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Volumn 280, Issue 1, 1997, Pages 73-82

Psychopharmacological profile of amisulpride: An antipsychotic drug with presynaptic D2/D3 dopamine receptor antagonist activity and limbic selectivity

Author keywords

[No Author keywords available]

Indexed keywords

2 DIPROPYLAMINO 7 HYDROXYTETRALIN; AMISULPRIDE; APOMORPHINE; BENZAMIDE DERIVATIVE; DEXAMPHETAMINE; DOPAMINE 2 RECEPTOR BLOCKING AGENT; DOPAMINE 3 RECEPTOR BLOCKING AGENT; HALOPERIDOL; NEUROLEPTIC AGENT; PRESYNAPTIC RECEPTOR; QUINPIROLE; REMOXIPRIDE;

EID: 0030933627     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article
Times cited : (240)

References (66)
  • 4
    • 0017853040 scopus 로고
    • Antipsychotic drugs, neurotransmitters and schizophrenia
    • CARLSSON, A.: Antipsychotic drugs, neurotransmitters and schizophrenia. Am. J. Psychiatry 135: 164-173, 1978.
    • (1978) Am. J. Psychiatry , vol.135 , pp. 164-173
    • Carlsson, A.1
  • 5
    • 0022517170 scopus 로고
    • Behavioral deficits induced by low doses of apomorphine in rats: Evidence for a moti- Vational and cognitive dysfunction which discriminates among neuroleptic drugs
    • CARNOY, P., RAVARD, S., WEMERMAN, B., SOUBRIE, PH. AND SIMON, P.: Behavioral deficits induced by low doses of apomorphine in rats: Evidence for a moti- vational and cognitive dysfunction which discriminates among neuroleptic drugs. Pharmacol. Biochem. Behav. 25: 503-509, 1986.
    • (1986) Pharmacol. Biochem. Behav. , vol.25 , pp. 503-509
    • Carnoy, P.1    Ravard, S.2    Wemerman, B.3    Soubrie, P.H.4    Simon, P.5
  • 6
    • 0019366354 scopus 로고
    • Swim-induced grooming in mice is mediated by a dopaminergic substrate
    • CHESHER, G. B. AND JACKSON, D. M.: Swim-induced grooming in mice is mediated by a dopaminergic substrate. J. Neural. Transm. 50: 47-55, 1981.
    • (1981) J. Neural. Transm. , vol.50 , pp. 47-55
    • Chesher, G.B.1    Jackson, D.M.2
  • 7
    • 0019196339 scopus 로고
    • Evidence for thermoregulatory dopaminergic receptors located in the preopticus medialis nucleus of the rat hypothalamus
    • COLBOC, O. AND COSTENTIN, J.: Evidence for thermoregulatory dopaminergic receptors located in the preopticus medialis nucleus of the rat hypothalamus. J. Pharm. Pharmacol. 32: 624-629, 1980.
    • (1980) J. Pharm. Pharmacol. , vol.32 , pp. 624-629
    • Colboc, O.1    Costentin, J.2
  • 8
    • 0015059469 scopus 로고
    • Cholinergic- And neuroleptic-induced catalepsy: Modification by lesions in the caudate-putamen
    • COSTALL, B. AND OLLEY, J. E.: Cholinergic- and neuroleptic-induced catalepsy: Modification by lesions in the caudate-putamen, Neuropharmaculogy 10: 297-306, 1971.
    • (1971) Neuropharmaculogy , vol.10 , pp. 297-306
    • Costall, B.1    Olley, J.E.2
  • 9
    • 0015596875 scopus 로고
    • On the mode of action of apomorphine
    • COSTALL, B. AND NAYLOR, R. J.: On the mode of action of apomorphine. Eur. J. Pharmacol. 21: 350-361, 1973.
    • (1973) Eur. J. Pharmacol. , vol.21 , pp. 350-361
    • Costall, B.1    Naylor, R.J.2
  • 10
    • 0017387026 scopus 로고
    • Differentiation of the dopamine mechanisms mediating stereotyped behaviour and hyperactivity in the nucleus accumbens and caudate-putamen
    • COSTALL, B., NAYLOR, R. J., CANNON, J. G. AND LEE, T.: Differentiation of the dopamine mechanisms mediating stereotyped behaviour and hyperactivity in the nucleus accumbens and caudate-putamen. J. Pharm. Pharmacol. 29: 337-342, 1977.
