Synthesis of a radiolabelled retinoid X receptor (RXR) specific ligand

Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 39, Issue 6, 1997, Pages 501-507

  Held, Pierre ^a   Heck, Marie Pierre ^b   Iyer, Jaya ^c   Gronemeyer, Hinrich ^c   Lebeau, Luc ^a   Mioskowski, Charles ^a,b  

^a UNIVERSITÉ DE STRASBOURG   (France)

^b CEA SACLAY   (France)

^c INSTITUT DE GÉNÉTIQUE ET DE BIOLOGIE MOLÉCULAIRE ET CELLULAIRE   (France)

Author keywords

Retinoid; SR11237; Synthesis; Tritium

Indexed keywords

BENZOIC ACID; CHELATION; LIGANDS;

% REDUCTIONS; DIHALIDES; RETINOID X RECEPTOR; RETINOIDS; SR11237; TETRAMETHYL;

TRITIUM;

4 [2 (5,6,7,8 TETRAHYDRO 5,5,8,8 TETRAMETHYL 2 NAPHTHYL) 1,3 DIOXOLAN 2 YL]BENZOIC ACID; RETINOID; RETINOID X RECEPTOR; TRITIUM;

ARTICLE; DRUG SYNTHESIS; IN VITRO STUDY; ISOTOPE LABELING; MASS SPECTROMETRY; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; RADIOCHEMISTRY; REACTION ANALYSIS; THIN LAYER CHROMATOGRAPHY;

TRITIUM;

EID: 0030981559     PISSN: 03624803     EISSN: None     Source Type: Journal    
DOI: 10.1002/(SICI)1099-1344(199706)39:6<501::AID-JLCR995>3.0.CO;2-S     Document Type: Article

References (11)

1. Leid, M.; Kastner, P.; Chambon, P. - TIBS 427-433 (1992).
2. Futoryan, T.; Gilchrest, B.A. - Nutr. Rev. 52: 299-310 (1994).
3. Pemrick, S.M.; Lucas, D.A.; Grippo, J.F. - Leukemia 8: 1797-1806 (1994).
4. Newcomer, M.E. - FASEB J. 9: 229-239 (1995).
5. Kastner, P.; Mark, M.; Chambon, P. - Cell 83: 859-869 (1995).
6. Chen, J.Y.; Clifford, J.; Zusi, C.; Starrett, J.; Tortolani, D.; Ostrowski, J.; Reczek, P.R.; Chambon, P.; Gronemeyer, H. - Nature 382: 819-822 (1996).
7. Chambon, P. - FASEB J. 10: 940-954 (1996).
8. Lehmann, J.; Jong, L.; Fanjul, A.; Cameron, J.F.; Lu, X.P.; Haefner, P.; Dawson, M.I.; Pfahl, M. - Science 258: 1944-1946 (1992).
9. Dawson, M.I.; Jong, L.; Hobbs, P.D.; Cameron, J.F.; Chao, W.R.; Pfahl, M.; Lee, M.O.; Shroot, B.; Pfahl, M. - J. Med. Chem. 38: 3368-3383 (1995).
10. Kageshika, H.; Kawachi, E.; Hashimoto, Y.; Himi, T.; Shudo, K. - J. Med. Chem. 31: 2182-2192 (1988).
11. Chan, T.H.; Brook, M.A.; Chaly, T. - Synthesis 203-205 (1983).