Transdermal iontophoresis of sodium nonivamide acetate. III. Combined effect of pretreatment by penetration enhancers

International Journal of Pharmaceutics

Volumn 149, Issue 2, 1997, Pages 183-193

  Fang, Jia You ^a,c   Fang, Chia Lang ^b   Huang, Yaw Bin ^a   Tsai, Yi Hung ^a  

^a KAOHSIUNG MEDICAL UNIVERSITY   (Taiwan)

^b TAIPEI MEDICAL UNIVERSITY   (Taiwan)

^c CHIA NAN UNIVERSITY OF PHARMACY AND SCIENCE   (Taiwan)

Author keywords

Iontophoresis; Penetration enhancer; Sodium nonivamide acetate; Transdermal absorption

Indexed keywords

BENZALKONIUM CHLORIDE; CETYLPYRIDINIUM SALT; DODECYL SULFATE SODIUM; MYRISTIC ACID ISOPROPYL ESTER; NONIVAMIDE; PENETRATION ENHANCING AGENT;

ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; DIFFUSION; HISTOLOGY; IONTOPHORESIS; MALE; NONHUMAN; PASSIVE TRANSPORT; PRIORITY JOURNAL; RAT; SKIN ABSORPTION; SKIN PENETRATION;

EID: 0030976074     PISSN: 03785173     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0378-5173(97)04870-9     Document Type: Article

References (33)

