Benzo[c]quinoliziniums: A new family of inhibitors for protein kinase CKII

Bioorganic and Medicinal Chemistry Letters

Volumn 7, Issue 8, 1997, Pages 961-964

  Mettey, Y ^a   Vierfond, J M ^a   Baudry, M ^a   Cochet, C ^b   Sarrouilhe, D ^a  

^a Faculte de Medicine et de Pharmacie   (France)

^b CEA GRENOBLE   (France)

Author keywords

[No Author keywords available]

Indexed keywords

ISOENZYME; PROTEIN KINASE C; PROTEIN KINASE C INHIBITOR; QUINOLIZINE DERIVATIVE;

ARTICLE; DOSE RESPONSE; DRUG SYNTHESIS; ENZYME INHIBITION; IN VITRO STUDY;

EID: 0030970110     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(97)00127-3     Document Type: Article

References (11)

1. Pinna, L. A. Biochim. Biophys. Acta 1990, 1054, 267.
2. Tuazon, P.T.; Traugh, J.A. Advances in Second Messenger and Phosphoprotein Research; Greengard, P.; Robinson, G.A., Ed. ; Raven Press : New-York, 1991; Vol. 23, pp. 123-164.
3. Friedrich, T.D.; Ingram, V.M. Biochim. Biophys. Acta 1989, 992, 41.
4. Münstermann, U.; Fritz, G.; Seitz, G.; Yiping, L.; Schneider, H.R.; Issinger, O-G. Eur. J. Biochem. 1990, 189, 251.
5. Seldin, D.C.; Leder, P. Science 1995, 267, 894.
6. Vierfond, J-M.; Mettey, Y.; Joubin, R.; Miocque, M. J. Heterocyclic Chem. 1979, 16, 753.
7. Bojanowski, K.; Filhol, O.; Cochet, C.; Chambaz, E.M.; Kragh Larsen, A. J. Biol. Chem. 1993, 268, 22920.
8. Cochet, C ; Feige, J.J.; Pirollet, F.; Keramidas, M.; Chambaz, E.M. Biochem. Pharmacol. 1982, 31, 1357.
9. Wang, Y.; Roach, P.J. Protein Phosphorylation. A practical Approach; Hardie, D.G., Ed.; Oxford University Press: Oxford, New York, Tokyo, 1993, 121-144.
10. Bolla, M.; Rostaing-Puissant, B.R.; Chedin, M.; Souvignet, C.; Marron-Charrière, J.; Colonna, M.; Berland, E.; Chambaz, E. M. Breast Cancer Res. Treat. 1993, 26, 283.
11. Azzi, L.; Meijer, L.; Reed, S.I.; Pidikiti, R.; Tung, H.Y.L. Eur. J. Biochem. 1992, 203, 353.