-
1
-
-
0019427126
-
8-Hydroxy-2-(di-n-propylamino)tetralin, a new centrally acting 5-hydroxytryptamine receptor agonist
-
Arvidsson, L.E., Hacksell, U., Nilsson, J.L.G., Hjorth, S., Carlsson, A., Lindberg, P., Sanchez, D. and Wikström, H. (1981) 8-Hydroxy-2-(di-n-propylamino)tetralin, a new centrally acting 5-hydroxytryptamine receptor agonist. J. Med. Chem. 24, 921-923.
-
(1981)
J. Med. Chem.
, vol.24
, pp. 921-923
-
-
Arvidsson, L.E.1
Hacksell, U.2
Nilsson, J.L.G.3
Hjorth, S.4
Carlsson, A.5
Lindberg, P.6
Sanchez, D.7
Wikström, H.8
-
3
-
-
0015440803
-
Simultaneous measurement of tyrosine and tryptophan hydroxylase activities in brain in vivo using an inhibitor of the aromatic amino acid decarboxylase
-
Carlsson, A., Davis, J.N., Kehr, W., Lindqvist, M. and Atack, C.V. (1972) Simultaneous measurement of tyrosine and tryptophan hydroxylase activities in brain in vivo using an inhibitor of the aromatic amino acid decarboxylase. Naunyn-Schmiedeberg's Arch. Pharmacol. 275, 153-168.
-
(1972)
Naunyn-Schmiedeberg's Arch. Pharmacol.
, vol.275
, pp. 153-168
-
-
Carlsson, A.1
Davis, J.N.2
Kehr, W.3
Lindqvist, M.4
Atack, C.V.5
-
4
-
-
0025767882
-
1A receptors that are negatively coupled to adenylate cyclase
-
1A receptors that are negatively coupled to adenylate cyclase. Mol. Pharmacol. 39, 780-787.
-
(1991)
Mol. Pharmacol.
, vol.39
, pp. 780-787
-
-
Cornfield, L.J.1
Lambert, G.2
Arvidsson, L.E.3
Mellin, C.4
Vallgårda, J.5
Hacksell, U.6
Nelson, D.L.7
-
5
-
-
0028990742
-
1A receptor agonists: Recent developments and controversial issues
-
1A receptor agonists: recent developments and controversial issues. Psychopharmacology 121, 1-26.
-
(1995)
Psychopharmacology
, vol.121
, pp. 1-26
-
-
De Vry, J.1
-
6
-
-
0023819059
-
1A sites in the rat brain. In vitro binding and autoradiographic studies
-
1A sites in the rat brain. In vitro binding and autoradiographic studies. J. Pharmacol. Exp. Ther. 244, 751-759.
-
(1988)
J. Pharmacol. Exp. Ther.
, vol.244
, pp. 751-759
-
-
Gozlan, H.1
Penchant, M.2
Daval, G.3
Verge, D.4
Menard, F.5
Vanhove, A.6
Beaucourt, J.P.7
Hamon, M.8
-
9
-
-
0020367109
-
8-Hydroxy-2-di-n-propylaminotetralin, 8-OHDPAT, a potent and selective simple ergot congener with 5-HT-receptor stimulating activity
-
Hjorth, S., Carlsson, A., Lindberg, P., Sanchez, D., Wikström, H., Arvidsson, L.E., Hacksell, U. and Nilsson, J.L.G. (1982) 8-Hydroxy-2-di-n-propylaminotetralin, 8-OHDPAT, a potent and selective simple ergot congener with 5-HT-receptor stimulating activity. J. Neural Transm. 55, 169-188.
-
(1982)
J. Neural Transm.
, vol.55
, pp. 169-188
-
-
Hjorth, S.1
Carlsson, A.2
Lindberg, P.3
Sanchez, D.4
Wikström, H.5
Arvidsson, L.E.6
Hacksell, U.7
Nilsson, J.L.G.8
-
10
-
-
0021956188
-
Hypothermia in the rat induced by the potent serotoninergic agent 8-OH-DPAT
-
Hjorth, S. (1985) Hypothermia in the rat induced by the potent serotoninergic agent 8-OH-DPAT. J. Neural Transm. 61, 131-135.
-
(1985)
J. Neural Transm.
, vol.61
, pp. 131-135
-
-
Hjorth, S.1
-
11
-
-
0017086367
-
An animal behaviour model for studying central serotonergic synapses
-
Jacobs, B.L. (1976) An animal behaviour model for studying central serotonergic synapses. Life Sci. 19, 777-786.
-
(1976)
Life Sci.
