The rational design of TAP inhibitors using peptide substrate modifications and peptidomimetics

European Journal of Immunology

Volumn 27, Issue 4, 1997, Pages 898-904

  Grommé, Monique ^a   Van der Valk, Richard ^a   Sliedregt, Karen ^b   Vernie, Leen ^a   Liskamp, Rob ^b   Hämmerling, Günter ^c   Koopmann, Jens Oliver ^c   Momburg, Frank ^c   Neefjes, Jacques ^a,d  

^a NETHERLANDS CANCER INSTITUTE   (Netherlands)

^b UTRECHT UNIVERSITY   (Netherlands)

^c GERMAN CANCER RESEARCH CENTER DKFZ   (Germany)

^d Department of Radiotherapy   (Netherlands)

Author keywords

Antigen presentation; Inhibitor; Major histocompatibility complex class I molecule; Peptide; Peptidomimetics; TAP

Indexed keywords

MAJOR HISTOCOMPATIBILITY ANTIGEN CLASS 1; PEPTIDE;

ANTIGEN PRESENTATION; ARTICLE; CYTOSOL; ENDOPLASMIC RETICULUM; MAJOR HISTOCOMPATIBILITY COMPLEX; PRIORITY JOURNAL;

AMINO ACID SEQUENCE; ATP-BINDING CASSETTE TRANSPORTERS; BINDING, COMPETITIVE; DRUG DESIGN; MAJOR HISTOCOMPATIBILITY COMPLEX; PEPTIDES; PROTEIN BINDING; STEREOISOMERISM; SUBSTRATE SPECIFICITY;

EID: 0030957403     PISSN: 00142980     EISSN: None     Source Type: Journal    
DOI: 10.1002/eji.1830270415     Document Type: Article

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