Design of kallidin-releasing tissue kallikrein inhibitors based on the specificities of the enzyme's binding subsites

Biochemical Journal

Volumn 323, Issue 1, 1997, Pages 167-171

  Portaro, Fernanda C V ^a   Cezari, Maria H S ^a   Juliano, Maria A ^a   Juliano, Luiz ^a   Walmsley, Adrian R ^b   Prado, Eline S ^a  

^a FEDERAL UNIVERSITY OF SÃO PAULO   (Brazil)

^b UNIVERSITY OF SHEFFIELD   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

ANILIDE; ARGININE; BENZOYLARGININE 4 NITROANILIDE; HYDROLASE INHIBITOR; KALLIDIN; KALLIKREIN; PHENYLALANINE;

AMINO ACID SUBSTITUTION; ARTICLE; BINDING SITE; ENZYME BLOOD LEVEL; ENZYME KINETICS; ENZYME SPECIFICITY; HUMAN; NONHUMAN; PRIORITY JOURNAL; RAT;

EID: 0030958118     PISSN: 02646021     EISSN: None     Source Type: Journal    
DOI: 10.1042/bj3230167     Document Type: Article

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