, vol.19
, pp. 777-786
-
-
Jacobs, B.L.1
-
12
-
-
0025234642
-
The long-term effects of 8-hydroxy-2-(di-n-propylamino)tetralin (8-OH-DPAT) on copulatory and exploratory behaviour in male rats
-
Johansson, C.E., Meyerson, B.J. and Höglund, A.U. (1990) The long-term effects of 8-hydroxy-2-(di-n-propylamino)tetralin (8-OH-DPAT) on copulatory and exploratory behaviour in male rats. Eur. J. Pharmacol. 178, 1-9.
-
(1990)
Eur. J. Pharmacol.
, vol.178
, pp. 1-9
-
-
Johansson, C.E.1
Meyerson, B.J.2
Höglund, A.U.3
-
13
-
-
0000861818
-
Improved preparation, chromatographic separation and X-ray crystallographic determination of the absolute configuration of the enantiomers of 8-hydroxy-2-(dipropylamino)tetralin (8-OH DPAT)
-
Karlsson, A., Pettersson, C., Sundell, S., Arvidsson, L.-E. and Hacksell, U. (1988) Improved preparation, chromatographic separation and X-ray crystallographic determination of the absolute configuration of the enantiomers of 8-hydroxy-2-(dipropylamino)tetralin (8-OH DPAT). Acta Chem. Scand. B42, 231-236.
-
(1988)
Acta Chem. Scand.
, vol.B42
, pp. 231-236
-
-
Karlsson, A.1
Pettersson, C.2
Sundell, S.3
Arvidsson, L.-E.4
Hacksell, U.5
-
16
-
-
0023872441
-
Distribution coefficient, a convenient term for the relation of predictable physico-chemical properties to metabolic processes
-
Manners, C.N., Payling, D.W. and Smith, D.A. (1988) Distribution coefficient, a convenient term for the relation of predictable physico-chemical properties to metabolic processes. Xenobiotica 18, 331-350.
-
(1988)
Xenobiotica
, vol.18
, pp. 331-350
-
-
Manners, C.N.1
Payling, D.W.2
Smith, D.A.3
-
17
-
-
0029415119
-
1A agonist 8-hydroxy-2-(N,N-di-n-propylamino)tetralin (8-OH-DPAT) in the rat after intravenous and oral administration
-
1A agonist 8-hydroxy-2-(N,N-di-n-propylamino)tetralin (8-OH-DPAT) in the rat after intravenous and oral administration. Xenobiotica 25, 1371-1380.
-
(1995)
Xenobiotica
, vol.25
, pp. 1371-1380
-
-
Mason, J.P.1
Dring, L.G.2
Caldwell, J.3
-
18
-
-
0023546796
-
Serotonergic neuronal systems: What their anatomic organization tells us about function
-
Molliver, M.E. (1987) Serotonergic neuronal systems: what their anatomic organization tells us about function. J. Clin. Psychopharmacol. 7, 3S-23S.
-
(1987)
J. Clin. Psychopharmacol.
, vol.7
-
-
Molliver, M.E.1
-
19
-
-
0022003468
-
The 5-HT syndrome and the drug discrimination paradigm in rats: Application in behavioral studies on the central 5-HT system
-
Ortmann, R. (1985) The 5-HT syndrome and the drug discrimination paradigm in rats: application in behavioral studies on the central 5-HT system. Pharmacopsychiatry 18, 198-201.
-
(1985)
Pharmacopsychiatry
, vol.18
, pp. 198-201
-
-
Ortmann, R.1
-
20
-
-
0017600519
-
Transport of metabolic substrates through the blood-brain barrier
-
Pardridge, W.M. and Oldendorf, W.H. (1977) Transport of metabolic substrates through the blood-brain barrier. J. Neurochem. 28, 5-12.
-
(1977)
J. Neurochem.
, vol.28
, pp. 5-12
-
-
Pardridge, W.M.1
Oldendorf, W.H.2
-
21
-
-
0021485840
-
Blood-brain barrier transport and brain sequestration of propranolol and lidocaine
-
Pardridge, W.M., Sakiyama, R. and Fierier, G. (1984) Blood-brain barrier transport and brain sequestration of propranolol and lidocaine. Am. J. Physiol. 247, R582-R588.
-
(1984)
Am. J. Physiol.
, vol.247
-
-
Pardridge, W.M.1
Sakiyama, R.2
Fierier, G.3
-
22
-
-
0022346190
-
Quantitative autoradiographic mapping of serotonin receptors in the rat brain. I. Serotonin-1 receptors
-
Pazos, A. and Palacios, J.M. (1985) Quantitative autoradiographic mapping of serotonin receptors in the rat brain. I. Serotonin-1 receptors. Brain Res. 346, 205-230.
-
(1985)
Brain Res.
