Binding of drugs to monoglyceride-based drug delivery systems

International Journal of Pharmaceutics

Volumn 147, Issue 2, 1997, Pages 135-142

  Chang, Chin Ming ^a   Bodmeier, Roland ^b  

^a UNIVERSITY OF TEXAS AT AUSTIN   (United States)

^b FREIE UNIVERSITÄT BERLIN   (Germany)

Author keywords

Cubic phase; Lipids; Liquid crystalline phase; Monoglycerides; Sustained drug release

Indexed keywords

CHLORPHENIRAMINE MALEATE; DILTIAZEM; GLYCEROL OLEATE; GRISEOFULVIN; MONOACYLGLYCEROL; PHENYLPROPANOLAMINE; PROPRANOLOL; PSEUDOEPHEDRINE; THEOPHYLLINE;

ARTICLE; COMPLEX FORMATION; DISSOLUTION; DRUG BINDING; DRUG DELIVERY SYSTEM; DRUG RELEASE; DRUG SOLUTION; PRIORITY JOURNAL; SOLUBILIZATION; SURFACE TENSION; SUSTAINED RELEASE PREPARATION;

EID: 0030950475     PISSN: 03785173     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0378-5173(96)04805-3     Document Type: Article

References (17)

1. Brokaw, G.Y. and Lyman, W.C., The behavior of distilled monoglycerides in the presence of water. J. Am. Oil Chem. Soc., 35 (1958) 49-53.
2. Bodmeier, R. and Chang, C.M., Solvent-or drug-induced monoglyceride based drug delivery systems transforming in situ into a highly viscous cubic phase. Eur. J. Pharm. Biopharm., 42 (1996) 32S.
3. Caffrey, M., The study of lipid phase transitions by time-resolved X-ray diffraction. Biochemistry, 26 (1987) 6349-6363.
4. Chang, C.M., Application of monoglyceride-based materials as sustained release drug carriers. Ph.D. dissertation, The University of Texas at Austin, May 1995.
5. Chang, C.M. and Bodmeier, R., Monoglyceride-based liquid crystalline injectable drug delivery systems. Pharm. Res., 12 (1995) S-228.
6. Engström, S., Drug delivery from cubic and other lipid-water phases. Lipid Technol, 2 (1990) 42-45.
7. Engström, S. and Engström, L., Phase behaviour of the lidocaine-monoolein-water system. Int. J. Pharm., 79 (1992) 113-122.
8. Engström, S., Lindahl, L., Wallin, R. and Engblom, J., A study of polar lipid drug carrier systems undergoing a thermoreversible lamellar-to-cubic phase transition. Int. J. Pharm., 86 (1992) 137-145.
9. Engström, S., Ljusberg-Wahren, H. and Gustafsson, A., Bioadhesive properties of the monoolein-water system. Pharm. Technol. Europe, (1995) 14-17.
10. Ericsson, B., Eriksson, P.O., Löfroth, J.E. and Engström, S., Cubic phase as delivery system for peptide drugs. In Dunn, R. and Ottenbritte, R.M. (Eds), Polymeric Drugs and Drug Delivery Systems, ACS Symposium Series 469, 1991, pp. 251-265.
11. Hyde, S.T., Andersson, S., Ericsson, B. and Larsson, K., A cubic structure consisting of a lipid bilayer forming an infinite periodic minimum surface of the gyroid type in the glycerol monooleate-water system. Z. Kristallogr., 168 (1984) 213-219.
12. Lutton, E.S., Phase behavior of aqueous systems of monoglycerides. J. Am Oil Chem. Soc., 42 (1965) 1068-1070.
13. Mitchell, D.J. and Ninham, B.W., Micelles, vesicles, and microemulsions, J. Chem Soc., Faraday Trans. 2, 77(4) (1981) 601-629.
14. Müller-Goymann, C.C. and Hamann, H.-J., Sustained release from reverse micellar solutions by phase transformations into lamellar liquid crystals. J. Control. Release, 23 (1993) 165-174.
15. Papantoniou, I. and Müller-Goymann, C.C., Influence of the phase transformation from reverse micellar solution into lamellar liquid crystal on sustained release. Part I. Physicochemical characterization of systems containing either diclofenac acid or diclofenac sodium. Pharm. Pharmacol. Lett., 5(1) (1995) 28-31.
16. Rosevear, F.B. The microscopy of the liquid crystalline neat and middle phases of soaps and synthetic detergents. J. Am. Oil Chem. Soc., 31 (1954) 628-639.
17. Wyatt, D.M. and Dorschel, D., A cubic-phase delivery system composed of glyceryl monooleate and water for sustained release of water-soluble drugs. Pharm. Technol, 16 (1992) 116-130.