Synthesis and analgesic effects of 3-substituted 4,6-diarylpyridazine derivatives of the arylpiperazine class

Bioorganic and Medicinal Chemistry

Volumn 5, Issue 4, 1997, Pages 655-659

  Rohet, Florence ^a   Rubat, Catherine ^a   Coudert, Pascal ^a   Couquelet, Jacques ^a  

^a Laboratoire de Pharmacochimie   (France)

Author keywords

[No Author keywords available]

Indexed keywords

5 HYDROXYTRYPTOPHAN; CARBIDOPA; MORPHINE; NALOXONE; PYRIDAZINE DERIVATIVE;

ANALGESIC ACTIVITY; ANIMAL EXPERIMENT; ANTINOCICEPTION; ARTICLE; CONTROLLED STUDY; DRUG SYNTHESIS; INTRAPERITONEAL DRUG ADMINISTRATION; MALE; MOUSE; NEUROTOXICITY; NONHUMAN; SEDATION; SUBCUTANEOUS DRUG ADMINISTRATION;

ACETAMINOPHEN; ANALGESICS, NON-NARCOTIC; ANALGESICS, OPIOID; ANIMALS; ANTI-INFLAMMATORY AGENTS, NON-STEROIDAL; ASPIRIN; BENZOQUINONES; DIPYRONE; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG DESIGN; DRUG INTERACTIONS; INJECTIONS, INTRAPERITONEAL; MALE; MICE; MORPHINE; MOTOR ACTIVITY; NALOXONE; NARCOTIC ANTAGONISTS; NEUROTOXINS; PAIN; PYRAZOLONES; PYRIDAZINES; RECEPTORS, OPIOID; REFERENCE STANDARDS; SEROTONIN UPTAKE INHIBITORS; STRUCTURE-ACTIVITY RELATIONSHIP; TRAZODONE;

ANIMALIA;

EID: 0030952723     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0968-0896(97)00006-0     Document Type: Article

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