    • (1977) J. Pharm. Pharmacol. , vol.29 , pp. 337-342
    • Costall, B.1    Naylor, R.J.2    Cannon, J.G.3    Lee, T.4
  • 11
    • 0018227116 scopus 로고
    • Climbing behaviour induced by apomorphine in mice: A potential model for the detection of neuroleptic activity
    • COSTALL, B., NAYLOR, R. J. AND NOHRIA, V.: Climbing behaviour induced by apomorphine in mice: A potential model for the detection of neuroleptic activity. Eur. J. Pharmacol. 50: 39-50, 1978.
    • (1978) Eur. J. Pharmacol. , vol.50 , pp. 39-50
    • Costall, B.1    Naylor, R.J.2    Nohria, V.3
  • 12
    • 0016786303 scopus 로고
    • Rapid and dissociated changes in sensitivities of different dopamine receptors in mouse brain
    • COSTENTIN, J., PROTAIS, P. AND SCHWARTZ, J. C.: Rapid and dissociated changes in sensitivities of different dopamine receptors in mouse brain. Nature (Lond.) 257: 405-407, 1975.
    • (1975) Nature (Lond.) , vol.257 , pp. 405-407
    • Costentin, J.1    Protais, P.2    Schwartz, J.C.3
  • 13
    • 0027446260 scopus 로고
    • Subcortical dopamine and aerotonin turnover during acute and subchronic administration of typical and atypical neuroleptics
    • CSERNANSKY, J. G., WRONA, C. T., BARDGETT. M. E., EARLY, T. S. AND NEWCOMER, J. W.: Subcortical dopamine and aerotonin turnover during acute and subchronic administration of typical and atypical neuroleptics. Psychopharmacology 110: 145-151, 1993.
    • (1993) Psychopharmacology , vol.110 , pp. 145-151
    • Csernansky, J.G.1    Wrona, C.T.2    Bardgett, M.E.3    Early, T.S.4    Newcomer, J.W.5
  • 15
    • 0025083023 scopus 로고
    • Amisulpride versus haloperidol in treatment of schizophrenic patients - Results of a double-blind study
    • DELCKER, A., SCHOON, M. L., OCZKOWSKI, B. AND GAERTNER, H. J.: Amisulpride versus haloperidol in treatment of schizophrenic patients - Results of a double-blind study. Pharmacopaychiatry 23: 125-130, 1990.
    • (1990) Pharmacopaychiatry , vol.23 , pp. 125-130
    • Delcker, A.1    Schoon, M.L.2    Oczkowski, B.3    Gaertner, H.J.4
  • 16
  • 17
    • 0017146682 scopus 로고
    • Evidence for dopamine receptors mediating sedation in the mouse brain
    • DICHIARA, G., PORCEDDU, M. L., VARGIU, L., ARGIOLAS, A. AND GESSA, G. L.: Evidence for dopamine receptors mediating sedation in the mouse brain. Nature (Lond.) 264: 564-567, 1976.
    • (1976) Nature (Lond.) , vol.264 , pp. 564-567
    • Dichiara, G.1    Porceddu, M.L.2    Vargiu, L.3    Argiolas, A.4    Gessa, G.L.5
  • 18
    • 0022358917 scopus 로고
    • Bilateral lesions of the striatum induced with 6-hydroxydopamine abolish apomorphine-induced yawning in rats
    • DOURISH, C. T. AND HUTSON, P. H.: Bilateral lesions of the striatum induced with 6-hydroxydopamine abolish apomorphine-induced yawning in rats. Neuropharmacology 24: 1051-1055, 1985.
    • (1985) Neuropharmacology , vol.24 , pp. 1051-1055
    • Dourish, C.T.1    Hutson, P.H.2
  • 19
    • 0024518016 scopus 로고
    • Biphasic effect of D-2 agonist quinpirole on locomotion and movements
    • EILAM D. AND SZECHTMAN, H.: Biphasic effect of D-2 agonist quinpirole on locomotion and movements. Eur. J. Pharmacol. 161: 151-157, 1989.
