(+)-WAY 100135, a partial agonist, at native and recombinant 5-HT(1B/1D) receptors

British Journal of Pharmacology

Volumn 121, Issue 4, 1997, Pages 737-742

  Davidson, Colin ^a,c   Ho, Michael ^b   Price, Gary W ^b   Jones, Brian J ^b   Stamford, Jonathan A ^a,d  

^a ST BARTHOLOMEW S HOSPITAL   (United Kingdom)

^b GLAXOSMITHKLINE   (United Kingdom)

^c UNIVERSITY OF ST ANDREWS   (United Kingdom)

^d ROYAL LONDON HOSPITAL   (United Kingdom)

Author keywords

(+) WAY100135; 5 HT(1B 1D) autoreceptor; 5 hydroxytryptamine (5 HT); 35S GTP S binding; Fast cyclic voltammetry; Lateral geniculate nucleus; Partial agonist

Indexed keywords

GUANOSINE 5' O (3 THIOTRIPHOSPHATE); METITEPINE; N [4 METHOXY 3 (4 METHYL 1 PIPERAZINYL)PHENYL] 2' METHYL 4' (5 METHYL 1,2,4 OXADIAZOL 3 YL)[1,1' BIPHENYL] 4 CARBOXAMIDE; N TERT BUTYL 3 [4 (2 METHOXYPHENYL) 1 PIPERAZINYL] 2 PHENYLPROPIONAMIDE; PAROXETINE; PARTIAL AGONIST; RADIOLIGAND; SEROTONIN; SEROTONIN 1A ANTAGONIST; SEROTONIN 1B RECEPTOR; SEROTONIN 1D RECEPTOR; SULFUR 35;

ANIMAL CELL; ARTICLE; CHO CELL; CONTROLLED STUDY; CYCLIC POTENTIOMETRY; FEMALE; HALF LIFE TIME; LATERAL GENICULATE NUCLEUS; LIGAND BINDING; NONHUMAN; PRIORITY JOURNAL; RECEPTOR AFFINITY;

ANIMALS; CHO CELLS; CRICETINAE; GENICULATE BODIES; HUMANS; MALE; PIPERAZINES; RATS; RATS, WISTAR; SEROTONIN; SEROTONIN AGONISTS; SEROTONIN ANTAGONISTS;

EID: 0030947665     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0701197     Document Type: Article

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