An aromatic moiety is not essential for pharmacophore binding to sigma binding sites: Synthesis of N-alkylazacycloheptane derivatives as potent sigma ligands

Bioorganic and Medicinal Chemistry Letters

Volumn 7, Issue 17, 1997, Pages 2303-2306

  Yamashita, Akitake ^a   Takahashi, Nobuyuki ^a   Mochizuki, Daisuke ^a   Tsujita, Ryiuchi ^a   Yamada, Shinji ^a   Kawakubo, Hiromu ^a   Suzuki, Yukio ^a   Watanabe, Hideyuki ^a  

^a ASAHI CHEMICAL INDUSTRY CO   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

HALOPERIDOL; HEXAMETHYLENEIMINE DERIVATIVE; N ALLYLNORMETAZOCINE; SIGMA OPIATE RECEPTOR; SIGMA RECEPTOR LIGAND;

ARTICLE; BINDING SITE; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; REACTION ANALYSIS; RECEPTOR AFFINITY;

EID: 0030967893     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(97)00417-4     Document Type: Article

References (9)

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