General approach to the synthesis of optically active 2-carboxy-4-[3'-(diethoxyphosphinyl)propyl]-5-alkylpip erazines (CPP analogues)

Tetrahedron Asymmetry

Volumn 8, Issue 10, 1997, Pages 1633-1639

  Falorni, Massimo ^a   Porcheddu, Andrea ^a   Giacomelli, Giampaolo ^a  

^a UNIVERSITY OF SASSARI   (Italy)

Author keywords

[No Author keywords available]

Indexed keywords

N METHYL DEXTRO ASPARTIC ACID RECEPTOR BLOCKING AGENT;

ALKYLATION; ARTICLE; DRUG SYNTHESIS; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; PRIORITY JOURNAL; REACTION ANALYSIS; STEREOCHEMISTRY;

EID: 0030940903     PISSN: 09574166     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0957-4166(97)00157-2     Document Type: Article

References (10)

1. See for examples: Johnson, R.L.; Koerner, J.F., J. Med. Chem., 1988, 31, 2057-2066. Hashimoto, K.; Shirahama, H., Tetrahedron Lett., 1991, 32, 2625-2628.
2. See for examples: Johnson, R.L.; Koerner, J.F., J. Med. Chem., 1988, 31, 2057-2066. Hashimoto, K.; Shirahama, H., Tetrahedron Lett., 1991, 32, 2625-2628.
3. Hays, S.J.; Bigge, C.F.; Novak, P.M.; Drummond, J.T.; Bobovski, T.P.; Rice, M.J.; Johnson, G.; Brahce, L.J.; Coughenour, L.L., J. Med. Chem., 1990, 33, 2916-2924.
4. Falorni, M.; Porcheddu, A.; Giacomelli, G., Tetrahedron: Asymmetry, 1996, 7, 1999-2005.
5. Carlsen, H.J.; Katsuki, T.; Martin, VS.; Sharpless K.B. J. Org. Chem., 1981, 46, 3936.
6. 3 as catalyst causes the oxidative decomposition of the substrates.
7. Shamma, M.; Deno, N.C.; Remar, J.F. Tetrahedron Lett., 1966, 1375.
8. Wilson, N.D.V.; Joule, J.A. Tetrahedron, 1968, 24, 5493-5497.
9. 2].
10. Falorni, M.; Satta, M.; Conti, S.; Giacomelli, G. Tetrahedron: Asymmetry 1993, 4, 2389-2398.