Methyl 2H-azirine-3-carboxylates as dienophiles: Synthesis of methyl 1-azabicyclo[4.1.0]hept-3-ene-6-carboxylates

Synthesis

Volumn , Issue 3, 1997, Pages 271-272

  Bhullar, Pamila ^a   Gilchrist, Thomas L ^b   Maddocks, Peter ^a  

^a GLAXOSMITHKLINE   (United Kingdom)

^b UNIVERSITY OF LIVERPOOL   (United Kingdom)

Author keywords

2H azirines; Diels Alder reaction; imines

Indexed keywords

1 AZABICYCLO[4.1.0]HEPT 3 ENE DERIVATIVE; BICYCLO COMPOUND; UNCLASSIFIED DRUG;

ARTICLE; DRUG SYNTHESIS; IN VITRO STUDY; INFRARED SPECTROPHOTOMETRY; NUCLEAR MAGNETIC RESONANCE; REACTION ANALYSIS;

EID: 0030983556     PISSN: 00397881     EISSN: None     Source Type: Journal    
DOI: 10.1055/s-1997-1192     Document Type: Article

References (8)

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3. Anderson, D. J.; Hassner A. Synthesis 1975, 483. Boger, D. L.; Weinreb, S. N. Hetero Diels Alder Methodology in Organic Synthesis; Academic: San Diego, 1987; p 57.
4. Hemetsberger, H.; Knittel, D. Monatsh. Chem. 1972, 103, 205.
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8. L'abbe, G.; Van Stappen, P.; Toppet, S.; Germain, G.; Scheefer, G. Bull. Soc. Chim. Belg. 1983, 92, 193. Law, K. W.; Lai, T. F.; Sammes, M. P.; Katritzky, A. R.; Mak, T. C. W. J. Chem. Soc., Perkin Trans. 1 1984, 111.