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Volumn 280, Issue 3, 1997, Pages 1201-1209

FK960 [N-(4-acetyl-1-piperazinyl)-p-fluorobenzamide monohydrate], a novel potential antidementia drug, improves visual recognition memory in rhesus monkeys: Comparison with physostigmine

Author keywords

[No Author keywords available]

Indexed keywords

DIZOCILPINE; N (4 ACETYL 1 PIPERAZINYL) 4 FLUOROBENZAMIDE; NEUROTROPIC AGENT; PHYSOSTIGMINE; SCOPOLAMINE; UNCLASSIFIED DRUG;

EID: 0030947805     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article
Times cited : (36)

References (46)
  • 1
    • 0022601116 scopus 로고
    • The effects of physostigmine and scopolamine on recognition memory in monkeys
    • AIGNER, T. G. AND MISHKIN, M.: The effects of physostigmine and scopolamine on recognition memory in monkeys. Behav. Neural. Biol. 45: 81-87, 1986.
    • (1986) Behav. Neural. Biol. , vol.45 , pp. 81-87
    • Aigner, T.G.1    Mishkin, M.2
  • 2
    • 0023248545 scopus 로고
    • Effects of scopolamine and physostigmine on recognition memory in monkeys with ibotenic-acid lesions of the nucleus basalis of Meynert
    • AIGNER, T. G., MITCHELL, S. J., AGGLETON, J. P., DELONG, M. R., STRUBLE, R. G., PRICE, D. L., WENK, G. L. AND MISHKIN, M.: Effects of scopolamine and physostigmine on recognition memory in monkeys with ibotenic-acid lesions of the nucleus basalis of Meynert. Psychopharmacology 92: 292-300, 1987.
    • (1987) Psychopharmacology , vol.92 , pp. 292-300
    • Aigner, T.G.1    Mitchell, S.J.2    Aggleton, J.P.3    Delong, M.R.4    Struble, R.G.5    Price, D.L.6    Wenk, G.L.7    Mishkin, M.8
  • 4
    • 0025165915 scopus 로고
    • Evidence that somatostatin enhances endogenous acetylcholine release in the rat hippocampus
    • ARAUJO, D. M., LAPCHAK, P. A., COLLIER, B. AND QUIRION, R.: Evidence that somatostatin enhances endogenous acetylcholine release in the rat hippocampus. J. Neurochem. 55: 1546-1555, 1990.
    • (1990) J. Neurochem. , vol.55 , pp. 1546-1555
    • Araujo, D.M.1    Lapchak, P.A.2    Collier, B.3    Quirion, R.4
  • 5
    • 0026539328 scopus 로고
    • Competitive and non-competitive NMDA receptor antagonists in spatial learning tasks
    • BISCHOFF, C. AND TIKDTKE, P. I.: Competitive and non-competitive NMDA receptor antagonists in spatial learning tasks. Eur. J. Pharmacol. 213: 269-273, 1992.
    • (1992) Eur. J. Pharmacol. , vol.213 , pp. 269-273
    • Bischoff, C.1    Tikdtke, P.I.2
  • 6
    • 0027476024 scopus 로고
    • A synaptic model of memory: Long-term potentiation in the hippocampus
    • BLISS, T. V. P. AND COLLINGRIDGE, G. L.: A synaptic model of memory: Long-term potentiation in the hippocampus. Nature (Lond.) 361: 31-39, 1993.
    • (1993) Nature (Lond.) , vol.361 , pp. 31-39
    • Bliss, T.V.P.1    Collingridge, G.L.2
  • 7
    • 0020647470 scopus 로고
    • Excitatory amino acids in synaptic transmission in the Schaffer collateral-commissural pathway of the rat hippocampus
    • Lond.
    • COLLINGRIDGE, G. L., KEHL, S. J. AND MCLENNAN, H.: Excitatory amino acids in synaptic transmission in the Schaffer collateral-commissural pathway of the rat hippocampus. J. Physiol. (Lond.) 334: 33-46, 1983.
    • (1983) J. Physiol. , vol.334 , pp. 33-46
    • Collingridge, G.L.1    Kehl, S.J.2    Mclennan, H.3
  • 8
    • 0024829451 scopus 로고
    • Excitatory amino acid receptors in the vertebrate central nervous system
    • COLLINGRIDGE, G. L. AND LESTER, R. A. J.: Excitatory amino acid receptors in the vertebrate central nervous system. Pharmacol. Rev. 40: 143-210, 1989.