    • (1989) Eur. J. Pharmacol. , vol.161 , pp. 151-157
    • Eilam, D.1    Szechtman, H.2
  • 20
    • 0014178399 scopus 로고
    • Mode of action of apomorphine and dexamphetamine on gnawing compulsion in rats
    • ERNST, A. M.: Mode of action of apomorphine and dexamphetamine on gnawing compulsion in rats. Psychopharmacologia 10: 316-323, 1967.
    • (1967) Psychopharmacologia , vol.10 , pp. 316-323
    • Ernst, A.M.1
  • 21
    • 0026718710 scopus 로고
    • 2 dopamine receptor occupancy in patients treated with classical neuroleptics and clozapine: Relation to extrapyramidal side effects
    • 2 dopamine receptor occupancy in patients treated with classical neuroleptics and clozapine: Relation to extrapyramidal side effects. Arch. Gen Psychiatry 49: 538-544, 1992.
    • (1992) Arch. Gen Psychiatry , vol.49 , pp. 538-544
    • Farde, L.1    Nordström, A.L.2    Wiesel, F.A.3    Pauli, S.4    Halldin, C.5    Sedvall, G.6
  • 23
    • 0015395994 scopus 로고
    • Hypothermic effect of apomorphine in the mouse
    • FUXE, K. AND SJÖQVIST, F.: Hypothermic effect of apomorphine in the mouse. J. Pharm. Pharmac. 24: 702-705, 1972.
    • (1972) J. Pharm. Pharmac. , vol.24 , pp. 702-705
    • Fuxe, K.1    Sjöqvist, F.2
  • 24
    • 0027452773 scopus 로고
    • Potentiation by low doses of selected neuroleptics of food-induced conditioned place preference in rata
    • GUYON, A., ASSOULY-BESSE, F., BIALA, G., PUECH, A. J. AND THIÉBOT, M. H.: Potentiation by low doses of selected neuroleptics of food-induced conditioned place preference in rata. Psychopharmacology 110: 460-466, 1993.
    • (1993) Psychopharmacology , vol.110 , pp. 460-466
    • Guyon, A.1    Assouly-Besse, F.2    Biala, G.3    Puech, A.J.4    Thiébot, M.H.5
  • 25
    • 0016826092 scopus 로고
    • Amphetamine and apomorphine responses in the rat following 6-OHDA lesions of the nucleus accumbens septi and corpus striatum
    • KELLY, P. H., SEVIOUR, P. W. AND IVERSEN, S. D.: Amphetamine and apomorphine responses in the rat following 6-OHDA lesions of the nucleus accumbens septi and corpus striatum. Brain Res. 94: 507-522, 1975.
    • (1975) Brain Res. , vol.94 , pp. 507-522
    • Kelly, P.H.1    Seviour, P.W.2    Iversen, S.D.3
  • 26
    • 0018760240 scopus 로고
    • 3H-spiperone binding in vivo: Biochemical and behavioural evidence for a preferential action on limbic and nigral dopamine receptors
    • 3H-spiperone binding in vivo: Biochemical and behavioural evidence for a preferential action on limbic and nigral dopamine receptors. Neurosci. Lett. 13: 51-56, 1979.
    • (1979) Neurosci. Lett. , vol.13 , pp. 51-56
    • Ogren, S.O.1    Haglund, L.2    Angeby, T.3
  • 29
    • 0024580391 scopus 로고
    • Hypothermia in mice: D2 dopamine receptor mediation and absence of spare receptors
    • MELLER, E., HIZAMI, R. AND KREUTER, L.: Hypothermia in mice: D2 dopamine receptor mediation and absence of spare receptors. Pharmacol. Biochem. Behav. 32: 141-145, 1989.
    • (1989) Pharmacol. Biochem. Behav. , vol.32 , pp. 141-145
    • Meller, E.1    Hizami, R.2    Kreuter, L.3
  • 30
    • 0018775859 scopus 로고
    • Hypothermic effects of apomorphine homologues in mice
    • MENON, M. K., CLARK, W. G. AND CANNON J. G.: Hypothermic effects of apomorphine homologues in mice. J. Pharm. Pharmacol. 31: 318-321, 1979.