, vol.346
, pp. 205-230
-
-
Pazos, A.1
Palacios, J.M.2
-
23
-
-
0024462182
-
Determination of brain concentrations of 8-hydroxy-2- (di-n-propylamino)tetralin by liquid chromatography with electrochemical detection
-
Perry, K.W. and Fuller, R.W. (1989) Determination of brain concentrations of 8-hydroxy-2- (di-n-propylamino)tetralin by liquid chromatography with electrochemical detection. Biochem. Pharmacol. 38, 3169-3173.
-
(1989)
Biochem. Pharmacol.
, vol.38
, pp. 3169-3173
-
-
Perry, K.W.1
Fuller, R.W.2
-
24
-
-
0022544893
-
The inhibition of the cage-leaving response: A model for studies of the serotonergic neurotransmission in the rat
-
Renyi, L., Archer, A., Minor, B.G., Tandberg, B., Fredriksson, A. and Ross, S.B. (1986) The inhibition of the cage-leaving response: a model for studies of the serotonergic neurotransmission in the rat. J. Neural Transm. 65, 193-210.
-
(1986)
J. Neural Transm.
, vol.65
, pp. 193-210
-
-
Renyi, L.1
Archer, A.2
Minor, B.G.3
Tandberg, B.4
Fredriksson, A.5
Ross, S.B.6
-
25
-
-
0027437721
-
Orally active central dopamine and serotonin receptor ligands: 5-, 6-, 7-, and 8-[[(trifluoromethyl)sulfonyl]oxy]- 2 -(di-n-propyl-amino)-tetralins and the formation of active metabolites in vivo
-
Sonesson, C., Boije, M., Svensson, K., Ekman, A., Carlsson, A., Romero, A.G., Martin, I.J., Duncan, J.N., King, L.J. and Wikström, H. (1993) Orally active central dopamine and serotonin receptor ligands: 5-, 6-, 7-, and 8-[[(trifluoromethyl)sulfonyl]oxy]- 2 -(di-n-propyl-amino)-tetralins and the formation of active metabolites in vivo. J. Med. Chem. 36, 3409-3416.
-
(1993)
J. Med. Chem.
, vol.36
, pp. 3409-3416
-
-
Sonesson, C.1
Boije, M.2
Svensson, K.3
Ekman, A.4
Carlsson, A.5
Romero, A.G.6
Martin, I.J.7
Duncan, J.N.8
King, L.J.9
Wikström, H.10
-
26
-
-
0021678913
-
The involvement of subtypes of the 5-HT1 receptor and of catecholaminergic systems in the behavioural response to 8-hydroxy-2-(di-n-propylamino)tetralin in the rat
-
Tricklebank, M.D., Forler, C. and Fozard, J.R. (1985) The involvement of subtypes of the 5-HT1 receptor and of catecholaminergic systems in the behavioural response to 8-hydroxy-2-(di-n-propylamino)tetralin in the rat. Eur. J. Pharmacol. 106, 271-282.
-
(1985)
Eur. J. Pharmacol.
, vol.106
, pp. 271-282
-
-
Tricklebank, M.D.1
Forler, C.2
Fozard, J.R.3
-
27
-
-
0023951984
-
Occurrence and pharmacological significance of metabolic ortho-hydroxylation of 5- and 8-hydroxy-2-(di-n-propylamino)tetralin
-
Wikström, H., Elebring, T., Hallnemo, G., Anderson, B., Svensson, K., Carlsson, A. and Rollema, H. (1988) Occurrence and pharmacological significance of metabolic ortho-hydroxylation of 5- and 8-hydroxy-2-(di-n-propylamino)tetralin. J. Med. Chem. 31, 1080-1084.
-
(1988)
J. Med. Chem.
, vol.31
, pp. 1080-1084
-
-
Wikström, H.1
Elebring, T.2
Hallnemo, G.3
Anderson, B.4
Svensson, K.5
Carlsson, A.6
Rollema, H.7
-
29
-
-
0029951557
-
Differential serotonergic and dopaminergic activities of the (R)- and (S)-enantiomers of 2-(di-n-propylamino)tetralin
-
Yu, H., Liu, Y., Malmberg, Å., Mohell, N., Hacksell, U. and Lewander, T. (1996) Differential serotonergic and dopaminergic activities of the (R)- and (S)-enantiomers of 2-(di-n-propylamino)tetralin. Eur. J. Pharmacol. 303, 151-162.
-
(1996)
Eur. J. Pharmacol.
, vol.303
, pp. 151-162
-
-
Yu, H.1
Liu, Y.2
Malmberg, Å.3
Mohell, N.4
Hacksell, U.5
Lewander, T.6
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