    • (1989) Pharmacol. Rev. , vol.40 , pp. 143-210
    • Collingridge, G.L.1    Lester, R.A.J.2
  • 9
    • 0020686674 scopus 로고
    • Alzheimer's disease: A disorder of cholinergic innervation
    • Wash. DC
    • COYLE, J. T., PRICE, D. L. AND DELONG, M. R.: Alzheimer's disease: A disorder of cholinergic innervation. Science (Wash. DC) 219: 1184-1190, 1983.
    • (1983) Science , vol.219 , pp. 1184-1190
    • Coyle, J.T.1    Price, D.L.2    Delong, M.R.3
  • 10
    • 0019256571 scopus 로고
    • Reduced somatostatin-like immunoreactivity in cerebral cortex from cases of Alzheimer disease and Alzheimer senile dementia
    • DAVIES, P., KATZMAN, R. AND TERRY, R. D.: Reduced somatostatin-like immunoreactivity in cerebral cortex from cases of Alzheimer disease and Alzheimer senile dementia. Nature (Lond.) 288: 279-280, 1980.
    • (1980) Nature (Lond.) , vol.288 , pp. 279-280
    • Davies, P.1    Katzman, R.2    Terry, R.D.3
  • 11
    • 0011162190 scopus 로고
    • Selective loss of central cholinergic neurons in Alzheimer's disease
    • DAVIES, P, AND MALONEY, A. J. F.: Selective loss of central cholinergic neurons in Alzheimer's disease. Lancet 2: 1403, 1976.
    • (1976) Lancet , vol.2 , pp. 1403
    • Davies, P.1    Maloney, A.J.F.2
  • 12
    • 0027363742 scopus 로고
    • Role of forebrain cholinergic systems in learning and memory: Relevance to the cognitive deficits of aging and Alzheimer's dementia
    • DUNNETT, S. B. AND FIBIGER, H. C.: Role of forebrain cholinergic systems in learning and memory: Relevance to the cognitive deficits of aging and Alzheimer's dementia. Prog. Brain Res. 98: 413-420, 1993.
    • (1993) Prog. Brain Res. , vol.98 , pp. 413-420
    • Dunnett, S.B.1    Fibiger, H.C.2
  • 13
    • 0022500305 scopus 로고
    • Somatostatin in the central nervous system: Physiology and pathological modifications
    • EPELBAUM, J.: Somatostatin in the central nervous system: Physiology and pathological modifications. Prog. Neurobiol. 27: 63-100, 1986.
    • (1986) Prog. Neurobiol. , vol.27 , pp. 63-100
    • Epelbaum, J.1
  • 15
    • 0025038034 scopus 로고
    • Treatment of Alzheimer's disease with short- and long-term oral THA and lecithin: A double blind study
    • FITTEN, L. J., PERRYMAN, K. M., GROSS, P. L., FINE, H., CUMMINS, J. AND MARSHALL, C.: Treatment of Alzheimer's disease with short-and long-term oral THA and lecithin: A double blind study. Am. J. Psychiatry 147: 239-242, 1990.
    • (1990) Am. J. Psychiatry , vol.147 , pp. 239-242
    • Fitten, L.J.1    Perryman, K.M.2    Gross, P.L.3    Fine, H.4    Cummins, J.5    Marshall, C.6
  • 16
    • 0022635720 scopus 로고
    • Scopolamine effects on memory retention in mice: A model of dementia?
    • FLOOD, J. F. AND CHERKIN, A.: Scopolamine effects on memory retention in mice: A model of dementia? Behav. Neural Biol. 45: 169-184, 1986.
    • (1986) Behav. Neural Biol. , vol.45 , pp. 169-184
    • Flood, J.F.1    Cherkin, A.2
  • 17
    • 0024363934 scopus 로고
    • Excitatory amino acids and Alzheimer's disease
    • GREENAMYRE, J. T. AND YOUNG, A. B.: Excitatory amino acids and Alzheimer's disease. Neurobiol. Aging 10: 593-602, 1989.
    • (1989) Neurobiol. Aging , vol.10 , pp. 593-602
    • Greenamyre, J.T.1    Young, A.B.2
  • 19
    • 0021710551 scopus 로고
    • Immunohistochemical distribution of somatostatin-like immunoreactivity in the central nervous system of the adult rat
    • JOHANSSON, O., HOKFELT, T. AND ELDE, R. P.: Immunohistochemical distribution of somatostatin-like immunoreactivity in the central nervous system of the adult rat. Neuroscience 13: 265-339, 1984.