    • (1979) J. Pharm. Pharmacol. , vol.31 , pp. 318-321
    • Menon, M.K.1    Clark, W.G.2    Cannon, J.G.3
  • 33
    • 0017759072 scopus 로고
    • Drugs affecting dopamine neurons and yawning behaviour
    • MOGILNICKA, E. AND KLIMEK, V.: Drugs affecting dopamine neurons and yawning behaviour. Pharmac. Biochem. Behav. 7: 303-305, 1977.
    • (1977) Pharmac. Biochem. Behav. , vol.7 , pp. 303-305
    • Mogilnicka, E.1    Klimek, V.2
  • 34
    • 0021322874 scopus 로고
    • Effects of apomorphine. TL-99 and 3-PPP on yawning in rats
    • MOGILNICKA, E., BOISSARD, C. G. AND DELINI-STULA, A.: Effects of apomorphine. TL-99 and 3-PPP on yawning in rats. Neuropharmacology 23: 19-22, 1984.
    • (1984) Neuropharmacology , vol.23 , pp. 19-22
    • Mogilnicka, E.1    Boissard, C.G.2    Delini-Stula, A.3
  • 36
    • 0025193887 scopus 로고
    • The role of multiple dopamine receptors in apomorphine and N-n-propylnorapomorphine-induced climbing and hypothermia
    • MOORE, N. A. AND AXTON, M. S.: The role of multiple dopamine receptors in apomorphine and N-n-propylnorapomorphine-induced climbing and hypothermia. Eur. J. Pharmacol. 178: 195-201, 1990.
    • (1990) Eur. J. Pharmacol. , vol.178 , pp. 195-201
    • Moore, N.A.1    Axton, M.S.2
  • 37
    • 0023866774 scopus 로고
    • Changes in dopamine autoreceptor sensitivity in animal model of depression
    • MUSCAT, R., TOWELL, A. AND WINNER, P.: Changes in dopamine autoreceptor sensitivity in animal model of depression. Psychopharmacology 94: 545-550, 1988.
    • (1988) Psychopharmacology , vol.94 , pp. 545-550
    • Muscat, R.1    Towell, A.2    Winner, P.3
  • 39
    • 0021251069 scopus 로고
    • Remoxipride, a new potential antipsychotic compound with selective anti-dopaminergic actions in the rat brain
    • ÖRGEN, S. O., HALL, H., KÖHLER, C., MAGNUSSON, O., LINDBOM, L. O., ANGEBY, K. AND FLORVALL, L.: Remoxipride, a new potential antipsychotic compound with selective anti-dopaminergic actions in the rat brain. Eur. J. Pharmacol. 102: 459-474, 1984.
    • (1984) Eur. J. Pharmacol. , vol.102 , pp. 459-474
    • Örgen, S.O.1    Hall, H.2    Köhler, C.3    Magnusson, O.4    Lindbom, L.O.5    Angeby, K.6    Florvall, L.7
  • 40
  • 41
    • 0017119483 scopus 로고
    • Climbing behaviour induced by apomorphine in mice: A simple test for the study of dopamine receptors in striatum
    • PHOTAIS, P., COSTENTIN, J. AND SCHWARTZ, J. C.: Climbing behaviour induced by apomorphine in mice: A simple test for the study of dopamine receptors in striatum. Psychopharmacology 50: 1-6, 1976.
    • (1976) Psychopharmacology , vol.50 , pp. 1-6
    • Photais, P.1    Costentin, J.2    Schwartz, J.C.3
  • 42
    • 0019834447 scopus 로고
    • Pharmacological properties of new antipsychotic agents: Use of animal models
    • PUECH, A. J., RIOUX, P., PONCELET, M., BROCHET, D., CHERMAT, R. AND SIMON, P.: Pharmacological properties of new antipsychotic agents: Use of animal models. Neuropharmacology 20: 1279-1284, 1981.
    • (1981) Neuropharmacology , vol.20 , pp. 1279-1284
    • Puech, A.J.1    Rioux, P.2    Poncelet, M.3    Brochet, D.4    Chermat, R.5    Simon, P.6
  • 43
    • 0026557084 scopus 로고
    • 2 receptor agonists with high and low efficacies
    • 2 receptor agonists with high and low efficacies. Eur. J. Pharmacol. 211: 9-14, 1992.