1. Chen, I.J., Yang, J.M., Yeh, J.L., Wu, B.N., Lo, Y.C. and Chen, S.J., Hypotensive and antinociceptive effects of ether-linked and relatively non-pungent analogues of N-nonanoyl vanillylamide. Eur. J. Med. Chem., 27 (1992) 187-192.
2. Chien, Y.W., Siddiqui, O., Shi, W.M., Lelawongs, P. and Liu, J.C., Direct current iontophoretic transdermal delivery of peptide and protein drugs. J. Pharm. Sci., 78 (1989) 376-383.
3. Clancy, M.J., Corish, J. and Corrigan, O.I., A comparison of the effects of electrical current and penetration enhancers on the properties of human skin using spectroscopic (FTIR) and calorimetric (DSC) methods. Int. J. Pharm., 105 (1994) 47-56.
4. Cooper, E.R., Increased skin permeability for lipophilic molecules. J. Pharm. Sci., 73 (1984) 1153-1156.
5. Dempski, R.E., De Marco, J.D. and Markus, A.D., An in vitro study of the relative moisture occlusive properties of several topical vehicles and saran wrap. J. Invest. Dermatol., 44 (1965) 361-363.
6. Fang, J.Y., Wu, P.C., Huang, Y.B. and Tsai, Y.H., In vitro permeation study of capsaicin and its synthetic derivatives from ointment bases using various skin types. Int. J. Pharm., 126 (1995) 119-128.
7. Fang, J.Y., Wu, P.C., Huang, Y.B. and Tsai, Y.H., Percutaneous absorption of capsaicin, nonivamide and sodium nonivamide acetate from gel and ointment bases: in vitro formulation evaluations in pigs and in vivo bioengineering methods in humans. Int. J. Pharm., 130 (1996a) 121-135.
8. Fang, J.Y., Wu, P.C., Huang, Y.B. and Tsai, Y.H., In vivo percutaneous absorption of capsaicin, nonivamide and sodium nonivamide acetate from ointment bases: skin erythema test and non-invasive surface recovery technique in humans. Int. J. Pharm., 131 (1996b) 143-151.
9. Fang, J.Y., Tsai, M.J., Wu, P.C., Huang, Y.B. and Tsai, Y.H., Percutaneous absorption and skin erythema quantification of capsaicin and its synthetic derivatives from gels incorpoated with benzalkonium chloride by using non-invasive bioengineering methods. Drug Dev. Res., (1996c) accepted for publication.
10. Fang, J.Y., Huang, Y.B., Wu, P.C. and Tsai, Y.H., Transdermal iontophoresis of sodium nonivamide acetate. I. Consideration of electrical and chemical factors. Int. J. Pharm., 143 (1996d) 47-58.
11. Fang, J.Y., Huang, Y.B., Wu, P.C. and Tsai, Y.H., Transdermal iontophoresis of sodium nonivamide acetate. II. Optimization and evaluation on solutions and gels. Int. J. Pharm., 145 (1996e) 175-186.
12. Gay, C.L., Green, P.G., Guy, R.H. and Francoeur, M.L., Iontophoretic delivery of piroxicam across the skin in vitro. J. Control. Release, 22 (1992) 57-68.
13. Grimnes, S., Pathways of ionic flow through human skin in vivo. Acta Derm. Venereal. (Stockholm), 64 (1984) 93-98.
14. Hosoya, K.I., Shudo, N., Sugibayashi, K. and Morimoto, Y., Effect of azone on the percutaneous absorption of 5-flurouracil from gels in hairless rats. Chem. Pharm. Bull., 35 (1987) 726-733.
15. Idson, B., Percutaneous absorption enhancers. Drug Cosmet. Ind., July (1985) 30-33.
16. Illel, B., Schaefer, H., Wepierre, J. and Doucet, O., Follicles play an important role in percutaneous absorption. J. Pharm. Sci., 80 (1991) 424-427.
17. Inagi, T., Marumatsu, T., Nagai, H and Terada, H., Influence of vehicle composition on the penetration of indomethacin through guinea-pig skin. Chem. Pharm. Bull., 29 (1981) 1708-1714.
18. Kasting, G.B. and Bowman, L.A., DC electrical properties of frozen, excised human skin. Pharm. Res., 1 (1990) 134-143.
19. Kushla, G.P. and Zatz, J.L., Correlation of water and lidocaine flux enhancement by cationic surfactants in vitro. J. Pharm. Sci., 80 (1991) 1079-1083.
20. Lashmar, U.T. and Manger, J., Investigation into the potential for iontophoresis facilitated transdermal delivery of acyclovir. Int. J. Pharm., 111 (1994) 73-82.
21. Miyazaki, S., Tobiyama, T., Takada, M. and Attwood, D., Percutaneous absorption of indomethacin from pluronic F127 gels in rats. J. Pharm. Pharmacol., 47 (1995) 455-457.
22. Quan, D., Takayama, K., Mitsuzono, T., Isowa, K. and Nagai, T., Influence of novel percutaneous absorption enhancers, cyclohexanone and piperidone derivatives on histopathology of rat skin. Int. J. Pharm., 68 (1991) 239-253.
23. Rantuccio, F., Scardigno, A., Conti, A., Sinise, D. and Coviello, C., Histological changes in rabbits after application of medicaments and cosmetic bases. Contact Dermatitis, 5 (1979) 392-397.
24. Rao, V.U. and Misra, A.N., Enhancement of iontophoretic permeation of insulin across human cadaver skin. Pharmazie, 49 (1994) 538-539.
25. Sims, S.M., Higuchi, W.I. and Srinivasan, V., Interaction of electric field and electro-osmotic effects in determining iontophoretic enhancement of anions and cations. Int. J. Pharm., 69 (1991)109-121.
26. Singh, P., Anliker, M., Smith, G.A., Zavortink, D. and Maibach, H.I., Transdermal iontophoresis and solute penetration across excised human skin. J. Pharm. Sci., 84 (1995) 1342-1346.
27. Srinivasan, V., Higuchi, W.I., Sims, S.M., Ghanem, A.H. and Behl, C.R., Transdermal iontophoretic drug delivery: mechanistic analysis and application to polypepide delivery. J. Pharm. Sci., 78 (1989) 370-375.
28. Srinivasan, V., Su, M.H., Higuchi, W.I. and Behl, C.R., Iontophoresis of polypeptides: effect of ethanol pretreatment of human skin. J. Pharm. Sci., 79 (1990) 588-591.
29. Tsai, Y.H., Huang, Y.B., Fang, J.Y. and Wu, P.C., Percutaneous absorption of capsaicin and its derivatives. Drug Dev. Ind. Pharm., 20 (1994) 719-730.
30. Tyle, P., Iontophoretic devices for drug delivery. Pharm. Res., 3 (1986) 318-326.
31. Wearley, L. and Chien, Y. W., Enhancement of the in vitro skin permeability of azidothymidine (AZT) via iontophoresis and chemical enhancer. Pharm. Res., 1 (1990) 34-40.
32. Wu, P.C., Fang, J.Y., Huang, Y.B. and Tsai, Y.H., In vitro effect of penetration enhancers on sodium nonivamide acetate in rat skin. Biol. Pharm. Bull., 18 (1995) 1790-1792.
33. Yoshida, N.H. and Roberts, M.S., Solute molecular size and transdermal iontophoresis across excised human skin. J. Control Release, 25 (1993) 177-195.