7,7-Difluoroprostacyclin derivative, AFP-07, a highly selective and potent agonist for the prostacyclin receptor

Prostaglandins

Volumn 53, Issue 2, 1997, Pages 83-90

  Chang, Chang Sheng ^b   Negishi, Manabu ^b   Nakano, Takashi ^a   Morizawa, Yoshitomi ^a   Matsumura, Yasushi ^a   Ichikawa, Atsushi ^b  

^a ASAHI GLASS CO LTD   (Japan)

^b KYOTO UNIVERSITY   (Japan)

Author keywords

EP1; EP2; EP3; EP4; PGE receptor; prostacyclin receptor

Indexed keywords

7,7 DIFLUOROPROSTACYCLIN DERIVATIVE; AFP 03; AFP 06; AFP 07; CYCLIC AMP; ILOPROST; PROSTACYCLIN DERIVATIVE; PROSTACYCLIN RECEPTOR; PROSTAGLANDIN E2; RECEPTOR SUBTYPE; TRITIUM; UNCLASSIFIED DRUG;

AGONIST; ANIMAL CELL; ARTICLE; CHO CELL; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; DRUG STRUCTURE; NONHUMAN; RECEPTOR AFFINITY;

ANIMALS; BINDING, COMPETITIVE; CHO CELLS; CRICETINAE; CYCLIC AMP; DINOPROSTONE; EPOPROSTENOL; ILOPROST; MICE; RECEPTORS, EPOPROSTENOL; RECEPTORS, PROSTAGLANDIN; RECEPTORS, PROSTAGLANDIN E;

ANIMALIA; CRICETINAE; CRICETULUS GRISEUS; TRITIUM;

EID: 0030948220     PISSN: 00906980     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0090-6980(97)00003-8     Document Type: Article

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