11: 1227-1240, 1986.
    • (1986) Neurochem Res , vol.11 , pp. 1227-1240
    • Aronstam, R.S.1    Daly, J.W.2    Spande, T.F.3    Narayanan, T.K.4    Albuquerque, E.X.5
  • 18
    • 0026003195 scopus 로고
    • Decahydroquinoline alkaloids: Noncompetitive blockers for nicotinic acetylcholine receptor-channels in pheochromocytoma cells and Torpedo electroplax
    • Daly JW, Nishizawa Y, Padgett WL, Tokuyama T, McCloskey PJ, Waykole L, Schultz AG and Aronstam RS, Decahydroquinoline alkaloids: Noncompetitive blockers for nicotinic acetylcholine receptor-channels in pheochromocytoma cells and Torpedo electroplax. Neurochem Res 16: 1207-1212, 1991.
    • (1991) Neurochem Res , vol.16 , pp. 1207-1212
    • Daly, J.W.1    Nishizawa, Y.2    Padgett, W.L.3    Tokuyama, T.4    McCloskey, P.J.5    Waykole, L.6    Schultz, A.G.7    Aronstam, R.S.8
  • 21
    • 0025364976 scopus 로고
    • Total synthesis of (±)-pseudophrynaminol
    • Mitchell MO and Le Quesne PW, Total synthesis of (±)-pseudophrynaminol. Tetrahedron Lett 31: 2681-2684, 1990.
    • (1990) Tetrahedron Lett , vol.31 , pp. 2681-2684
    • Mitchell, M.O.1    Le Quesne, P.W.2
  • 24
    • 0022452310 scopus 로고
    • Inhibition of acetylcholinesterase from electric eel by (-) and (+)-physostigmine and related compounds
    • Brossi A, Schonenberger B, Clark OE and Ray R, Inhibition of acetylcholinesterase from electric eel by (-) and (+)-physostigmine and related compounds. FEBS Lett 201: 190-192, 1986.
    • (1986) FEBS Lett , vol.201 , pp. 190-192
    • Brossi, A.1    Schonenberger, B.2    Clark, O.E.3    Ray, R.4
  • 25
    • 0016246242 scopus 로고
    • Effects of local anesthetics and calcium on the interaction of cholinergic ligands with the nicotinic receptor protein from Torpedo marmorata
    • Cohen JB, Weber M and Changeux J-P, Effects of local anesthetics and calcium on the interaction of cholinergic ligands with the nicotinic receptor protein from Torpedo marmorata. Mol Pharmacol 10: 904-932, 1974.
    • (1974) Mol Pharmacol , vol.10 , pp. 904-932
    • Cohen, J.B.1    Weber, M.2    Changeux, J.-P.3
  • 26
    • 0025344828 scopus 로고
    • Effect of noncompetitive nicotinic receptor blockers on catecholamine release from cultured adrenal chromaffin cells
    • McKay DB and Trent-Sanchez P, Effect of noncompetitive nicotinic receptor blockers on catecholamine release from cultured adrenal chromaffin cells. Pharmacology 40: 224-230, 1990.
    • (1990) Pharmacology , vol.40 , pp. 224-230
    • McKay, D.B.1    Trent-Sanchez, P.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.