    • (1984) Neuroscience , vol.13 , pp. 265-339
    • Johansson, O.1    Hokfelt, T.2    Elde, R.P.3
  • 20
    • 0028204233 scopus 로고
    • A screening concept based on a hypothesis led to the development of a putative cognitive enhancer that stimulates penile erection
    • MAEDA, N., MATSUOKA, N., YAMAZAKI, M., ARAKAWA, H., OHKUBO, Y. AND YAMAGUCHI, I.: A screening concept based on a hypothesis led to the development of a putative cognitive enhancer that stimulates penile erection. Jpn. J. Pharmacol. 64: 147-153, 1994.
    • (1994) Jpn. J. Pharmacol. , vol.64 , pp. 147-153
    • Maeda, N.1    Matsuoka, N.2    Yamazaki, M.3    Arakawa, H.4    Ohkubo, Y.5    Yamaguchi, I.6
  • 21
    • 0030436895 scopus 로고    scopus 로고
    • D-Cycloserine, a partial agonist at the glycine site coupled to NMDA receptors, improves visual recognition memory in rhesus monkeys
    • MATSUOKA, N. AND AIGNER, T. G.: D-Cycloserine, a partial agonist at the glycine site coupled to NMDA receptors, improves visual recognition memory in rhesus monkeys. J. Pharmacol. Exp. Ther. 278: 891-897, 1996a.
    • (1996) J. Pharmacol. Exp. Ther. , vol.278 , pp. 891-897
    • Matsuoka, N.1    Aigner, T.G.2
  • 22
    • 0029867042 scopus 로고    scopus 로고
    • Cholinergic-glutamatergic interactions in visual recognition memory of rhesus monkeys
    • MATSUOKA, N. AND AIGNER, T. G.: Cholinergic-glutamatergic interactions in visual recognition memory of rhesus monkeys. NeuroReport 7: 565-568, 1996b.
    • (1996) NeuroReport , vol.7 , pp. 565-568
    • Matsuoka, N.1    Aigner, T.G.2
  • 23
    • 0025738845 scopus 로고
    • Somatostatin augments long-term potentiation of the mossy fiber-CA3 system in guinea-pig hippocampal slices
    • MATSUOKA, N., KANEKO, S. AND SATOH, M.: Somatostatin augments long-term potentiation of the mossy fiber-CA3 system in guinea-pig hippocampal slices. Brain Res. 553: 188-194, 1991.
    • (1991) Brain Res. , vol.553 , pp. 188-194
    • Matsuoka, N.1    Kaneko, S.2    Satoh, M.3
  • 24
    • 0028210630 scopus 로고
    • Possible involvement of brain somatostatin in the memory formation of rats and the cognitive enhancing action of FR121196 in passive avoidance task
    • MATSUOKA, N., MAEDA, N., YAMAGUCHI, I. AND SATOH, M.: Possible involvement of brain somatostatin in the memory formation of rats and the cognitive enhancing action of FR121196 in passive avoidance task. Brain Res. 642: 11-19, 1994.
    • (1994) Brain Res. , vol.642 , pp. 11-19
    • Matsuoka, N.1    Maeda, N.2    Yamaguchi, I.3    Satoh, M.4
  • 25
    • 0026490858 scopus 로고
    • Effects of FR121196, a novel cognitive enhancer, on the memory impairment of rats in passive avoidance and radial arm maze tasks
    • MATSUOKA, N., MAEDA, N., YAMAZAKI, M., OHKUBO, Y. AND YAMAGUCHI, I.: Effects of FR121196, a novel cognitive enhancer, on the memory impairment of rats in passive avoidance and radial arm maze tasks. J. Pharmacol. Exp. Ther. 263: 436-444, 1992.
    • (1992) J. Pharmacol. Exp. Ther. , vol.263 , pp. 436-444
    • Matsuoka, N.1    Maeda, N.2    Yamazaki, M.3    Ohkubo, Y.4    Yamaguchi, I.5
  • 26
    • 0027220292 scopus 로고
    • Role of somatostatin in the augmentation of hippocampal long-term potentiation by FR121196, a putative cognitive enhancer
    • MATSUOKA, N., YAMAGUCHI, I. AND SATOH, M.: Role of somatostatin in the augmentation of hippocampal long-term potentiation by FR121196, a putative cognitive enhancer. Eur. J. Pharmacol. 241: 27-34, 1993.
    • (1993) Eur. J. Pharmacol. , vol.241 , pp. 27-34
    • Matsuoka, N.1    Yamaguchi, I.2    Satoh, M.3
  • 27
    • 0029058321 scopus 로고
    • Changes in brain somatostatin in memory deficient rats: Comparison with cholinergic markers
    • MATSUOKA, N., YAMAZAKI, M. AND YAMAGUCHI, I.: Changes in brain somatostatin in memory deficient rats: Comparison with cholinergic markers. Neuroscience 66: 617-626, 1995.