    • (1992) Eur. J. Pharmacol. , vol.211 , pp. 9-14
    • Sanchez, C.1    Arnt, J.2
  • 44
    • 0028869750 scopus 로고
    • Effects of typical and atypical antipsychotic drugs on response decrement patterns in rats
    • SANGER, D. J. AND PERRAULT, GH.: Effects of typical and atypical antipsychotic drugs on response decrement patterns in rats. J. Pharmacol. Exp. Ther. 272: 708-713, 1995.
    • (1995) J. Pharmacol. Exp. Ther. , vol.272 , pp. 708-713
    • Sanger, D.J.1    Perrault, Gh.2
  • 46
    • 0017744479 scopus 로고
    • Regional effects of neuroleptics on dopamine metabolism and dopamine-sensitive adenylate cyclase activity
    • SCATTON, B., BISCHOFF, S., DEDEK, J. AND KORF, J.: Regional effects of neuroleptics on dopamine metabolism and dopamine-sensitive adenylate cyclase activity. Eur. J. Pharmacol. 44: 287-292, 1977.
    • (1977) Eur. J. Pharmacol. , vol.44 , pp. 287-292
    • Scatton, B.1    Bischoff, S.2    Dedek, J.3    Korf, J.4
  • 47
    • 0020041211 scopus 로고
    • Effect of dopamine agonists and neuroleptic agents on striatal acetylcholine transmission in the rat: Evidence against dopamine receptor multiplicity
    • SCATTON, B.: Effect of dopamine agonists and neuroleptic agents on striatal acetylcholine transmission in the rat: Evidence against dopamine receptor multiplicity. J. Pharmacol. Exp. Ther. 220: 197-202, 1982.
    • (1982) J. Pharmacol. Exp. Ther. , vol.220 , pp. 197-202
    • Scatton, B.1
  • 49
    • 0027743268 scopus 로고
    • Occupancy of central neurotransmitter receptors by risperidone, clozapine and haloperidol, measured ex vivo by quantitative autoradiography
    • SCHOTTE, A., JANSSEN, P. F. M., MEGENS, A. A. H. P. AND LEYSEN, J. E.: Occupancy of central neurotransmitter receptors by risperidone, clozapine and haloperidol, measured ex vivo by quantitative autoradiography. Brain Research 631: 191-202, 1993.
    • (1993) Brain Research , vol.631 , pp. 191-202
    • Schotte, A.1    Janssen, P.F.M.2    Megens, A.A.H.P.3    Leysen, J.E.4
  • 51
    • 0018805131 scopus 로고
    • Chronic treatment with antidepressants prevents the inhibitory effect of small doses of apomorphine on dopamine synthesis and motor activity
    • SERRA, G., ARGIOLAS, A., KLIMEK, V., FADDA, F. AND GESSA, G. L.: Chronic treatment with antidepressants prevents the inhibitory effect of small doses of apomorphine on dopamine synthesis and motor activity. Life Sci. 25: 415-424, 1979.
    • (1979) Life Sci. , vol.25 , pp. 415-424
    • Serra, G.1    Argiolas, A.2    Klimek, V.3    Fadda, F.4    Gessa, G.L.5
  • 52
  • 56
    • 0026800560 scopus 로고
    • Do autoreceptors mediate dopamine agonist induced yawning and suppression of exploration? A critical review
    • STÄHLE, L.: Do autoreceptors mediate dopamine agonist induced yawning and suppression of exploration? A critical review. Psychopharmacology 106: 1-13, 1992.
    • (1992) Psychopharmacology , vol.106 , pp. 1-13
    • Stähle, L.1
  • 57
    • 0022461560 scopus 로고
    • Effects of neuroleptic drugs on the inhibition of exploratory behaviour induced by a low dose of apomorphine: Implications for the identity of dopamine receptors
    • STÄHLE, L. AND UNGERSTEDT, U.: Effects of neuroleptic drugs on the inhibition of exploratory behaviour induced by a low dose of apomorphine: Implications for the identity of dopamine receptors. Pharmacol. Biochem. Behav. 25: 473-480, 1986.
