N-substituted phenyltropanes as in vivo binding ligands for rapid imaging studies of the dopamine transporter

Synapse

Volumn 25, Issue 4, 1997, Pages 345-349

  Scheffel, Ursula ^a   Lever, John R ^a   Abraham, Philip ^b   Parham, Karol R ^b   Mathews, William B ^a   Kopajtic, Theresa ^c   Carroll, F Ivy ^b   Kuhar, Michael J ^d  

^a DEPARTMENT OF PATHOLOGY   (United States)

^b RTI INTERNATIONAL   (United States)

^c NATIONAL INSTITUTE ON DRUG ABUSE   (United States)

^d EMORY UNIVERSITY   (United States)

Author keywords

cocaine; dopamine; imaging

Indexed keywords

3BETA (4 IODOPHENYL) 2BETA TROPANECARBOXYLIC ACID ISOPROPYL ESTER; 3BETA (4 IODOPHENYL) 2BETA TROPANECARBOXYLIC ACID METHYL ESTER; DESIPRAMINE; DOPAMINE TRANSPORTER; PAROXETINE; RTI 310; RTI 311; RTI 312; RTI 313; RTI 98; TROPANE DERIVATIVE; UNCLASSIFIED DRUG; VANOXERINE;

ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; CEREBELLUM; CONTROLLED STUDY; CORPUS STRIATUM; DOPAMINERGIC NERVE CELL; DRUG COMPETITION; INTRAVENOUS DRUG ADMINISTRATION; ISOTOPE LABELING; LIGAND BINDING; MALE; MOUSE; NONHUMAN; PRIORITY JOURNAL; PROTEIN LOCALIZATION; RADIOISOTOPE DISTRIBUTION; TISSUE DISTRIBUTION;

ANALYSIS OF VARIANCE; ANIMALS; BINDING, COMPETITIVE; BRAIN; CARRIER PROTEINS; CEREBELLUM; COCAINE; CORPUS STRIATUM; DESIPRAMINE; DOPAMINE PLASMA MEMBRANE TRANSPORT PROTEINS; IODINE RADIOISOTOPES; KINETICS; LIGANDS; MALE; MEMBRANE GLYCOPROTEINS; MEMBRANE TRANSPORT PROTEINS; MICE; NERVE TISSUE PROTEINS; NOREPINEPHRINE PLASMA MEMBRANE TRANSPORT PROTEINS; PAROXETINE; RADIOLIGAND ASSAY; RATS; STRUCTURE-ACTIVITY RELATIONSHIP; SYMPORTERS;

EID: 0030989552     PISSN: 08874476     EISSN: None     Source Type: Journal    
DOI: 10.1002/(SICI)1098-2396(199704)25:4<345::AID-SYN5>3.0.CO;2-A     Document Type: Article

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