    • (1995) Neuroscience , vol.66 , pp. 617-626
    • Matsuoka, N.1    Yamazaki, M.2    Yamaguchi, I.3
  • 28
    • 0027302996 scopus 로고
    • Glutamate: Its role in learning, memory, and the aging brain
    • MCENTEE, W. J. AND CROOK, T. H.: Glutamate: Its role in learning, memory, and the aging brain. Psychopharmacology 111: 391-401, 1993.
    • (1993) Psychopharmacology , vol.111 , pp. 391-401
    • Mcentee, W.J.1    Crook, T.H.2
  • 30
    • 0022650213 scopus 로고
    • Selective impairment of learning and blockade of long-term potentiation by an N-methyl-D-aspartate receptor antagonist, AP5
    • MORRIS, R. G. M., ANDERSON, E., LYNCH, G. S. AND BAUDRY, M.: Selective impairment of learning and blockade of long-term potentiation by an N-methyl-D-aspartate receptor antagonist, AP5. Nature (Lond.) 319: 774-776, 1986.
    • (1986) Nature (Lond.) , vol.319 , pp. 774-776
    • Morris, R.G.M.1    Anderson, E.2    Lynch, G.S.3    Baudry, M.4
  • 31
    • 0026437728 scopus 로고
    • Molecular diversity of glutamate receptors and implications for brain function
    • Wash. DC
    • NAKANISHI, S.: Molecular diversity of glutamate receptors and implications for brain function. Science (Wash. DC) 258: 597-603, 1992.
    • (1992) Science , vol.258 , pp. 597-603
    • Nakanishi, S.1
  • 32
    • 0027361335 scopus 로고
    • MK-801 impairs recognition memory in rhesus monkeys: Comparison with cholinergic drugs
    • OGURA, H. AND AIGNER, T. G,: MK-801 impairs recognition memory in rhesus monkeys: Comparison with cholinergic drugs. J. Pharmacol. Exp. Ther. 266: 60-64, 1993.
    • (1993) J. Pharmacol. Exp. Ther. , vol.266 , pp. 60-64
    • Ogura, H.1    Aigner, T.G.2
  • 33
    • 0025282045 scopus 로고
    • Is the neuronal basis of Alzheimer's disease cholinergic or glutamatergic?
    • PALMER, A. M. AND GERSHON, S.: Is the neuronal basis of Alzheimer's disease cholinergic or glutamatergic? FASEB J. 4: 2745-2752, 1990.
    • (1990) FASEB J. , vol.4 , pp. 2745-2752
    • Palmer, A.M.1    Gershon, S.2
  • 34
    • 0018078940 scopus 로고
    • Correlation of cholinergic abnormalities with senile Plaques and mental test scores in senile dementia
    • PERRY, E. K., TOMLINSON, B. E., BLESSED, G., BERGMANN, K., GIBSON, P. H. AND PERRY, R. H.: Correlation of cholinergic abnormalities with senile Plaques and mental test scores in senile dementia. Br. Med. J. 2: 1457-1459, 1978.
    • (1978) Br. Med. J. , vol.2 , pp. 1457-1459
    • Perry, E.K.1    Tomlinson, B.E.2    Blessed, G.3    Bergmann, K.4    Gibson, P.H.5    Perry, R.H.6
  • 35
    • 0017755565 scopus 로고
    • Scopolamine induced learning failures in man
    • PETERSEN, R.: Scopolamine induced learning failures in man. Psychopharmacology 52: 283-289, 1977.
    • (1977) Psychopharmacology , vol.52 , pp. 283-289
    • Petersen, R.1
  • 37
    • 0025818607 scopus 로고
    • A critical evaluation of monkey models of amnesia and dementia
    • RIDLEY, R. M. AND BAKER, H. F.: A critical evaluation of monkey models of amnesia and dementia. Brain Res. Rev. 16: 15-37, 1991.
    • (1991) Brain Res. Rev. , vol.16 , pp. 15-37
    • Ridley, R.M.1    Baker, H.F.2
  • 38
    • 0024343129 scopus 로고
    • Comparison of the effects of four cholinomimetic agents on cognition in primates following disruption by scopolamine or by lists of objects
    • RUPNIAK, N. M., STEVENTON, M. J., FIELD, M. J., JENNINGS, C. A. AND IVERSEN, S. D.: Comparison of the effects of four cholinomimetic agents on cognition in primates following disruption by scopolamine or by lists of objects. Psychopharmacology 99: 189-195, 1989.