    • (1986) Pharmacol. Biochem. Behav. , vol.25 , pp. 473-480
    • Stähle, L.1    Ungerstedt, U.2
  • 58
    • 0023126754 scopus 로고
    • Differential effects of the dopamine antagonist remoxipride on apomorphine induced behaviour in the rat
    • STÄHLE, L., LJUNGBERG, T., RODEBJER, A., OGREN S. O. AND UNGERSTEDT, U.: Differential effects of the dopamine antagonist remoxipride on apomorphine induced behaviour in the rat. Pharmacol. Toxicol. 60: 227-232, 1987.
    • (1987) Pharmacol. Toxicol. , vol.60 , pp. 227-232
    • Stähle, L.1    Ljungberg, T.2    Rodebjer, A.3    Ogren, S.O.4    Ungerstedt, U.5
  • 61
    • 0023832391 scopus 로고
    • Climbing and stereotyped behaviours in mice require the stimulation of D-1 dopamine receptors
    • VASSE, M., CHAGRAOUI, A. AND PROTAIS, P.: Climbing and stereotyped behaviours in mice require the stimulation of D-1 dopamine receptors. Eur. J. Pharmacol. 148: 221-229, 1988.
    • (1988) Eur. J. Pharmacol. , vol.148 , pp. 221-229
    • Vasse, M.1    Chagraoui, A.2    Protais, P.3
  • 62
    • 0021824086 scopus 로고
    • Unexpected potentiation by discriminant benzamide derivatives of stereotyped behaviours elicited by dopamine agonists in mice
    • VASSE, M., PROTAIS, P., COSTENTIN, J. AND SCHWARTZ, J. C.: Unexpected potentiation by discriminant benzamide derivatives of stereotyped behaviours elicited by dopamine agonists in mice. Naunyn-Schmied. Arch. Pharmacol. 329: 108-116, 1985.
    • (1985) Naunyn-Schmied. Arch. Pharmacol. , vol.329 , pp. 108-116
    • Vasse, M.1    Protais, P.2    Costentin, J.3    Schwartz, J.C.4
  • 63
    • 0018392288 scopus 로고
    • Predictability and specificity of behavioral screening tests for neuroleptics
    • WORMS, P. AND LLOYD, K. G.: Predictability and specificity of behavioral screening tests for neuroleptics. Pharmacol. Ther. 5: 445-450, 1979.
    • (1979) Pharmacol. Ther. , vol.5 , pp. 445-450
    • Worms, P.1    Lloyd, K.G.2
  • 64
    • 0018841172 scopus 로고
    • Direct evidence for involvement of dopaminergic inhibition and cholinergic activation in yawning
    • YAMADA, K. AND FUKUKAWA, T.: Direct evidence for involvement of dopaminergic inhibition and cholinergic activation in yawning. Psychopharmacology 67: 39-43, 1980.
    • (1980) Psychopharmacology , vol.67 , pp. 39-43
    • Yamada, K.1    Fukukawa, T.2
  • 65
    • 0028170936 scopus 로고
    • 1 dopamine receptor-mediated behaviors in normal mice and in mice lesioned with 6-hydroxydopamine
    • 1 dopamine receptor-mediated behaviors in normal mice and in mice lesioned with 6-hydroxydopamine. J. Pharmacol. Exp. Ther. 271: 1462-1470, 1994.
    • (1994) J. Pharmacol. Exp. Ther. , vol.271 , pp. 1462-1470
    • Zhang, S.P.1    Zhou, L.W.2    Weiss, B.3
  • 66
    • 0016815658 scopus 로고
    • Effects of thioridazine. clozapine and other antipsychotics on the kinetic state of tyrosine hydroxylase and on the turnover rate of dopamine in striatum and nucleus accumbens
    • ZIVKOVIC, B., GUIDOTTI, A., REVUELTA, A. AND COSTA, E.: Effects of thioridazine. clozapine and other antipsychotics on the kinetic state of tyrosine hydroxylase and on the turnover rate of dopamine in striatum and nucleus accumbens. J. Pharmacol. Exp. Ther. 194: 37-46, 1975.
    • (1975) J. Pharmacol. Exp. Ther. , vol.194 , pp. 37-46
    • Zivkovic, B.1    Guidotti, A.2    Revuelta, A.3    Costa, E.4


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