Novel cyclic peptide agonist of high potency and selectivity for the type II vasoactive intestinal peptide receptor

Journal of Pharmacology and Experimental Therapeutics

Volumn 281, Issue 2, 1997, Pages 629-633

  Xia, Menghang ^a   Sreedharan, Sunil P ^a   Bolin, David R ^b   Gaufo, Gary O ^a   Goetzl, Edward J ^a  

^a UNIVERSITY OF CALIFORNIA   (United States)

^b HOFFMANN LA ROCHE INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

4 (2 HYDROXYETHYL) 1 PIPERAZINEETHANESULFONIC ACID; 4 (3 BUTOXY 4 METHOXYBENZYL) 2 IMIDAZOLIDINONE; CALCIUM ION; CYCLIC AMP; CYCLOPEPTIDE; FURA 2 ACETOXYMETHYL ESTER; ISOBUTYLMETHYLXANTHINE; RECEPTOR SUBTYPE; RO 25 1392; UNCLASSIFIED DRUG; VASOACTIVE INTESTINAL POLYPEPTIDE DERIVATIVE; VASOACTIVE INTESTINAL POLYPEPTIDE RECEPTOR;

AGONIST; ANIMAL CELL; ARTICLE; CALCIUM CELL LEVEL; CHO CELL; COMPETITIVE INHIBITION; CONTROLLED STUDY; DRUG BIOAVAILABILITY; DRUG POTENCY; DRUG SELECTIVITY; LIGAND BINDING; NONHUMAN; PRIORITY JOURNAL; RECEPTOR DOWN REGULATION; SIGNAL TRANSDUCTION;

ANIMALS; CHO CELLS; CRICETINAE; DOWN-REGULATION; HUMANS; PEPTIDES, CYCLIC; RADIOLIGAND ASSAY; RECEPTORS, VASOACTIVE INTESTINAL PEPTIDE; TRANSFECTION; VASOACTIVE INTESTINAL PEPTIDE;

EID: 0030975009     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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