    • (1989) Psychopharmacology , vol.99 , pp. 189-195
    • Rupniak, N.M.1    Steventon, M.J.2    Field, M.J.3    Jennings, C.A.4    Iversen, S.D.5
  • 39
    • 0020047820 scopus 로고
    • Depletion of somatostatin-like immunoreactivity in the rat central nervous system by cysteamine
    • SAGAR, S. M., LANDRY, D., MILLABD, W. J., BADGER, T. M., ARNOLD, M. A. AND MARTIN, J. B.: Depletion of somatostatin-like immunoreactivity in the rat central nervous system by cysteamine. J. Neurosci. 2: 225-231, 1982.
    • (1982) J. Neurosci. , vol.2 , pp. 225-231
    • Sagar, S.M.1    Landry, D.2    Millabd, W.J.3    Badger, T.M.4    Arnold, M.A.5    Martin, J.B.6
  • 40
    • 0023081892 scopus 로고
    • Some limitations of indices derived from signal detection theory: Evaluation of an alternative index for measuring bias in memory tasks
    • SAHGAL, A.: Some limitations of indices derived from signal detection theory: Evaluation of an alternative index for measuring bias in memory tasks. Psychopharmacology 91: 517-520, 1987.
    • (1987) Psychopharmacology , vol.91 , pp. 517-520
    • Sahgal, A.1
  • 41
    • 0021168402 scopus 로고
    • Cholinergic hypothesis of human memory: Review of basic and clinical studies
    • SITARAM, N.: Cholinergic hypothesis of human memory: Review of basic and clinical studies. Drug Dev. Res. 4: 481-488, 1984.
    • (1984) Drug Dev. Res. , vol.4 , pp. 481-488
    • Sitaram, N.1
  • 42
    • 0021261726 scopus 로고
    • Long-term potentiation as a candidate mnemonic device
    • TEYLER, T. J. AND DISCENNA, P.: Long-term potentiation as a candidate mnemonic device. Brain Res. Rev. 7: 15-28, 1984.
    • (1984) Brain Res. Rev. , vol.7 , pp. 15-28
    • Teyler, T.J.1    Discenna, P.2
  • 43
    • 0027732608 scopus 로고
    • A primate model of Alzheimer's disease
    • WENK, G. L.: A primate model of Alzheimer's disease. Behav. Brain Res. 57: 117-122, 1993.
    • (1993) Behav. Brain Res. , vol.57 , pp. 117-122
    • Wenk, G.L.1
  • 44
    • 0024412746 scopus 로고
    • Immediate and long-lasting effects of MK-801 on motor activity, spatial navigation in a swimming pool and EEG in the rat
    • WHISHAW, I. Q. AND AUER, R. N.: Immediate and long-lasting effects of MK-801 on motor activity, spatial navigation in a swimming pool and EEG in the rat. Psychopharmacology 98: 500-507, 1989.
    • (1989) Psychopharmacology , vol.98 , pp. 500-507
    • Whishaw, I.Q.1    Auer, R.N.2
  • 45
    • 0030426833 scopus 로고    scopus 로고
    • FK960, N-(4-Acetyl-1-piperazinyl)-p-fluorobenzamide monohydrate, ameliorates the memory defects in rats through a novel mechanism of action
    • YAMAZAKI, M., MATSUOKA, N., MAEDA, N., OHKUBO, Y. AND YAMAGUCHI, I.: FK960, N-(4-Acetyl-1-piperazinyl)-p-fluorobenzamide monohydrate, ameliorates the memory defects in rats through a novel mechanism of action. J. Pharmacol. Exp. Ther., 279: 1157-1173, 1996.
    • (1996) J. Pharmacol. Exp. Ther. , vol.279 , pp. 1157-1173
    • Yamazaki, M.1    Matsuoka, N.2    Maeda, N.3    Ohkubo, Y.4    Yamaguchi, I.5
  • 46
    • 0025737591 scopus 로고
    • Behavioural, electrophysiological and histopathological changes following sustained stimulation of the perforant pathway input to the hippocampus: Effect of the NMDA receptor antagonist, CGP 39551
    • YLINEN, A., LAHTINEN, H., SIRVIO, J., PARTANEN, J., ASIKAINEN, A., GULYAS, A., FREUND, T. F. AND RIEKKINEN, P.: Behavioural, electrophysiological and histopathological changes following sustained stimulation of the perforant pathway input to the hippocampus: Effect of the NMDA receptor antagonist, CGP 39551. Brain Res. 553: 195-200, 1991.
    • (1991) Brain Res. , vol.553 , pp. 195-200
    • Ylinen, A.1    Lahtinen, H.2    Sirvio, J.3    Partanen, J.4    Asikainen, A.5    Gulyas, A.6    Freund, T.F.7    Riekkinen, P.8


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