Effect of an active metabolite of the antiallergic agent tazanolast on histamine release from rat mast cells

Arzneimittel-Forschung/Drug Research

Volumn 47, Issue 4, 1997, Pages 390-394

  Kamei, Chiaki ^a   Mio, Mitsunobu ^a   Yoshida, Tomokazu ^a   Saito, Yoko ^b   Toyoda, Yoshihiro ^b   Tsuriya, Yoshihiro ^b  

^a OKAYAMA UNIVERSITY   (Japan)

^b Wakamoto Pharmaceutical Co Ltd   (Japan)

Author keywords

antiallergic agents; CAS 114607 46 4; CAS 82989 25 1; tazanolast, active metabolite; WP 871, effect on histamine release

Indexed keywords

3 (1H TETRAZOL 5 YL)OXANILIC ACID; ANTIALLERGIC AGENT; CALCIUM; COMPOUND 48-80; CROMOGLYCATE DISODIUM; CYCLIC AMP; DRUG METABOLITE; INOSITOL 1,4,5 TRISPHOSPHATE; PHOSPHOLIPASE C; PROTEIN KINASE C; TAZANOLAST;

ANIMAL CELL; ARTICLE; CALCIUM TRANSPORT; CONTROLLED STUDY; DOSE RESPONSE; HISTAMINE RELEASE; IN VITRO STUDY; ISOTOPE LABELING; MALE; MAST CELL; NONHUMAN; RAT;

ANIMALS; ANTI-ALLERGIC AGENTS; CALCIUM RADIOISOTOPES; CYCLIC AMP; DOSE-RESPONSE RELATIONSHIP, DRUG; HISTAMINE RELEASE; INOSINE TRIPHOSPHATE; MALE; MAST CELLS; PHOSPHOLIPASE C; PROTEIN KINASE C; RATS; RATS, WISTAR; TETRAZOLES;

EID: 0030926980     PISSN: 00044172     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (25)

1. Miyamoto, T., Takahashi, T., Ito, K. et al., Ther. Res. 15, 2747 (1994)
2. Esumi, Y., Mitsugu, K., Hayashi, K. et al., Clin. Rep. 23, 451 (1989)
3. Hashimoto, T., Edanami, K., Naito, A. et al., Folia Pharmacol. Japon. 95, 159 (1990)
4. Hashimoto, T., Yamada, M., Toyoda, Y. et al., Kokyu 12, 484 (1993)
5. Tasaka, K., Mio, M., Okamoto, M., Ann. Allergy 56, 464 (1986)
6. Spataro, A. C., Bosmann, H. B., Biochem. Pharmacol. 25, 505 (1976)
7. Tanizaki, Y., Ohtani, J., Kimura, I., Agents Actions 37, 8 (1992)
8. Mio, M., Izushi, K., Tasaka, K., Immunopharmacology 22, 59 (1991)
9. Komatsu, H., Kojima, M., Tsutsumi, N. et al., Japan. J. Pharmacol. 46, 43 (1988)
10. Tasaka, K., Akagi, M., Mio, M. et al., Int. Arch. Allergy Appl. Immunol. 83, 348 (1987)
11. Shore, P. A., Burkhalter, A., Cohn, V. H. Jr., J. Pharmacol. Exp. Ther. 127, 182 (1959)
12. Enerbäck, L., Svensson, I., J. Immunol. Methods 39, 135 (1980)
13. Izushi, K., Shirasaka, T., Chokki, M. et al., FEBS Letters 314, 241 (1992)
14. Martin, T. F. J., Kowalchyk, J. A., J. Biol. Chem. 264, 20917 (1989)
15. Izushi, K., Tasaka, K., Pharmacology 44, 61 (1992)
16. Tasaka, K., Sugimoto, Y., Mio, M., Int. Arch. Allergy Appl. Immunol. 91, 211 (1990)
17. Scharenberg, A. M., Kinet, J. P., J. Allergy Clin. Immunol. 94, 1142 (1994)
18. Izushi, K., Tasaka, K., Immunopharmacology 18, 177 (1989)
19. Aridor, M., Traub, L. M., Sagi-Eisenberg, R., J. Cell Biol. 111, 909 (1990)
20. Gat-Yablonski, G., Sagi-Eisenberg, R., Biochem. J. 270, 679 (1990)
21. Ozawa, K., Yamada, K., Kazanietz, M. G. et al., J. Biol. Chem. 268, 2280 (1993)
22. Kurosawa, M., Okayama, Y., Kobayashi, S., Ann. Allergy 63, 231 (1989)
23. Gilfillan, A. M., Wiggan, G. A., Welton, A. F., Agents Actions 30, 418 (1990)
24. Nagao, S., Nagata, K., Kohmura, Y. et al., Biochem. Biophys. Res. Commun. 142, 645 (1987)
25. Toyoda, Y., Igarashi, A., Yamada, M. et al., Clin. Rep. 29, 907 (1995)